Heterocycles an International Journal for Reviews and Communications in Heterocyclic Chemistry 2001: Vol 54 Index

29 Pages·2001·5.1 MB·English

HETEROCYCLES, Vol. 54, No. 2, 2001
Author Index Azaheptafulvenes and 6-Amino-1-azafulvenes. 209
Volume 54, 2001 Asakawa, Yoshinori.
Biotransformation of Terpenoids from the Crude Drugs
and Animal Origin by Microorganisms. 529
Asakawa, Yoshinori.
Sesquiterpene Lactones and Acetogenin Lactones from
the Hepaticae and Chemosystematics of the Liverworts
Frullania, Plagiochila and Porella. 1057
A Asao, Toyonobu.
Reaction of 2-Aminoazulenes with Aldehydes. One Pot
Abe, Hitoshi. Synthesis of Diazuleno[2,1-b:1,2-e]pyridines. 667
Revision of the Structure of a New Coumarin Isolated Aso, Yoshio.
from Artemisia carviforia Wall. 319 Bis(ethylenethio)tetraselenafulvalene and Related Hybrid
Abe, Noritaka. Diselenadithiafulvalenes as Novel Electron Donors
Reductive Cyclization of 8-(2-Nitrophenyl)-1-azaazulene Forming Highly Conductive Complexes with 7,7,8,8-
Derivatives; Formation of 6a,7-Diazanaphth{3,2, 1-col- Tetracyanoquinodimethane. 225
azulene and 7H-1,7-Diazaindeno[1,2-e]azulene Systems,
a New DNA Intercalater. 329
Aikawa, Kohsuke.
Lewis Acid Catalysis of Second-Generation Metallosalen B
Complexes: An Explanation for Stereochemistry of
Asymmetric Hetero Diels-Alder Reaction. 395 Bando, Masahiko.
Akasaka, Takeshi. An Efficient Synthesis of Optical Isomers of Vasopressin
Photoinduced Electron-Transfer Reactions between Cen Vo Receptor Antagonist OPC-41061 by Lipase-catalyzed
and Cyclic Disiliranes (c-RoSi-X-SiRo; X=SiRo, CHa, O, Enantioselective Transesterification. 131
Bibart, Richard Todd.
NPh, S). 777
Resolution and Absolute Configurational Assignments to
Alvarez, Miriam.
1-Oxa- and 1-Thia-6-ketospiro[4.4]nonany! Platforms.
Resolution and Absolute Configurational Assignments to
49
1-Oxa- and 1-Thia-6-ketospiro[4.4]nonanyl Platforms.
Bickelhaupt, Friedrich.
49
3-Aza[5]metacyclophanes: Synthesis and Reactions
Amano, Tetsuya.
799
Synthesis and Biological Evaluation of Water Soluble
Bouaziz, Zouhair.
Taxoids Bearing Sugar Moieties. 561
Cycloadditions of a,B-Unsaturated N,N-Dimethylhydra-
Ando, Akira.
zones. A Diels-Alder Strategy for the Building of Aza-
Synthesis of a-(Trifluoromethy!)pyrrolidines by Cycliza-
Hetero Rings. 1095
tion of N-Tosyl-a-(trifluoromethyl)homoallylamine Deriva-
Button, Martin A. C.
tives. 589
Xanthate Mediated Generation of the Benzotriazol-1-
Ando, Masayoshi.
ylmethy! Radical and Its Subsequent Addition to a
Two Taxoids from Taxus cuspidata as Modulators of
Variety of Olefins. 301
Multidrag Resistant Tumor Cells. 999
Aoyagi, Taiyo.
A Molecule Detection Sensor of Modified Cyclodextrin
Based on Guest-responsive Intramolecular Fluorescence
Cc
Quenching. 597
Aoyama, Kinuyo.
Chong, Hyun-Soon.
1,3-Dipolar Cycloaddition of 1-Phenylpropa-1,2-diene
Synthesis and Alkali Metal Picrate Extraction Studies of
with Pyridinium Dicyanomethylides: 1-Phenylpropa-1 ,2-
an Unusual Cage-functionalized Cryptand. 151
diene as a Synthetic Equivalent of 1-Phenyipropyne.
Chou, Chuan-Hung.
611
Photochemistry of Pyrazino- and Quinoxalino-fused
Aoyama, Toyohiko.
Naphthobarrelenes. 61
Cycloaddition Reactions of Trimethylsilylketene with 8-
HETEROCYCLES, Vol. 54, No. 2, 2001
Esumi, Tomoyuki.
Concise Synthesis of (3A,4S)-3-Hydroxy-4-methyl-+
D
butyrolactone. 69
Daich, Adam.
Azepine and [1,3]Oxazepine Fused Ring Construction
through a Cationic Cyclization: An N-Acyliminium lon
Trapping of an Oxygen Atom or Olefin. 275
D'Auria, Maurizio.
Fabris, Fabrizio.
Photochemical Dimerization in Solution of Heterocyclic Resolution and Absolute Configurational Assignments to
Substituted Alkenes Bearing an Electron Withdrawing 1-Oxa- and 1-Thia-6-ketospiro[4.4]nonanyl Platforms.
Group. 475 49
Decroix, Bernard.
Fillion, Houda.
Azepine and [1,3]Oxazepine Fused Ring Construction
Cycloadditions of a,B-Unsaturated N,N-Dimethylhydra-
through a Cationic Cyclization: An N-Acyliminium lon
zones. A Diels-Alder Strategy for the Building of Aza-
Trapping of an Oxygen Atom or Olefin. 275
Hetero Rings. 1095
de Kanter, Franciscus J. J.
Fujii, Hiroyuki.
3-Aza[5]metacyclophanes: Synthesis and Reactions.
Reductive Cyclization of 8-(2-Nitrophenyl)-1-azaazulene
799
Derivatives; Formation of 6a,7-Diazanaphth[31,-c2o,] -
Denisenko, Sergey N.
azulene and 7H-1,7-Diazaindeno[1,2-e]azulene Systems,
Xanthate Mediated Generation of the Benzotriazol-1-
a New DNA Intercalater. 329
ylmethy! Radical and Its Subsequent Addition to a
Fujii, Kazushige.
Variety of Olefins. 301
Synthesis of 2,5-Disubstituted Tetrahydrofurans Cata-
de Rijke, Marianne.
lyzed by Palladium(0). 419
3-Aza[5]metacyclophanes: Synthesis and Reactions.
Fujii, Masako.
799
Revision of the Structure of a New Coumarin Isolated
de Wolf, Willem H.
from Artemisia carviforia Wall. 319
3-Aza[5]metacyclophanes: Synthesis and Reactions.
Fujimori, Kunihide.
799
Preparation, Structure, and Properties of 1,3-Bis(1,4-
dithiafulven-6-yl)azulenes. 377
Fujioka, Shozo.
Efficient and Stereoselective B-Epoxidation of the 16(17)-
Double Bond of Gibberellic Acid Derivatives with an Acyl-
Egberts, Arne. peroxy Radical Generated by Irradiation of a-Diketones
3-Aza[5]metacyclophanes: Synthesis and Reactions. and Oxygen. 81
799 Fujisawa, Naoki.
El Bialy, Serry A. A. Preparation, Structure, and Properties of 1,3-Bis(1,4-
5-endo-trig Radical Cyclization of N- Benzyl-2-halo-N-(6- dithiafulven-6-yl)azulenes. 377
oxo-1-cyclohexen-1-yl)acetamides. 1021 Fujita, Kasuke.
Ei Hassane, Lahiou. Synthesis of a,a'-Asymmetric Nitroxide Radicals by C- or
Sesquiterpene Lactones and Acetogenin Lactones from O-Acylation of Radical-Enolate Intermediates Generated
the Hepaticae and Chemosystematics of the Liverworts by Reduction of Homoallylic Nitro Enones with Samarium
Frullania, Plagiochila and Porella. 1057 (Il) lodide. 217
Emoto, Yoshitaka. Fujitsuka, Mamoru.
Photochemistry of Heterocyclic Cage Compound: Photo- Photoinduced Electron-Transfer Reactions between Cgo
reaction of 2,7-Dihydroazepine to Give 2,3-Dihydroaze-
and Cyclic Disiliranes (c-RaSi-X-SiRo; X=SiRo, CHo, O,
pine and Photoreaction of the 2,3-Dihydroazepine to
NPh, S). 777
Form 1,2-Dihydroaniline. 567
Fujiwara, Kenshu.
Enoki, Toshiaki.
Benzyloxymethy!l Group as a Convertible Internal Ligand
Syntheses, Structure and Conducting Properties of Halo-
for La(OTf)3-catalyzed 7-endo Ring-Openig of Hydroxy
genated Ethylenedioxytetrathiafulvalenes. 833
HETEROCYCLES, Vol. 54, No. 2, 2001
Epoxide. 109 3-Aza[5]metacyclophanes: Synthesis and Reactions.
Fukal, Toshio. 799
Structure of Sanggenon O, a Diels-Alder Type Adduct Gruza, Henryk.
Derived from a Chalcone and a Dehydroprenylated Efficient Stereoselective Synthesis of (25,3S,5A)-(+)-
Sanggenon-Type Flavanone from Morus cathayana. Preussin. 581
39
Fukazawa, Yoshimasa.
Intramolecular Complex Formation between Flexible Mo-
lecular Tweezers and Weak Electron Acceptor. 849 H
Fukuta, Atsushi.
Synthesis and Properties of anti6,15-Epithia-183,- Hagino, Yasumichi.
methanobenzo[e][14]annulene-7,14-dione, anti-5,14- A Convenient Determination of Chiral Pteridines; Applica-
Epithia-7,12-methanofu14r ]oan[n3ul,e4ne--e5,] 1[3 - tion of Fluorescence Detected Circular Dichroism (FDCD)
diones, and Their lonic Species. 159 to the Major Pterin from Escherichia coli. 283
Fukuyama, Tohru. Halada, P.
A Practical Route to Quinolines from Anilines. 105 Chemoenzymatic Preparation of Oligoglycosides of Sily-
Fukuyama, Yoshiyasu. bin, the Flavonolignan from Silybum marianum. 901
Total Syntheses of Plagiochins A and D, Macrocyclic Hamada, Masahiro.
Bis(bibenzyls), by Pd(0) Catalyzed Intramolecular Stille- Stereospecific Substitution of 1-(2-Pyridinyl)ethyl Methane-
Kelly Reaction. 259 sulfonate with S- and O-Nucleophiles. 735
Fumoto, Yumiko. Hamada, Yasumasa.
Preparation of Meso-unsubstituted Porphyrins Substituted Synthesis of 2,5-Disubstituted Tetrahydrofurans Cata-
with Mono- and Tetraformy!l and Other Electron-withdraw- lyzed by Palladium(0). 419
ing Groups. 705 Hara, Kenji.
Funaki, Takashl. Syntheses, Structure and Conducting Properties of Halo-
Synthesis of Pyridinocrownophanes Exhibiting High Ag*- genated Ethylenedioxytetrathiafulvalenes. 833
Affinity. 123 Hara, Ko-ji.
Funayama, Shinji. Synthesis and Biological Evaluation of Water Soluble
Quinoline Alkaloids of Orixa japonica 1139 Taxoids Bearing Sugar Moieties. 561
Furukawa, Yoshiro. Hara, Ko-zo.
Synthesis of N-Boc-3-amino-1,2-epoxy-4-phenylbutane Synthesis and Biological Evaluation of Water Soluble
Taxoids Bearing Sugar Moieties. 561
from (3S)-Hydroxy-y-butyrolactone by Means of the
Hara, Osamu.
Hofmann Rearrangement. 77
Synthesis of 2,5-Disubstituted Tetrahydrofurans Cata-
Furuta, Shinji.
lyzed by Palladium(0). 419
Synthesis and Properties of ant+6,15-Epithia-183,-
Harada, Kazuho.
methanobenzo[e][14]annulene-7,14-dione, antr5,14-
Epithia-7,12-methanofu14 rJoan[n3ul,en4e--5e,] 1[3 - Formation of Trisubstituted y-Butyrolactones by Novel
diones, and Their lonic Species. 159 Ring Transformation of 2-lsoxazoline-2-oxides. 1033
Harayama, Takashi.
Revision of the Structure of a New Coumarin Isolated
from Artemisia carviforia Wall. 319
G Hariprakasha, H. K.
Synthesis and Alkali Metal Picrate Extraction Studies of
GaZak, R. an Unusual Cage-functionalized Cryptand. 151
Chemoenzymatic Preparation of Oligoglycosides of Sily- Hashimoto, Kimiko.
bin, the Flavonolignan from Silybum marianum. 901 Synthesis of Alternariolide Analogs for Photoaffinity-
Gebert, Andreas. Labeling. 917
Synthesis of 1,3-Thiazolidines from Aromatic Thio- Hashimoto, Shunichi.
Enantiocontrol in Tandem Allylic Sulfonium Vlide Genera-
ketones and N-Benzylidene a-Amino Acid Esters via
tion and [2,3] Sigmatropic Rearrangement Catalyzed by
1,3-Dipolar Cycloaddition of Azomethine Ylides. 691
Chiral Dirhodium(Il) Complexes. 623
Gret, Norbert.
Hashimoto, Toshihiro.
HETEROCYCLES, Vol. 54, No. 2, 2001
Biotransformation of Terpenoids from the Crude Drugs Hirao, Ken-ichi.
and Animal Origin by Microorganisms. 529 Synthesis of a,a'-Asymmetric Nitroxide Radicals by C- or
Hashimoto, Toshihiro. O-Acylation of Radical-Enolate Intermediates Generated
Sesquiterpene Lactones and Acetogenin Lactones from by Reduction of Homoallylic Nitro Enones with Samarium
the Hepaticae and Chemosystematics of the Liverworts
(Il) lodide. 217
Frullania, Plagiochila and Porelia. 1057
Hirata, Naonori.
Hatakeyama, Susumi. Two Taxoids from Taxus cuspidata as Modulators of
Concise Synthesis of (3A,4S)-3-Hydroxy-4-methyl-y~- Multidrag Resistant Tumor Cells. 999
butyrolactone. 69 Hirol, Kunio.
Hatanaka, Minoru. Asymmetric Pauson-Khand Reactions of Chiral Sulfin-
Application of Phthalimidine Synthesis with Use of 1,2,3- amides: Asymmetric Synthesis of 3-Azabicyclo[3.3.0]oct-
1H-Benzotriazole and 2-Mercaptoethanol as Dual Syn- 5-en-7-one Derivatives. 73
thetic Auxiliaries. 2. Effective Synthesis of Phthalimidines Hirose, Katutoshi.
Possessing Bulky Group at 2-Position. 635 Two Taxoids from Taxus cuspidata as Modulators of
Hatsui, Toshihide. Multidrag Resistant Tumor Cells. 999
Intramolecular Photocycloaddition of 2-Cycloalkenyl-1,3- Hirotani, Seiko.
dioxin-4-one. Stereoselective Synthesis of cis-Eudes- Formation of Trisubstituted yButyrolactones by Novel
mane-4,11-diols. 765
Ring Transformation of 2-lsoxazoline-2-oxides. 1033
Hayashi, Naoto.
Hirowatari, Katsuji.
1,3-Dipolar Cycloaddition of 1-Phenylpropa-1,2-diene 1,3-Dipolar Cycloadditions of 3-Bromo-1,5- and 3-Bromo-
with Pyridinium Dicyanomethylides: 1-Phenylpropa-,12- 1,7-azulenequinones with Diazomethane, DiphenyInitril-
diene as a Synthetic Equivalent of 1-Phenylpropyne.
imine, and Benzonitrile Oxide. 291
611 Holzer, Wolfgang.
Heimgartner, Heinz.
Synthesis of Azanaphthoquinone Annelated Pyrroles.
Synthesis of 1,3-Thiazolidines from Aromatic Thio-
111
ketones and N-Benzylidene a-Amino Acid Esters via Honda, Konomi.
1,3-Dipolar Cycloaddition of Azomethine Ylides. 691 Synthesis of 2,3,4,5-Tetrahydro-1H-2-benzazepines via
Higashiyama, Kimio. Pummerer-Type Cyclization of N-Arylmethyl-N-(3-phenyl-
Photosubstitution Reaction of Cyanoaromatics with Ali- sulfinylpropyl)formamides. 967
phatic Amides. 1027 Honda, Toshio.
Hinoue, Kazumasa. Diastereoselective Addition of Organometallic Reagents
Synthesis of N-Boc-3-amino-1,2-epoxy-4-phenylbutane to (A)-2,3-lsopropylidenedioxy-1 -(2-fury!)-1-propanone
from (3S)-Hydroxy-y-butyrolactone by Means of the Yielding Chiral Tertiary Furyl Carbinols. 341
Hofmann Rearrangement. 77 Hong, Young-Taek.
Hirama, Masahiro. Palladium-catalyzed Carbonylative Coupling of Hyper-
Contributions of Professor Sho Ito in Organic Chemistry. valent lodonium Salts with Amidoximes: Synthesis of
» Oxadiazoles. 985
/
Hirama, Masahiro. Hongo, Hiroshi.
Convergent Strategy for Synthesizing Polycyclic Ether Synthesis of New Chiral Catalysts, 2-Azanorbornyloxa-
Marine Toxins: Synthesis of the ABCDE Ring Fragment zolidines, for Enantioselective Addition of Diethylzinc to
of Ciguatoxin CTX3C. 93 Aldehydes. 411
Hirano, Etsushi. Hori, Mikio.
Application of Phthalimidine Synthesis with Use of 1,2,3- Synthesis and Properties of Novel Medium-sized Hetero-
1H-Benzotriazole and 2-Mercaptoethanol as Dual Syn- cyclic Compounds Containing Two Sulfur Atoms in the
thetic Auxiliaries. 2. Effective Synthesis of Phthalimidines Ring and Synthetic Approaches to Conjugated Cyclic
Possessing Bulky Group at 2-Position. 635 Disulfonium Ylides. 139
Hirano, Yukiyasu. Horiguchi, Yoshie.
Synthesis and Properties of anti-6,15-Epithia-183,- Synthesis of 2,3,4,5-Tetrahydro-1H-2-benzazepines via
methanobenzo[e][14]annuiene-7,14-dione, anti5,14- Pummerer-Type Cyclization of N-Arylmethyl-N-(3-phenyl-
Epithia-7,12-methanofu14 r]oan[n3ul,e4ne--e5,] 1[3 - sulfinylpropyl)formamides. 967
diones, and Their lonic Species. 159 Hoshino, Mikio.
HETEROCYCLES, Vol. 54, No. 2, 2001
Efficient and Stereoselective B-Epoxidation of the 16(17)- phenanthridine from 2-Phenyl-1-tetralone. 433
Double Bond of Gibberellic Acid Derivatives with an Acyl- Ishikawa, Tsutomu.
peroxy Radical Generated by Irradiation of a-Diketones Triphosgene: A Versatile Reagent for Bischler-
Napieralski Reaction. 437
and Oxygen. 81
Isobe, Minoru.
Synthesis of Ciguatoxin (2S,5A)-ABC Segment. 789
Ito, Osamu.
Photoinduced Electron-Transfer Reactions between Ceo
and Cyclic Disiliranes (c-RoSi-X-SiRo; X=SiRo, CHo, O,
ichinose, Hiroshi. NPh, S). 777
A Convenient Determination of Chiral Pteridines; Applica- Ito, Shunji.
tion of Fluorescence Detected Circular Dichroism (FDCD) Reaction of 2-Aminoazulenes with Aldehydes. One Pot
to the Major Pterin from Escherichia coli. 283 Synthesis of Diazuleno[2,1-b:1,2-e]pyridines. 667
Ihara, Masataka. Ito, Shunji.
Synthesis of a Novel Artemisinin Analogue Having An Efficient Preparation of 2H-Cycloheptafbjfuran-2-
Potent Antimalarial Activity. 607 ones. 679
Ikeda, Masazumi. Ito, Suketaka.
Regioselective Synthesis of Bridged Azabicyclic Com- Preparation of New Nitrogen-bridged Heterocycles. 50.
pounds Using Radical Translocation/Cyclization Reac- Syntheses of Some Heterocyclic Compounds Starting
tions of 4-Alkynyl-1-(o-iodobenzoyl)piperidines. 747 from Pyridinium 1-(Ethoxycarbonylacetyl)methylides.
Ikeda, Masazumi. 185
5-endo-trig Radical Cyclization of N- Benzy|l-2-halo-N-(6- Ito, Suketaka.
oxo-1-cyclohexen-1-yl)acetamides. 1021 Thermolysis of Ethoxycarbony|[2-phenyl-2-(phenylsulfo-
ikem, Yukio. nylhydrazono)ethy!]methylenetriphenylphosphoranes.
1,3-Dipolar Cycloaddition of 1-Phenyipropa-1,2-diene Formation of Substituted Pyridazinones. 237
with Pyridinium Dicyanomethylides: 1-Phenylpropa-1 ,2- Iwabuchi, Yoshiharu.
diene as a Synthetic Equivalent of 1-Phenylpropyne. Concise Synthesis of (3A,4S)-3-Hydroxy-4-methyl-+
611
butyrolactone. 69
ikemoto, Isao.
lwasa, Kazuto.
Syntheses, Structure and Conducting Properties of Halo-
Synthesis of New Chiral Catalysts, 2-Azanorbornyloxa-
genated Ethylenedioxytetrathiafulvalenes. 833 zolidines, for Enantioselective Addition of Diethylzinc to
Ikemoto, Kazuhisa. Aldehydes. 411
A Convenient Determination of Chiral Pteridines; Applica-
Iwatani, Wakao.
tion of Fluorescence Detected Circular Dichroism (FDCD) Synthesis and Biological Evaluation of Water Soluble
to the Major Pterin from Escherichia coli. 283 Taxoids Bearing Sugar Moieties. 561
Imafuku, Kimiakl.
lyoda, Masahiko.
New Synthetic Approach to Azuleno[1,2-c]pyrroles and Syntheses, Structure and Conducting Properties of Halo-
Conversion to Benz[alazulenes. 647
genated Ethylenedioxytetrathiafulvalenes. 833
Imagawa, Hiroshi.
Intramolecular Oxymercuration of 4-Hexen-1-ols: Kinetic
vs. Thermodynamic Products Regulated by Mercuric
Salts. 629
Inokuma, Selichi.
Synthesis of Pyridinocrownophanes Exhibiting High Ag*- Jigami, Tetsuya.
Affinity. 123 Bis(ethylenethio)tetraselenafulvalene and Related Hybrid
Irie, Ryo. Diselenadithiafulvalenes as Novel Electron Donors
Lewis Acid Catalysis of Second-Generation Metallosalen Forming Highly Conductive Complexes with 7,7,8,8-
Complexes: An Explanation for Stereochemistry of Tetracyanoquinodimethane. 225
Asymmetric Hetero Diels-Alder Reaction. 395 Jonoshita, Shuichi.
Ishikawa, Tsutomu. Synthesis of a-(Trifluoromethy!)pyrrolidines by Cycliza-
Alternative Synthesis of B/C-cis Hexahydrobenzo[c]-
tion of N-Tosyl-c-(trifluoromethyl)homoallylamine Deriva-
HETEROCYCLES, Voi. 54, No. 2, 2001
tives. 589 1H-Benzotriazole and 2-Mercaptoethanol as Dual Syn-
Jurczak, Janusz. thetic Auxiliaries. 2. Effective Synthesis of Phthalimidines
Efficient Stereoselective Synthesis of (2S,3S,5A)-(+)- Possessing Bulky Group at 2-Position. 635
Preussin. 581 Kang, Suk-Ku.
Palladium-catalyzed Carbonylative Coupling of Hyper-
valent lodonium Salts with Amidoximes: Synthesis of
Oxadiazoles. 985
K Kashima, Choji.
Preparation of B-Substituted y-Keto Esters by the
Kageura, Yuichi. Grignard Reaction on N-Acylpyrazoles. 309
Reductive Cyclization of 8-(2-Nitrophenyl)-1-azaazulene Kashima, Terumi.
Derivatives; Formation of 6a,7-Diazanaphth{31,-c2a,}- Intramolecular Oxymercuration of 4-Hexen-1-ols: Kinetic
azulene and 7H-1,7-Diazaindeno[1,2-e]azulene Systems, vs. Thermodynamic Products Regulated by Mercuric
a New DNA Intercalater. 329 Salts. 629
Kaji, Eisuke. Katagiri, Ruriko.
Formation of Trisubstituted y-Butyrolactones by Novel Synthesis of a Novel Artemisinin Analogue Having
Ring Transformation of 2-Ilsoxazoline-2-oxides. 1033 Potent Antimalarial Activity. 607
Kajikawa, Shougo. Kataoka, Masahiro.
Convenient Construction of Hexahydrobenzo[b]furan Solvent Effects on Relative Stability of Meridine and Its
Skeleton Containing Heteroatoms. Choice of Mn(IIl)- and Tautomer: MO Calculations. 55
Ce(IV)-based Radical Cyclization. 171 Kataoka, Tadashi.
Kajioka, Takanori. Synthesis and Properties of Novel Medium-sized Hetero-
Synthesis and Properties of ant#6,15-Epithia-813,- cyclic Compounds Containing Two Sulfur Atoms in the
methanobenzo[e][14]annulene-7,14-dione, anti-5,14- Ring and Synthetic Approaches to Conjugated Cyclic
Epithia-7,12-methanofu14 r]oan[n3ul,en4e--5e,] 1[3 - Disulfonium Ylides. 139
diones, and Their lonic Species. 159 Kato, Masako.
Kakehl, Akikazu. Optical Resolution of 2-Azabicyclo[2.2.1]hept-5-en-3-one
Preparation of New Nitrogen-bridged Heterocycles. 50. by Inclusion Complexation with Brucine. 405
Syntheses of Some Heterocyclic Compounds Starting Kato, Masako.
from Pyridinium 1-(Ethoxycarbonylacetyl)methylides. Synthesis, Structure and Spectroscopic Characteristics of
185 2'-Boryl-4"-dimethylaminochalcones. Effect of an Intra-
Kakehi, Akikazu. molecular Boron-Oxygen Coordinate Bond to the Conju-
Thermolysis of Ethoxycarbony|[2-phenyl-2-(pheny|sulfo- gated System. 929
nylhydrazono)ethy!]methylenetriphenylphosphoranes. Kato, Nobuo.
Formation of Substituted Pyridazinones. 237 1,3-Dipolar Cycloadditions of 3-Bromo-1,5- and 3-Bromo-
Kakehi, Akikazu. 1,7-azulenequinones with Diazomethane, Diphenyinitril-
Reductive Cyclization of 8-(2-Nitropheny!)-1-azaazulene imine, and Benzonitrile Oxide. 291
Derivatives; Formation of 6a,7-Diazanaphth{32,, 1-ca}- Kato, Takehiro.
azulene and 7H-1,7-Diazaindeno[1,2-e]azulene Systems, Syntheses, Structure and Conducting Properties of Halo-
a New DNA Intercalater. 329 genated Ethylenedioxytetrathiafulvalenes. 833
Kakehl, Akikazu. Katoh, Tadashi.
1,3-Dipolar Cycloaddition of 1-Phenylpropa-1,2-diene An Efficient and Expeditious Synthesis of a Novel 5H-
with Pyridinium Dicyanomethylides: 1-Phenylpropa-,12 - Naphth[1',2':5,6][1,4]oxazino[2,3-b]quinoxalin-5-one and
diene as a Synthetic Equivalent of 1-Phenylpropyne. Its Unique Inhibitory Activity against a Panel of Human
611 Cancer Cell Lines. 619
Kako, Masahiro. Katritzky, Alan R.
Photoinduced Electron-Transfer Reactions between Cgg Xanthate Mediated Generation of the Benzotriazol-1-
and Cyclic Disiliranes (c-RoSi-X-SiRo; X=SiRo, CHp, O, ylmethy! Radical and Its Subsequent Addition to a
Variety of Olefins. 301
NPh, S). 777
Katsuki, Tsutomu.
Kamimura, Shigeki.
Lewis Acid Catalysis of Second-Generation Metallosalen
Application of Phthalimidine Synthesis with Use of 1,2,3-
Complexes: An Explanation for Stereochemistry of
HETEROCYCLES, Vol. 54, No. 2, 2001
Asymmetric Hetero Diels-Alder Reaction. 395 Synthesis of 2,3,4,5-Tetrahydro-1 H-2-benzazepines via
Katsumura, Shigeo. Pummerer-Type Cyclization of N-Aryimethy!-N-(3-phenyl-
Synthesis of N-Boc-3-amino-1,2-epoxy-4-phenylibutane sulfinylpropy!l)formamides. 967
from (3S)-Hydroxy-y-butyrolactone by Means of the Kishi, Akinobu.
Hofmann Rearrangement. 77 Chemical Constituents of Two Oriental Orchids, Calanthe
Katsuno, Keiko. discolor and C. liukiuensis: Precursor Indole Glycoside of
Revision of the Structure of a New Coumarin Isolated Tryptanthrin and Indirubin. 957
from Artemisia carviforia Wall. 319 Kishimoto, Yaeko.
Katsuyama, Isamu. Quinolone Analogues 3. Synthesis of 1,3-Dialkyl-4-oxo-
The Identification, Mechanism, and Improved Synthesis 1,4-dihydropyridazino[3,4-b]quinoxalines. 359
of a New and Unique Heterocyclic System with a Fused Kitagaki, Shinji.
Imidazole Ring. 721 Enantiocontrol in Tandem Allylic Sulfonium Ylide Genera-
tion and [2,3] Sigmatropic Rearrangement Catalyzed by
Kawakami, Teruki.
Chiral Dirhodium(Il) Complexes. 623
Application of Phthalimidine Synthesis with Use of 1,2,3-
1H-Benzotriazole and 2-Mercaptoethanol as Dual Syn- Kitahara, Takeshi.
Synthesis of Brevicompanines, Plant Growth Regulators.
thetic Auxiliaries. 2. Effective Synthesis of Phthalimidines
727
Possessing Bulky Group at 2-Position. 635
Kitajima, Hidehiko.
Kawakami, Yusuke.
Application of Phthalimidine Synthesis with Use of 1,2,3-
Substitution vs. Addition. Regioselective Electrobromi-
1H-Benzotriazole and 2-Mercaptoethanol as Dual Syn-
nation of Benzofuran. 825
thetic Auxiliaries. 2. Effective Synthesis of Phthalimidines
Kawano, Yoshikazu.
Possessing Bulky Group at 2-Position. 635
An Efficient Synthesis of Optical Isomers of Vasopressin
Kitano, Kazuyoshi.
Vo Receptor Antagonist OPC-41061 by Lipase-catalyzed
An Efficient Synthesis of Optical Isomers of Vasopressin
Enantioselective Transesterification. 131
Vo Receptor Antagonist OPC-41061 by Lipase-catalyzed
Khalil, Ashraf A.
Enantioselective Transesterification. 131
The Identification, Mechanism, and Improved Synthesis
Kobayashi, Kaoru.
of a New and Unique Heterocyclic System with a Fused
Photoinduced Electron-Transfer Reactions between Ceo
Imidazole Ring. 721
Kido, Masaru. and Cyclic Disiliranes (c-RoSi-X-SiRo; X=SiRo, CHa, O,
An Efficient Synthesis of Optical lsomers of Vasopressin NPh, S). 777
Vo Receptor Antagonist OPC-41061 by Lipase-catalyzed Koéevar, Marijan.
Enantioselective Transesterification. 131 4-Acylhydrazinomethylene-2-phenyloxazol-5(4H)-ones as
Kim, Eun Young. Acylating Agents: Synthesis of Salicylanilides and 1,2,4-
Synthesis of a Macroheterocyclic Compound through Triazolo[4,3-b]pyridazines. 1011
Photodecarboxylation of Potassium w-Phthalimidoalkyn- Kodama, Mitsuaki.
Total Syntheses of Plagiochins A and D, Macrocyclic
oate. 1049
Bis(bibenzyls), by Pd(0) Catalyzed Intramolecular Stille-
Kim, Ho Sik.
Kelly Reaction. 259
Quinolone Analogues 3. Synthesis of 1,3-Dialkyl-4-oxo-
Kodani, Mie.
1,4-dihydropyridazino[3,4-b]quinoxalines. 359
Bis(ethylenethio)tetraselenafulvalene and Related Hybrid
Kim, Hye-Sook.
Diselenadithiafulvalenes as Novel Electron Donors
Synthesis of a Novel Artemisinin Analogue Having
Forming Highly Conductive Complexes with 7,7,8,8-
Potent Antimalarial Activity. 607
Tetracyanoquinodimethane. 225
Kimino, Mako.
Kokubo, Susumu.
Application of Phthalimidine Synthesis with Use of 1,2,3-
Haterumaimides A-E, Five New Dichlorolissoclimide-Type
1H-Benzotriazole and 2-Mercaptoethanol as Dual Syn-
Diterpenoids from an Ascidian, Lissoclinum Sp. 1039
thetic Auxiliaries. 2. Effective Synthesis of Phthalimidines
Konakahara, Takeo.
Possessing Bulky Group at 2-Position. 635
Reductive Cyclization of 8-(2-Nitrophenyl)-1-azaazulene
Kimura, Koichl.
Derivatives; Formation of 6a,7-Diazanaphth[3,2,1-co]-
Synthesis of Pyridinocrownophanes Exhibiting High Agt-
azulene and 7H-1,7-Diazaindeno[1,2-e]azulene Systems,
Affinity. 123
a New DNA Intercalater. 329
Kimura, Tomoko.
Kosugi, Katsuhiko.
HETEROCYCLES, Vol. 54, No. 2, 2001
Two Taxoids from Taxus cuspidata as Modulators of Kurasawa, Yoshihisa.
Multidrag Resistant Tumor Cells. 999 Quinolone Analogues 3. Synthesis of 1,3-Dialkyi-4-oxo-
Koulourl, Alexandra. 1,4-dihydropyridazino[3,4-b]quinoxalines. 359
Synthesis of Azanaphthoquinone Annelated Pyrroles. Kurebayashi, Hirotaka.
111 Intramolecular Complex Formation between Flexible Mo-
Kozawa, Kozo. lecular Tweezers and Weak Electron Acceptor. 849
Synthesis and Properties of Benzimidazole and Naph- Kurihara, Teruo.
thoimidazole Derivatives of Perylenedicarboximide. Syntheses and Properties of Tetraazaazulenocoronands
757 and Octaazaazulenocryptand. 87
Krasinski, Antoni. Kuroboshi, Manabu.
Efficient Stereoselective Synthesis of (2S,3S,5A)-(+)- Substitution vs. Addition. Regioselective Electrobromi-
Preussin. 581 nation of Benzofuran. 825
Krassnig, Roland. Kuroda, Shigeyasu.
Synthesis and Pharmacological Evaluation of 18,19- Synthesis and Properties of anti-6,15-Epithia-183,-
Dehydrobuprenorphine. 989 methanobenzo[e][14]annulene-7,14-dione, anti-5,14-
Kratzel, Martin. Epithia-7, 12-methanofuro[3,4-e][1 4Jannulene-5,13-
Synthesis of Azanaphthoquinone Annelated Pyrroles. diones, and Their lonic Species. 159
111 Kurosawa, Kazu.
K¥en, V. Convenient Construction of Hexahydrobenzo[b]furan
Chemoenzymatic Preparation of Oligoglycosides of Sily- Skeleton Containing Heteroatoms. Choice of Mni(Ill)- and
bin, the Flavonolignan from Silybum marianum. 901 Ce(IV)-based Radical Cyclization. 171
Krenn, Petra. Kusumi, Takenori.
Synthesis of Azanaphthoquinone Annelated Pyrroles. Carbon-13 Spin-Lattice Relaxation Time (7}) for Assign-
111 ment of Brominated Carbons. 577
Kubisch, J.
Kuwatanl, Yoshiyuki.
Chemoenzymatic Preparation of Oligoglycosides of Sily- Syntheses, Structure and Conducting Properties of Halo-
bin, the Flavonolignan from Silybum marianum. 901 genated Ethylenedioxytetrathiafulvalenes. 833
Kubo, Hajime.
Kyogoku, Mayumi.
Photosubstitution Reaction of Cyanoaromatics with Ali- Synthesis and Properties of anti-6,15-Epithia-183,-
phatic Amides. 1027 methanobenzo[e][14]annulene-7,14-dione, anti-5,14-
Kubo, Kanji.
Epithia-7,12-methanofuro[3,4-e][14]annulene-5,13-
1,3-Dipolar Cycloadditions of 3-Bromo-1,5- and 3-Bromo-
diones, and Their lonic Species. 159
1,7-azulenequinones with Diazomethane, DiphenyInitril-
imine, and Benzonitrile Oxide. 291
Kubo, Kanji.
Synthesis and Mercurophilic Properties of Acyclic and
Thiolariat Ethers Having a Tropone Pendant. 351
Kudo, Masao.
Lanter, James C.
An Efficient Preparation of 2H-Cyclohepta[b]furan-2- Resolution and Absolute Configurational Assignments to
ones. 679
1-Oxa- and 1-Thia-6-ketospiro[4.4]nonanyl Platforms.
Kumadaki, Itsumaro.
49
Synthesis of a-(Trifluoromethy!)pyrrolidines by Cycliza- Lattanzi, Roberta.
tion of N-Tosyl-a-(trifluoromethy!)homoallylamine Deriva- Synthesis and Pharmacological Evaluation of 18,19-
tives. 589 Dehydrobuprenorphine. 989
Kumazawa, Keita. Li, Ka.
Formation of Trisubstituted y-Butyrolactones by Novel Intramolecular Photocycloaddition of 2-Cycloalkenyl-1,3-
Ring Transformation of 2-lsoxazoline-2-oxides. 1033 dioxin-4-one. Stereoselective Synthesis of cis-Eudes-
Kuramoto, Shin-ya. mane-4,11-diols. 765
Synthesis and Properties of anti#6,15-Epithia-183,- Li, Yanzhong.
methanobenzo[e][14]annulene-7,14-dione, anti5,14- Preparation of Benzoheterocycles Containing Group 14
Epithia-7,12-methanofuro[3,4-e][14]annulene-153,- Elements Using Zirconacyclopentadienes. 943
diones, and Their lonic Species. 159 Liao, Chun-Chen.
HETEROCYCLES, Vol. 54, No. 2, 2001
Photochemistry of Pyrazino- and Quinoxalino-fused discolor and C. liukiuvensis: Precursor Indole Glycoside of
Naphthobarrelenes. 61 Tryptanthrin and Indirubin. 957
Linden, Anthony. Matsuda, Noriko.
Synthesis of 1,3-Thiazolidines from Aromatic Thio- Preparation of Azulenequinones Containing Azacrown
ketones and N-Benzylidene a-Amino Acid Esters via Moieties and the Singular Complexation of Sodium or
1,3-Dipolar Cycloaddition of Azomethine Ylides. 691 Potassium Cation by 3,5-Bis(aza-18-crown-6)-1,7-azu-
lenequinone in Solution. 439
Matsumoto, Kiyoshi.
1,3-Dipolar Cycloaddition of 1-Phenylpropa-1,2-diene
with Pyridinium Dicyanomethylides: 1-Phenylpropa-1,2-
diene as a Synthetic Equivalent of 1-Phenylpropyne.
Maeda, Kenji. 611
Convergent Strategy for Synthesizing Polycyclic Ether Matsumoto, Koichiro.
Marine Toxins: Synthesis of the ABCDE Ring Fragment Chiral Ketone-catalyzed Asymmetric Epoxidation of Stil-
of Ciguatoxin CTX3C. 93 bene with Oxone®. 615
Maeda, Yutaka. Matsumura, Koji.
Photoinduced Electron-Transfer Reactions between Ceo Synthesis of Brevicompanines, Plant Growth Regulators.
and Cyclic Disiliranes (c-RoSi-X-SiRo; X=SiRo, CHa, O, 727
NPh, S). 777 Matsuyama, Haruo.
Makosza, Mieczystaw. Syntheses, Structure and Conducting Properties of Halo-
Nucleophilic Aromatic Substitution of Hydrogen as a Tool genated Ethylenedioxytetrathiafulvalenes. 833
for the Synthesis of Indole and Quinoline Derivatives. Mihara, Jun.
445 Lewis Acid Catalysis of Second-Generation Metallosalen
Mamounl, Aicha. Complexes: An Explanation for Stereochemistry of
Azepine and [1,3]Oxazepine Fused Ring Construction Asymmetric Hetero Diels-Alder Reaction. 395
through a Cationic Cyclization: An N-Acyliminium lon Mikami, Koichi.
Trapping of an Oxygen Atom or Olefin. 275 Diastereocontrol in the Reaction of (A)- 2,2-Dimethyl-4-
Mandai, Tadakatsu. acyl-1,3-dioxolanes with Alkylmetals: A Facile Entry to
Synthesis and Biological Evaluation of Water Soluble Enantiopure Terpenetriols. 585
Taxoids Bearing Sugar Moieties. 561 Mikata, Yuji.
Marchalin, Stefan. Synthesis, Structure and Spectroscopic Characteristics of
Azepine and [1,3]Oxazepine Fused Ring Construction 2'-Bory!-4"-dimethylaminochalcones. Effect of an Intra-
through a Cationic Cyclization: An N-Acyliminium lon molecular Boron-Oxygen Coordinate Bond to the Conju-
Trapping of an Oxygen Atom or Olefin. 275 gated System. 929
Marchand, Alan P. Mikoshiba, Hisashi.
Synthesis and Alkali Metal Picrate Extraction Studies of Diastereocontrol in the Reaction of (A)- 2,2-Dimethyl-4-
acyl-1,3-dioxolanes with Alkyimetals: A Facile Entry to
an Unusual Cage-functionalized Cryptand. 151
Maruoka, Keiji. Enantiopure Terpenetriols. 585
Facile Conversion of Trialkylsilyl Esters to Alkyl Esters Mikunl, Katsuhiko.
Synthesis and Biological Evaluation of Water Soluble
Mediated by Tetrabutylammonium Fluoride Trihydrate.
593 Taxoids Bearing Sugar Moieties. 561
Maruyama, Megumi. Minami, Hiroyuki.
Convergent Strategy for Synthesizing Polycyclic Ether Total Syntheses of Plagiochins A and D, Macrocyclic
Marine Toxins: Synthesis of the ABCDE Ring Fragment Bis(bibenzyls), by Pd(0) Catalyzed Intramolecular Stille-
of Ciguatoxin CTX3C. 93 Kelly Reaction. 259
Matsubara, Jun. Mitchell, Reginald H.
An Efficient Synthesis of Optical Isomers of Vasopressin [25]Metacyclophanedienes with Furan Bridges. 249
Vo Receptor Antagonist OPC-41061 by Lipase-catalyzed Miyashita, Masaaki.
Enantioselective Transesterification. 131 Short-Step Synthesis of Some Santanolides, Dehydro-
Matsuda, Hisashi. isoerivanin, lsoerivanin, Ludovicin C, and 1a,3a-Di-
Chemical Constituents of Two Oriental Orchids, Calanthe hydroxyarbusculin B by the Use of the Organoselenium
HETEROCYCLES, Vol. 54, No. 2, 2001
Reduction Method of Epoxy Ketones. 865 Benzyloxymethyl Group as a Convertible Internal Ligand
Miyata, Fusae. for La(OTf)3-catalyzed 7-endo Ring-Openig of Hydroxy
An Efficient and Expeditious Synthesis of a Novel 5H- Epoxide. 109
Naphth[1',2':5,6][1,4Joxazino[2,3-b]quinoxalin-5-one and
Morita, Chikanori.
Its Unique Inhibitory Activity against a Panel of Human Synthesis of Alternariolide Analogs for Photoaffinity-
Cancer Cell Lines. 619 Labeling. 917
Miyatake, Ryuta.
Morita, Noboru.
Synthesis and Properties of ant+6,15-Epithia-813,- Reaction of 2-Aminoazulenes with Aldehydes. One Pot
methanobenzo[e][14]annulene-7,14-dione, anti5,14-
Synthesis of Diazuleno[2,1-b:1,2-e]pyridines. 667
Epithia-7,12-methanofu14 r]oan[n3ul,e4ne--5e,] 1[3 - Morita, Noboru.
diones, and Their lonic Species. 159 An Efficient Preparation of 2H-Cyclohepta[b]furan-2-
Miyawakl, Kazuhiro.
ones. 679
Synthesis of Indeno[1,2-b]phenanthrene-Type Hetero-
Morita, Seiji.
cycles by Cycloaromatization of Acyclic Non-conjugated An Efficient Synthesis of Optical Isomers of Vasopressin
Benzotetraynes. 887 Vo Receptor Antagonist OPC-41061 by Lipase-catalyzed
Miyazaki, Akira.
Enantioselective Transesterification. 131
Syntheses, Structure and Conducting Properties of Halo-
Moriya, Tomokazu.
genated Ethylenedioxytetrathiafulvalenes. 833
Synthesis, Structure and Spectroscopic Characteristics of
Mizukami, Yoshihiro.
2'-Boryl-4"-dimethylaminochalcones. Effect of an Intra-
Synthesis and Properties of ant+6,15-Epithia-183,-
molecular Boron-Oxygen Coordinate Bond to the Conju-
methanobenzo[e][14]annulene-7,14-dione, ant+5,14-
gated System. 929
Epithia-7,12-methanofu14 r]oan[n3ul,e4ne--5e,] 1[3 -
Murafuji, Toshihiro.
diones, and Their lonic Species. 159
Synthesis, Structure and Spectroscopic Characteristics of
Mizuno, Masahiro.
2'-Bory!-4"-dimethylaminochalcones. Effect of an Intra-
Synthesis and Properties of Novel Medium-sized Hetero-
molecular Boron-Oxygen Coordinate Bond to the Conju-
cyclic Compounds Containing Two Sulfur Atoms in the
gated System. 929
Ring and Synthetic Approaches to Conjugated Cyclic
Murai, Akio.
Disulfonium Ylides. 139
Benzyloxymethy! Group as a Convertible Internal Ligand
Mizuta, Yutaka.
for La(OTf)3-catalyzed 7-endo Ring-Openig of Hydroxy
Studies on Pyrimidine-annulated Heterocycles: Synthe-
sis and Function of Novel 9-Substituted Cycloheptal[b]- Epoxide. 109
pyrimido[5,4-d]furan-8,10(9H)-diones. 601 Murakami, Masahiro.
Monden, Yoshiko. Synthesis of N-Boc-3-amino-1,2-epoxy-4-phenylbutane
Synthesis of N-Boc-3-amino-1,2-epoxy-4-phenylbutane from (3S)-Hydroxy-y-butyrolactone by Means of the
from (3S)-Hydroxy-ybutyrolactone by Means of the Hofmann Rearrangement. 77
Hofmann Rearrangement. 77 Murakami, Satoshi.
Morl, Akira. Bis(ethylenethio)tetraselenafulvalene and Related Hybrid
1,3-Dipolar Cycloadditions of 3-Bromo-1,5- and 3-Bromo- Diselenadithiafulvalenes as Novel Electron Donors
1,7-azulenequinones with Diazomethane, DiphenylInitril- Forming Highly Conductive Complexes with 7,7,8,8-
imine, and Benzonitrile Oxide. 291 Tetracyanoquinodimethane. 225
Morl, Akira. Murakami, Toshiyuki.
Synthesis and Mercurophilic Properties of Acyclic and Chemical Constituents of Two Oriental Orchids, Calanthe
Thiolariat Ethers Having a Tropone Pendant. 351 discolor and C. liukiuensis: Precursor Indole Glycoside of
Morl, Akira. Tryptanthrin and Indirubin. 957
intramolecular Photocycloaddition of 2-Cycloalkenyl-1,3- Murashima, Takashi.
dioxin-4-one. Stereoselective Synthesis of cis-Eudes- Preparation of Meso-unsubstituted Porphyrins Substituted
mane-4,11-diols. 765 with Mono- and Tetraformy! and Other Electron-withdraw-
Mori, Takashi. ing Groups. 705
Tota! Syntheses of Plagiochins A and D, Macrocyclic Murata, Kiyoshi.
Bis(bibenzyls), by Pd(0) Catalyzed Intramolecular Stille- Quinoline Alkaloids of Orixa japonica. 1139
Kelly Reaction. 259 Murata, Shizuaki.
Morishita, Hiroshi. A Convenient Determination of Chiral Pteridines; Applica-