Heterocycles an International Journal for Reviews and Communications in Heterocyclic Chemistry 2000: Vol 53 Index

53 Pages·2000·11.9 MB·English

HETEROCYCLES, Vol . 53, No. 12, 2000
Author index Akita, Hiroyuki.
Volume 53, 2000 Total Synthesis of (+)-Galanolactone. 1811
Akita, Hiroyuki.
First Total Syntheses of (+)-Polyoxin B and (+)-Polyoxin
D. 2253
Al-Abed, Yousef.
Synthesis and Properties of a-Thiagra. A Substituted 5-
(2-Thieny!)pyrazolo[4,3-d]pyrimidin-7-one Bioisostere of
A Viagra®. 2643
Alcaro, Stefano.
Abdeligaleil, Samir A. M. Synthesis of the 4-Hydroxyimino-3-carboxamide-2-
Novel Rings B,D-Secolimonoids from the Stem Bark of quinolone with a New Heterocyclization Mechanism of
Khaya senegalensis. 2233 the Reaction between Carbon Suboxide and 2-Amino-
Abdel-Jalil, Raid J. benzamidoxime. 2789
Synthesis and Properties of a-Thiagra. A Substituted 5- Alguacil, Raquel.
(2-Thienyl)pyrazolo[4,3-d]pyrimidin-7-one Bioisostere of Polycyclic Hydroxyquinones. Part 31. Regioselective
Reactions of 6-Ethylsulfony!-3-phenyfuro[3,4-d]isoxazol-
Viagra®. 2643
4(6H)-one Anion with Quinone Monoketals. Application
Abdulkakhimovna, Atazhanova Gayane.
to the Preparation of Heteroanthracyclinone Analogues.
Synthesis and Crystal Structure of Pyrazoline Derivative
1029
of Pulegone. 2661
Almerico, Anna Maria.
Abe, Hitoshi.
Dipyrrolo{1 ,2-a:1',2’-c]quinazoline, a New Ring System
Reaction of N-Acylated Isofebrifugine with Acid. 2247
of Biological Interest. 1975
Abe, Noritaka.
Al-Thebeiti, Marzoog S.
Synthesis and Some Reactions of 1,8-Diamino-1-aza-
Synthesis of Some New Spiropyrazolo[4',5':5,6]pyrano-
azulenium Salts. 323
[2,3-d]pyrimidines. 621
Abe, Noritaka.
Amano, Tomohiro.
Reaction of 2-Hydrazino-1-azaazulene with Dipheny!-
A Facile Synthesis of 1-Alkyl-7-azaisatins. 1145
nitrone: Unexpected Formation of Phenylimino-p-benzo-
Ando, Masayoshi.
quinone-N-oxide. 353
Synthesis of Methylenebis(4-hydroxy-2-pyrone) or
Abele, Edgars.
Methylenebis(4-hydroxycoumarin) Derivatives by
Recent Advances in the Synthesis of Heterocycles from
Organic Solid State Reaction. 549
Oximes. 2285
Ando, Shinichi.
Abushamieh, Ahmad S.
Cycloaddition Reaction of Naphtho[bjcyclopropene with
Transition Metal Complexes of Derivatized Chiral
Tropone Derivatives under the Presence of Ytterbium
Dihydro-1 ,2,4-triazin-6-ones. Part. |. Nickel(II) Complex
Complex to Form Cyclic Ethers or Cyclic Ketones:
of (D)-3-Acety|-5-benzyl-1-phenyl-4,5-dihydro-1 ,2,4-
Solvent Effect of Chloroform and Benzene on the Reac-
triazin-6-one Oxime. An Instance of a Carbon-Carbon
tion Path. 2601
Coupling Reaction. 1155
Andoh, Jun-ichi.
Abushamieh, Ahmad S.
New Reduction Reaction of Benzylic Alcohols with
Synthesis and Structural Characterization of Palladium(Il)
Acid and Proof of the Intermolecular Hydride Shift
Complex with (L)-3-Acety|-5-benzyl-1-pheny|-4,5-dihydro-
Mechanism. 359
1,2,4-triazin-6-one Oxime. Part Il. 1737
Anoro, Sonia.
Adachi, Norihide.
1,3-Dipolar Cycloaddition between Hetary! Nitrones and
Preparation and Spectral Properties of the Nitrogen
Methy! Acrylate: Theoretical Study and Application to the
Analogs of (&)-5,5'-Diary|-3,3'-bifuranylidene-2,2'-diones
Synthesis of Functionalized Pyrrolidines. 861
and Their Derivatives. 135
Antunes, Octavio A. C.
Ahmad, Habib.
5-Butyl-3,5-diaryl-4,5-dihydro-1,2,4-oxadiazoles, and a
Royleinine, a New Norditerpenoid Alkaloid from Delphi-
One-Step Synthesis of 4,4-Dibutyl-2-phenylbenzo-1,3-
nium roylei. 2279
oxazine. 191
Ahmad, Manzoor.
Anzai, Jun-ichi.
Royleinine, a New Norditerpenoid Alkaloid from Delphi-
Selective Electrocatalytic Oxidation of Amines Mediated
nium roylei. 2279
HETEROCYCLES, Vol . 53, No. 12, 2000
by Decahydroquinolinyl-N-oxy! Radical. 1583 6-one Derivatives with Cytotoxic Activity. 93
Aoyagi, Harumi. Atassi, Ghanem.
Catalytic Asymmetric Synthesis of Chiral 4-Pyrazoly!- Access to New Cytotoxic Bisindole Alkaloids by a Modi-
alkanols by the Enantioselective Alkylation of Pyrazole- fied Borch Reductive Amination Process. 2353
4-carbaldehydes with Dialkyizincs. 381 Atta-ur-Rahman.
Aral, Yoshitsugu. Synthesis and Crystal Structure of Pyrazoline Derivative
B-Lactam Synthesis by Diastereoselective Conden- of Pulegone. 2661
sation of Chiral 3-(p-Tolylsulfiny!)-2-furaldimine and Avendafio, Carmen.
Ester Enolate. 1479 Synthesis of a Seco Analogue of Ardeemin. 1765
Arakl, Lisa. Avila-Zarraga, José Gustavo.
Synthesis of the New Triheterocyclic System C3N-C4N-
Synthesis of 4(5)-(5'-Amino-5'-deoxy-a-L-arabinofurano-
syl)imidazole and Its 5'-Derivatives Using Modified CN. 3-Aryl-2,5,5-trimethyl-9a-methylsulfany!-9-phenoxy-
Mitsunobu Cyclization: Synthetic Studies toward Novel 4,5,6,8,9,9a-hexahydro-3H-azetof[1 ,2-a]pyrrolo[3,2-cj-
Histamine H3-Ligands. 1957 azepin-8-ones. 557
Araki, Lisa. Awadu, Yasutaka.
Stereoselective Synthesis of 4(5)-[(2S,3S)- and (2A,3A)- Electrochemistry of 1,3-Diazadihydroazulanone: Electro-
3-Aminotetrahydrofuran-2-yl)imidazoles Using Modified chemical Reduction and Oxidation of 1-Tosyl-3-aryl-1,3-
and Standard Mitsunobu Cyclizations: Synthetic Studies diazadihydroazulanone Leading to Migration and Elimi-
toward Novel Histamine H3-Ligands. 2739 nation of the Tosy! Group. 519
Azuma, Kumiko.
Arfan, Muhammed.
Reaction of N-Acylated Isofebrifugine with Acid. 2247
Royleinine, a New Norditerpenoid Alkaloid from Delphi-
Azuma, Mayumi.
nium roylei. 2279
Dimerization and Denitration of 1-Methyl-3,6,8-trinitro-
Argade, Narshinha P.
2-quinolone. 543
Ring Closure Reactions of Suitably ortho-Substituted
Maleanilic Acids: An Avenue for Heterocycles. 475
Ariga, Masahiro.
Dimerization and Denitration of 1-Methyl-3,6,8-trinitro-
2-quinolone. 543
Artali, Roberto.
Bae, Jaehoon.
Structural and Conformational Studies of 3,8-Diazabi-
An Efficient Synthesis of Novel Analogs of Water-soluble
cyclo[3.2.1]octane Derivatives, Selective Agonists of
and Hydrolytically Stable Deoxoartemisinin. 261
p-Opioid Receptors. 2403
Bae, Su-Hak.
Artico, Marino.
Reactions of Tetrasulfur Tetranitride Antimony Penta-
Reductive Smiles Rearrangement of 1-[(5-Chloro-2-nitro-
chloride Complex (S4N4°SbCls) with Primary B-
phenyl)sulfonyl]-1 H-pyrrole-2-carbohydrazide to 1-Amino-
6-chloro-2-(1H-pyrrol-2-yl)benzimidazole. 2163 Enaminones and B-Enamino Esters: Synthesis of
Asai, Koosuke. 4-Substituted 3-Aroyl- and 3-Ethoxycarbonyl-1,2,5-
Stereochemical Aspects during Addition Reaction of thiadiazoles. 159
2-Cyano-1 ,2-dihydroisoquinolines with Bromine in Baek, Daejin.
Methanol with and without Pyridine. 821 The Synthesis of 2-Ethylthio-6-(3-hydroxy-1,2-O-isopro-
Asaka, Noriko. pylidenepropyl)pteridin-4(3H)-one. 1551
Dimerization and Denitration of 1-Methyl-3,6,8-trinitro- Baik, Woonphil.
2-quinolone. 543 Electrochemical Synthesis of 2-Aryl-2H-benzotriazoles
Asakawa, Yoshinori. and Their N-Oxides by Controlled Potential Cathodic
A Novel Dimeric Coumarin from Citrus lumia. 441 Electrolysis. 841
Ata, Athar. Balasubramanlyan, Vaidhyanatha.
12-Acetoxypseudopterolide: A New Diterpene from Ring Closure Reactions of Suitably ortho-Substituted
Pseudopterogorgia elisabethae. 717 Maleanilic Acid: An Avenue for Heterocycles. 475
Atassi, Ghanem. Balazs, Mihaly.
Synthesis and Conformational Analysis of Some New Chemistry of Indoles Carrying a Basic Function. Part VI.
Pyrano[2,3-c]xanthen-7-one and Pyrano[3,2-b]xanthen- Synthesis of a New Ring System with Indole Nucleus.
HETEROCYCLES, Vol. 53, No. 12, 2000
1515 Reactivity of 7-Aminoindazole as a Bidendate Nucleo-
Balci, Metin. phile. 2617
Trapping of Unsaturated Fulvene Endoperoxides with Bendi, Markus.
Dimethy! 1,2,4,5-Tetrazine-3,6-dicarboxylate: A New GABA-analogous Spirocyclic Amino Acid Esters, 5. N-
Synthesis of Alkylidene- and Arylidenemalonaldehydes. Benzyl-7-azaspiro[4.5}decane-1-carboxylates. 115
761 Benezech, Véronique.
Balogh, Gabor. Reactivity of Heterocyclic Enaminones: Regioselective
Synthesis of Pentacyclic Ring Systems, Indolo[2,3-alf1,2]- Synthesis of Polyfused Indolones. 905
oxazino[5,6-/quinolizine and Indolo[2,3-a]pyrano[3,2-/- Bernat, Juraj.
quinolizine, and Their Application for the Synthesis of A Novel Convenient Synthesis of 1,3,5,5-Tetrasubstituted
Eburnamine-Vincamine Alkaloids. 1697 Hexahydropyrimidine-4-thiones. 1171
Banik, Bimal K. Berner, Mathias.
Indium-mediated Facile Synthesis of 3-Unsubstituted A Synthesis of Dihydronitraraine. 2241
Ferroceny! B-Lactams. 2769 Bhagavatula, Lakshmi.
Barba, Fructuoso. Efficient Route to 1-Dimethylsulfamoyl-4-iodoimidazole,
Electrochemical Synthesis of 5-Amino- 4-benzoy!-3- lsomerisation of 1-Dimethylsulfamoyl-5-iodoimidazole
phenylfuran-2-carbonitrile. 1337 to 1-Dimethylsulfamoyl-4-iodoimidazole. 729
Barbe, Jean M. Bhaket, Pushpal.
Synthesis of New Heterocyclic Systems: Spirothiadi- Total Synthesis of a Novel Cytotoxic Metabolite Gymna-
azolepyrazolo[1,5,4-efl[1,5]benzodiazepines. 571 statinA. 143
Barbier, Christine. Bhat, Krishna L.
Preparation of Lavendamycin Analogues. 37 An Expeditious Synthesis of Pyrrolo[3,4-d]pyrimidine-2,4-
Barlocco, Daniela. dione from Uracil. 205
Structural and Conformational Studies of 3,8-Diazabi- Bhattacharyya, Kinkini.
cyclo[3.2.1]octane Derivatives, Selective Agonists of Norditerpenoid and Diterpenoid Alkaloids from the Roots
of Aconitum nasutum Fisch. ex Reichb. 1987
p-Opioid Receptors. 2403
Biehl, Edward R.
Barlocco, Daniela.
5,6-Dinitropheny! and 5-Aminophenyl-6-nitropheny! Preparation of N 1_Alkyl- and N1,N 1_Dialkylisoquinoline-
Analogues of the ACAT Inhibitor 5,6-Dipheny!-3-alkyl- 1,3-diamines and 1-Alkyl- and 1-Phenylisoquinolin-3-
aminopyridazines. 2709 amines from the Reaction of a-Cyano-o-tolunitrile with
Barraja, Paola. Lithium Amides, Alkyllithiums, and Phenyllithium. 291
Dipyrrolof1 ,2-a:1',2'-c]quinazoline, a New Ring System Biehl, Edward R.
of Biological Interest. 1975 Investigation on the Reaction of 2-Chloro-10H-pheno-
Batanero, Belén. thiazine under Aryne Forming Conditions. 373
Electrochemical Synthesis of 5-Amino-4-benzoy|-3- Biehl, Edward R.
phenylfuran-2-carbonitrile. 1337 Convenient Synthesis of 1-Substituted Derivatives of
Baurzhanovich, Khasenov Bekboliat. 4-([E]-1-Propenyl)- and 4-Allyl-3-aminoisoquinolines.
Synthesis and Crystal Structure of Pyrazoline Derivative 1183
of Pulegone. 2661 Bitter, Istvan.
Becker, Frederick F. Synthesis of 5-Substituted Indole Derivatives, Part Il.
Indium-mediated Facile Synthesis of 3-Unsubstituted Synthesis of Sumatriptan through the Japp-Klingemann
Ferrocenyl B-Lactams. 2769 Reaction. 665
Begum, Sabira. Blache, Yves.
Two New Pentacyclic Triterpenoids from the Aerial Parts Reactivity of Heterocyclic Enaminones: Regioselective
of Lantana camara Linn. 681 Synthesis of Polyfused Indolones. 905
Beltrame, Paolo. Blazquez, J. A. Serrano.
Reactions of a Stable Benzonitrile Oxide with Amino- Synthesis of Polycylic Systems via Diels-Alder Reactions
pyridines. 1915 of Sugar Derived Dienes. 81
Benchidmi, Mohammed. Bock, Charles W.
Synthesis of New Heterocyclic Systems: Spirothiadi- An Expeditious Synthesis of Pyrrolo[3,4-d]pyrimidine-2,4-
azolepyrazolo[1,5,4-ef[1,5]benzodiazepines. 571 dione from Uracil. 205
Benchidmi, Mohammed. Bogdal, Dariusz.
HETEROCYCLES, Vol. 53, No. 12, 2000
Carbazoly! Nitrenium Cations: Generation and Reactions. Total Synthesis and Conformational Analysis of Mono-
2679 phenyl! Substituted Protoporphyrins. IX. 2127
Bolasco, Adriana. Burtin, Gullilaume E.
Synthesis of the 4-Hydroxyimino-3-carboxamide-2- New Synthesis of KT5823 Indolocarbazole Aglycone.
quinolone with a New Heterocyclization Mechanism of 2119
the Reaction between Carbon Suboxide and 2-Amino- Buscemi, Silvestre.
benzamidoxime. 2789 Sensitized Photoreduction of Nitrosoazoles on Titanium
Bombieri, Gabriella. Dioxide. 183
Structural and Conformational Studies of 3,8-Diazabi-
cyclo[3.2.1}octane Derivatives, Selective Agonists of
p-Opioid Receptors. 2403
Cc
Bompart, Jacques.
Solution Parallel Synthesis of Cyclic Guanidines.
Caballero, Esmeralda.
1317
Synthesis of a Seco Analogue of Ardeemin. 1765
Bonnet, Pierre-Antoine.
Solution Parallel Synthesis of Cyclic Guanidines. Cadoni, Enzo.
Reactions of a Stable Benzonitrile Oxide with Amino-
1317
pyridines. 1915
Bonsignore, Leonardo.
Caignard, Daniel H.
Synthesis of the 4-Hydroxyimino-3-carboxamide-2-
Synthesis and Conformational Analysis of Some New
quinolone with a New Heterocyclization Mechanism of
Pyrano[2,3-c]xanthen-7-one and Pyrano[3,2-b]xanthen-
the Reaction between Carbon Suboxide and 2-Amino-
6-one Derivatives with Cytotoxic Activity. 93
benzamidoxime. 2789
Calas, Michéle.
Boryczka, Stanistaw.
Solution Parallel Synthesis of Cyclic Guanidines.
Reactions of Thioquinanthrene with Disodium Salts of
Glycols. 1905 1317
Cafiada-Rudner, Pedro.
Boule, Pierre.
Solvent-free Synthesis of Thio-alkyixanthines from Alkyl-
Reactivity of Heterocyclic Enaminones: Regioselective
xanthines Using Microwave Irradiation. 2275
Synthesis of Polyfused Indolones. 905
Boyer, Gérard. Caronna, Tullio.
Sensitized Photoreduction of Nitrosoazoles on Titanium
Synthesis of New N-Alkyl- and N-Acylidioxinopheno-
thiazine and Acridinone Derivatives. 2535 Dioxide. 183
Bravo, P. Areces. Carrero, M. C. Pozo.
Synthesis of Polycylic Systems via Diels-Alder Reactions
Synthesis of Polycylic Systems via Diels-Alder Reactions
of Sugar Derived Dienes. 81 of Sugar Derived Dienes. 81
Bremner, John B. Carta, Antonio.
Synthesis of Two Novel Tricyclic Rings: Triazolo[4,5-g]-
Novel Indole-fused, Medium-sized Ring Heterocycles
quinolines and Pyrido[2,3-g]quinoxalines Derived from
via Chloroacetamide Photochemistry. 277
6,7-Diaminoquinolines. 423
Brinn, tra M.
5-Buty!-3,5-diaryl-4,5-dihydro-1,2,4-oxadiazoles, and a Carvalho, Carlos Eduardo M.
5-Butyl-3,5-diaryl-4,5-dihydro-1,2,4-oxadiazoles, and a
One-Step Synthesis of 4,4-Dibutyl-2-phenylbenzo-1 ,3-
One-Step Synthesis of 4,4-Dibutyl-2-phenylbenzo-1,3-
oxazine. 191
Broggini, Giantuigl. oxazine. 191
Dipolarophilic Behavior of the Isoxazole Ring in Intra- Castedo, Luis.
New Synthetic Applications of Phenylacetylphenylacetic
molecular Nitrilimine Cycloadditions. 831
Broggini, Gianluigi. Acids: A Divergent Synthesis of Benzo[a]carbazoles and
Nitrilimine Cycloadditions onto Partially Saturated Furo- Indolo[2,1-a]isoquinolines. 1041
[3,4-c}thieno[2,3-d]pyrazoles. A Problem in Site Selecti- Celentano, Giuseppe.
5,6-Dinitropheny! and 5-Aminophenyl-6-nitrophenyl
vity. 917
Analogues of the ACAT Inhibitor 5,6-Dipheny|-3-alkyl-
Bruno, Maurizio.
Hydrogenation Derivatives of Neo-clerodanes and Their aminopyridazines. 2709
Antifeedant Activity. 599 Cha, Ki Suk.
Buldain, Graciela Y. 1,3-Dihydro-1 ,3-diacetyl-2H-benzimidazol-2-one: A New
Versatile and Selective Acetylating Agent. 529
HETEROCYCLES, Vol. 53, No. 12, 2000
Chapat, Jean-Pierre. benzamidoxime. 2789
Reactivity of Heterocyclic Enaminones: Regioselective Chimirri, Alba.
Synthesis of Polyfused Indolones. 905 Synthesis and Structural Features of New Cyclofunction-
Chatel, Florence. alized Benzimidazoles. 613
Synthesis of New N-Alkyl- and N-Acyldioxinopheno- Chol, Sang Uk.
thiazine and Acridinone Derivatives. 2535 Stereoselective Synthesis of 1,4-Dideoxy-1,4-imino-L-
Chavignon, Olivier. lyxitol and 1,5-Dideoxy-1,5-imino-D-ribitol. 887
Reactivity of Heterocyclic Enaminones: Regioselective Choméa, Igor.
Synthesis of Polyfused Indolones. 905 A Novel Convenient Synthesis of 1,3,5,5-Tetrasubstituted
Chen, Hul. Hexahydropyrimidine-4-thiones. 1171
Stereoselective Synthesis of (Z)-a-Phenoxymethylene- Choshl, Tominari.
y-butyrolactone and Its Sulfur Analogues from 2-Pro- The First Total Synthesis of (A)-(-)-Pyridindolol K2 and
Its Enantiomer. 1877
pynyloxy- or 2-Propynylthiobenzene. 2055
Choudhary, Muhammad Iqbal.
Chen, Jianxin.
Synthesis and Crystal Structure of Pyrazoline Derivative
Reactions of 1,2-Dimethyl-3-arylsulfony|-4,5-dihydro-3H-
of Pulegone. 2661
imidazol-1-ium lodides with Bifunctional Nucleophiles.
433 Chung, Bong Young.
1,3-Dihydro-1 ,3-diacetyl-2H-benzimidazol-2-one: A New
Chen, Kuo-Tung.
Versatile and Selective Acetylating Agent. 529
Cathylation of 4,6-Dimethy|-2-oxopyridine-3-carbonitrile
Chung, In Hwa.
Derivatives Leading to the Synthesis of Furo[2,3-b;4,5-b']-
dipyridines and Novel Tricyclic Furo[2,3,4-jj[2, 7]naphthy- 1,3-Dihydro-1 ,3-diacetyl-2H-benzimidazol-2-one: A New
Versatile and Selective Acetylating Agent. 529
ridine. 15
Cignarella, Giorgio.
Chen, Shul-Tein.
Structural and Conformational Studies of 3,8-Diazabi-
A Synthesis of Cytonin (Taiwanin A), an Antitumor
cyclo[3.2.1]octane Derivatives, Selective Agonists of
Lignan. 1569
Chen, Zhi-He. u-Opioid Receptors. 2403
Three New Diterpene Alkaloids from Spiraea japonica. Commercon, Alain.
1343 Preparation of Lavendamycin Analogues. 37
Cheng, Qian. Copp, Richard R.
Chemical Oxidation of Taxoids with m-CPBA and Synthesis of a 5-Substituted Benzo[b]thiophene. 1175
Dimethy! Dioxirane: Regioselective Epoxidation of Corsaro, Antonino.
Taxinine J Derivatives. 2629 1,3-Dipolar Cycloaddition Reactions of Benzonitrile Oxide
Cheng, Qian. to 2(1H)-Pyrazinone and Its N- and O-Methy! Derivatives.
High Regio- and Stereoselectivity in Facile One-Pot 69
Conversion of Taxoids to the Primary Alcohols: Croce, Piero Dalia
Precursors for the Synthesis of 4-Deacetoxypacilitaxel Studies on Ring Opening Reactions of N-Phenylsulfony!
and Analogues. 2759 Substituted Spiro-B-lactams. 2653
Chezal, Jean-Michel. Crozet, Michel P.
Reactivity of Heterocyclic Enaminones: Regioselective Preparation of 2-Substituted Naphth[2,3-djoxazole-4,9-
Synthesis of Polyfused Indolones. 905 diones via a Radical Chain Process. 1075
Chiacchio, Ugo. Cruces, Jacobo.
1,3-Dipolar Cycloaddition Reactions of Benzonitrile Oxide New Synthetic Applications of Phenylacetylphenylacetic
to 2(1H)-Pyrazinone and Its N- and O-Methy! Derivatives. Acids: A Divergent Synthesis of Benzo[ajcarbazoles and
69 Indolo[2,1-a]isoquinolines. 1041
Chiba, Jun. Csende, Ferenc.
Synthesis and Antitumor Activity of Non-Prodrug Water- 4- and 5-Oxocarboxylic Acids as Versatile Synthons for
soluble Taxoid: 10-C-Aminoalkylated Docetaxel Analogs. the Preparation of Heterocycles. 1379
2719 Czibula, Laszid.
Chimenti, Franco. Synthesis of Pentacyclic Ring Systems, Indolo[2,3-a][1,2]-
Synthesis of the 4-Hydroxyimino-3-carboxamide-2- oxazino[5,6-i ]quinolizine and Indolo[2,3-a]pyrano[3,2-/}-
quinolone with a New Heterocyclization Mechanism of quinolizine, and Their Application for the Synthesis of
the Reaction between Carbon Suboxide and 2-Amino- Eburnamine-Vincamine Alkaloids. 1697
HETEROCYCLES, Vol. 53, No. 12, 2000
Czugler, Matyas. cean briareum Sp. 1789
Chemistry of Heterocyclic Pseudobasic Amino-Carbinols. Doe, Matsumi.
Part 37. Correction of a Structure — A New Heterocyclic Novel Rings B,D-Secolimonoids from the Stem Bark of
Ring System. 697 Khaya senegalensis. 2233
Dondela, Barbara.
Cyclodextrin Host-Guest Systems Containing Aza-
aromatic Moieties. 1595
D
Danagulyan, Gevorg G.
Exchange Aminations in Conversions of Pyrimidinium E
lodides to 2-Alkylaminonicotinic Acids. 419
Davoll, Paolo. Eckert, Katrin.
A Novel Approach to a Precursor of the Carbapenem New Syntheses of 2-Alkylthio-4-oxo-3,4-dihydroquinazo-
Antibiotic PS-5 via Aziridine Stereospecific Carbonylation. lines, 2-Alkylthioquinazolines, as well as Their Hetero
2379 Analogues. 2363
Dellios, Constantinos C. Eder, Michael.
A New Synthesis of (-)-(5A,6S)-6-Acetoxy-5-hexadeca- GABA-analogous Spirocyclic Amino Acid Esters, 5. N-
nolide, the Mosquito Culex pipiens fatigans Oviposition Benzyl-7-azaspiro[4.5]decane-1-carboxylates. 115
Attractant Pheromone. 703 El-Abadelah, Mustafa M.
De Martino, Gabriella. Transition Metal Complexes of Derivatized Chiral
Reductive Smiles Rearrangement of 1-[(5-Chioro-2-nitro- Dihydro-1 ,2,4-triazin-6-ones. Part |. Nickel(II) Complex
pheny!)sulfony/]-1 H-pyrrole-2-carbohydrazide to 1-Amino- of (D)-3-Acetyl-5-benzyl-1-phenyl-4,5-dihydro-1 ,2,4-
6-chloro-2-(1H-pyrrol-2-yl)benzimidazole. 2163 triazin-6-one Oxime. An Instance of a Carbon-Carbon
Deniaud, David. Coupling Reaction. 1155
[4+2] Cycloaddition Reactions between 2,4-Diamino- El-Abadelah, Mustafa M.
1-thia-3-azabutadienes and Ketene. Synthesis of New Synthesis and Structural Characterization of Palladium(ll)
1,3-Thiazin-6-ones, 1,3-Thiazine-6-thiones and 2- Complex with (L)-3-Acetyl-5-benzyl-1-phenyl-4,5-dihydro-
Thioxopyrimidin-4-ones. 2667 1,2,4-triazin-6-one Oxime. Part Il. 1737
Denisenko, Sergey N. El-Abadelah, Mustafa M.
Exchange Aminations in Conversions of Pyrimidinium Synthesis and Properties of a-Thiagra. A Substituted 5-
lodides to 2-Alkylaminonicotinic Acids. 419 (2-Thieny!)pyrazolo[4,3-d]pyrimidin-7-one Bioisostere of
Depreux, Patrick.
Viagra®, 2643
Synthesis of 4-[4'-(N, N-Dimethylsulfamoyl)piperazin-1 -yl]-
E! Bouadili, Abdelazi0z.
pyridine Derivatives as Sorbito! Dehydrogenase Potential
Synthesis of New Heterocyclic Systems: Spirothiadi-
Inhibitors. 797
azolepyrazolo[1,5,4-ef][1,5]}benzodiazepines. 571
Desal, Haridutt K.
El Bouadill, Abdelaziz.
Norditerpenoid and Diterpenoid Alkaloids from the Roots
Reactivity of 7-Aminoindazole as a Bidendate Nucleo-
of Aconitum nasutum Fisch. ex Reichb. 1987
phile. 2617
Diana, Patrizia.
El-Hiti, Gamal A.
Dipyrrolo[1 ,2-a:1',2'-c]quinazoline, a New Ring System
Synthesis of Substituted Quinazolin-4(3H)-ones and
of Biological Interest. 1975
Quinazolines via Directed Lithiation. 1839
Dittami, James P.
Endo, Yasuyuki.
The Synthesis of an Aminohexyl-containing Analog of
Anionic [3,3] Rearrangements of Cyclic Hydrazine
the Chromanol Leukotriene B4 Receptor Antagonist
Diacylates to Medium-Size Cyclic Diamides and Their
CP-195543: A Scaffold for the Preparation of Derivatized Structures. 151
Analogs. 1713
Enomoto, Yasuko.
Dmitrievich, Dembitsky Alexandr. A Selective Synthesis of Both Enantiomers of a 1-Allyi-
Synthesis and Crystal Structure of Pyrazoline Derivative
B-carboline Using the Same Chiral Auxiliary Derived
of Pulegone. 2661
from L-Proline. 2357
Doe, Matsumi.
Escale, Roger.
Violides N-P, New Briarane Diterpenes from a Gorgona-
Solution Parallel Synthesis of Cyclic Guanidines.
HETEROCYCLES, Vol . 53, No. 12, 2000
1317 pyridine Derivatives as Sorbitol Dehydrogenase Potential
Essassi, El Mokhtar. Inhibitors. 797
Synthesis of New Heterocyclic Systems: Spirothiadi- Fujieda, Mieko.
azolepyrazolo[1,5,4-efl[1,5]benzodiazepines. 571 Total Syntheses of Naamine A and Naamidine A, Marine
Essassi, El Mokhtar. Imidazole Alkaloids. 1939
Reactivity of 7-Aminoindazole as a Bidendate Nucleo- Fujii, Hiroyuki.
phile. 2617 Synthesis and Some Reactions of 1,8-Diamino-1-aza-
Estévez, Juan C. azulenium Salts. 323
New Synthetic Applications of Phenylacetylphenylacetic Fujii, Hiroyuki.
Acids: A Divergent Synthesis of Benzo[a]carbazoles and Reaction of 2-Hydrazino-1-azaazulene with Diphenyl-
Indolo[2,1-alisoquinolines. 1041 nitrone: Unexpected Formation of Phenylimino-p-benzo-
Estévez, Ramon J. quinone-N-oxide. 353
New Synthetic Applications of Phenylacetylphenylacetic Fujimoto, Norikazu.
Acids: A Divergent Synthesis of Benzo[a]carbazoles and Synthesis of Methylenebis(4-hydroxy-2-pyrone) or
Indolo[2,1-alJisoquinolines. 1041 Methylenebis(4-hydroxycoumarin) Derivatives by
Eszenyjl, Tibor. Organic Solid State Reaction. 549
Synthesis of 2,2-Dimethy|-2H-chromenes. 1193 Fujisawa, Kenji.
Eto, Masashi. Stereoselective Synthesis of the 3-Hydroxytetrahydro-
X-Ray Structures of a Pair of Atropisomers of 1-(3'- pyran Part of Mucocin, an Antitumor Agent, Based on
Substituted Benzoy!)-2-naphthylindolines and Some Rearrangement-Ring Expansion Reaction of a Tetra-
Comments. 1 hydrofuran Derivative. 1361
Fujita, Reiko.
Novel Synthesis of Tetrahydro-2(1H)-quinolones Using
Diels-Alder Reactions of 1-Aryisulfonyl-2(1H)-pyridones
Acting as Dienophiles. 2607
Fujita, Tsutomu.
Fang, Yunfeng. Palladium-catalyzed Asymmetric Allylic Alkylation Using
A Convenient Route to B-Phenylthioalky! Ketones. Chiral P,N-Ligands. 1485
331 Fujiwara, Hidetoshi.
Fang, Yunfeng. Synthesis of Pyridopyranoquinolines by the Skraup
Benzotriazole-mediated [1,2] Wittig Rearrangement. Reaction of Amino-5H-benzopyrano[2,3-b]pyridin-
The Preparation of Homoalcohols from Ethers. 1783 5-ones. 409
Farkas, Maria. Fukal, Toshio.
Synthesis of Pentacyclic Ring Systems, Indolo[2,3-al[1,2]- LI-F Antibiotics, a Family of Antifungal Cyclic Depsi-
oxazino[5,6-/ }quinolizine and Indolo[2,3-a]pyrano[3,2-]i - peptides Produced by Bacillus polymyxaL-1129. 1533
quinolizine, and Their Application for the Synthesis of Fukui, Yoshikazu.
Eburnamine-Vincamine Alkaloids. 1697 Syntheses of Melatonin and Its Derivatives. 1725
Faure, Robert. Fukuman, Yukari.
Synthesis of New Thiazolo[5,4-a]acridine Derivatives. Nimbolinins, C-Seco Limonoids from the Fruits of Melia
387 toosendan. 689
Fawcett, John. Fukuzawa, Yuichi.
Synthesis of 2H-Naphtho[2,3-b]thiopyranoquinones and Photochemistry of N-3-Butenyl- and N-4-Pentenyl-
Density Functional Study for the Diels-Alder Reaction of glutarimides: Intramolecular Thietane Formation and
a Benzothiopyranoquinone. 585 the Fission of Thietane Ring. 2781
Feng, Daming. Fille, Friederike.
A Convenient Route to B-Phenylthioalky! Ketones. A Novel Ring Closure Reaction for the Preparation of
331 6-Aminouracils with an a-Branched 1-Substituent. 347
Floris, Costantino. Funabashi, Makoto.
Reactions of a Stable Benzonitrile Oxide with Amino- Synthesis of New Mesomeric Betaines Containing a
pyridines. 1915 Triazolopyridiniumolate System and Their Unexpected
Fourmaintraux, Eric. Function as Masked Isocyanates. 265
Synthesis of 4-[4'-(N, N-Dimethylsulfamoy!)piperazin-1 -yl]- Furule, Hisakazu.
HETEROCYCLES, Vol. 53, No. 12, 2000
Synthesis of Bornene Ring-fused Dihydrothiopyrans, a Ge, Xuejun.
New Class of Chiral Cyclic Sulfides, via Intramolecular 1-epi-Deacetylaconitine, a New Norditerpenoid Alkaloid
Hetero Diels-Alder Reaction of Homochiral Thiabutadi- from Aconitum nemorum. 2027
enes, 3-(Aryimethylene)thiocamphors. 1685 Gelli, Gioanna.
Furukawa, Hiroshi. Reactions of a Stable Benzonitrile Oxide with Amino-
A Novel Dimeric Coumarin from Citrus lumia. 441 pyridines. 1915
Gewald, Karl.
New Syntheses of 2-Alkylthio-4-oxo-3,4-dihydroquinazo-
lines, 2-Alkylthioquinazolines, as well as Their Hetero
G Analogues. 2363
Ghatak, Anjan.
Gacs-Baltz, Eszter. Indium-mediated Facile Synthesis of 3-Unsubstituted
Chemistry of Indoles Carrying a Basic Function. Part VI. Ferrocenyl B-Lactams. 2769
Synthesis of a New Ring System with Indole Nucleus.
Ghirtis, Konstantinos.
1515 Synthesis and Conformational Analysis of Some New
Galan, E. Roman. Pyrano[2,3-c]xanthen-7-one and Pyrano[3,2-b]xanthen-
Synthesis of Polycylic Systems via Diels-Alder Reactions 6-one Derivatives with Cytotoxic Activity. 93
of Sugar Derived Dienes. 81 Gilheany, Declan G.
Galeazzi, Roberta. Easy Access to Medium Rings by Entropy/Strain Reduc-
The Cleavage of Sulfonylurea Herbicide Rimsulfuron® tion, Part 4. A Simple and Mild Route to Some Substitu-
under Basic Conditions: A Computational Investigation. ted 2,7-Dihydro-1H-oxepins, thiepins and a Phosphepin.
2517 897
Gallos, John K. Giovannonl, Maria Paola.
A New Synthesis of (-)-(5A,6S)-6-Acetoxy-5-hexadeca- 5,6-Dinitropheny! and 5-Aminopheny!-6-nitropheny|
nolide, the Mosquito Culex pipiens fatigans Oviposition Analogues of the ACAT Inhibitor 5,6-Diphenyl-3-alkyI-
Attractant Pheromone. 703 aminopyridazines. 2709
Galy, Jean-Pierre. Girreser, Ulrich.
Synthesis of New Thiazolo[5,4-a]lacridine Derivatives. 3-(2-Benzoylallyl)-4-hydroxy-6-methylpyran-2-ones:
387 Synthesis and Intra- and Intermolecular Nucleophilic
Galy, Jean Pierre. Additions. 2421
Synthesis of New N-Alkyl- and N-Acyldioxinopheno- Gmeiner, Peter.
thiazine and Acridinone Derivatives. 2535 Synthesis of Enantiopure 8-Aminomethylindolizines from
Gama, Yasuo. Glutamine by Stereoelectronically Controlled Cationic
A Novel and Convenient Synthesis of 1,3,5-Triazine- Cyclization. 1371
2,4(1H,3H)-diones. 929 Golic, Ljubo.
Gama, Yasuo. A Synthesis and Transformations of Alkyl 2-[2-Cyano-2-
Sythesis of 2-(2-Alkoxycarbonylpheny!thio)-1,2-benziso- (2-pyridinyl)etheny!]Jamino-3-dimethylaminopropenoates.
thiazolin-3-ones from 2-Sulfenamoylbenzoates. 2803 A One-Pot Synthesis of Pyrrolo[3,2-d]pyrimidin-4-ones.
Garanti, Luisa. 805
Dipolarophilic Behavior of the Isoxazole Ring in Intra- Golobié, Amalija.
molecular Nitrilimine Cycloadditions. 831 A Synthesis and Transformations of Alkyl! 2-[2-Cyano-2-
Garanti, Luisa. (2-pyridinyl)ethenyl]jamino-3-dimethylaminopropenoates.
Nitrilimine Cycloadditions onto Partially Saturated Furo- A One-Pot Synthesis of Pyrrolo[3,2-d]pyrimidin-4-ones.
[3,4-c]thieno[2,3-d]pyrazoles. A Problem in Site Selecti- 805
vity. 917 Goto, Aya.
Garate, Miriam C. Synthesis of 3a-(Indol-3-yl)-1,2,3,3a,8,8a-hexahydro-
Synthesis of 2H-Naphtho[2,3-bjthiopyranoquinones and pyrrolo[2,3-b]lindole Core of Leptosins D-F Based on
Density Functional Study for the Diels-Alder Reaction of Nucelophilic Substitution Reaction on Indole Nucleus.
a Benzothiopyranoquinone. 585 1255
Garcia, Maria B. Goto, Aya.
Synthesis of 1-Aryl-1,4,5,6-tetrahydropyrimidines and 1- Reactions of 1-Hydroxyindoles with p-Toluenesulfonyl
Aryl-3-substituted1,4,5,6-Tetrahydropyrimidinium Salts. Chloride and p-Toluenesulfonic Acid. 2487
2437
HETEROCVolY. 5C3,L NoE. 1S2, ,20 00
Gromov, Sergey P. Hamada, Nobuo.
Ring Transformation of Pyridines and Benzo Derivatives Two lsocoumarins from the Cultured Lichen Mycobiont
under the Action of C-Nucleophiles. 1607 of Graphis Sp. 723
Gruner, Margit. Hamada, Nobuo.
New Syntheses of 2-Alkylthio-4-oxo-3,4-dihydroquinazo- 2,3-Dialkyichromones from Mycobiont Cultures of the
lines, 2-Alkytthioquinazolines, as well as Their Hetero Lichen Graphis scripta. 1589
Analogues. 2363 Hamada, Yosikl.
Gu, Xiao-Hul. Stereochemical Aspects during Addition Reaction of
Syntheses of Bis(3'-indoly!)-2(1H)pyrazinones. 1559 2-Cyano-1,2-dihydroisoquinolines with Bromine in
Gundersen, Lise-Lotte. Methanol with and without Pyridine. 821
Synthesis of Heteromine C from Guanine. 935 Han, Rongbi.
Guo, Dean. Electrochemical Synthesis of 2-Aryl-2H-benzotriazoles
Gaultthrins C and D, Two New Lignans from the Roots and Their N-Oxides by Controlled Potential Cathodic
of Gaultheria yunnanensis. 675 Electrolysis. 841
Gurjar, Mukund K. Handa, Masaki.
Total Synthesis of a Novel Cytotoxic Metabolite Gymna- Total Syntheses of Kurasoins A and B, Novel Protein
statinA. 143 Farnesyltransferase Inhibitors, and Absolute Structures
Gurjar, Mukund K. of Kurasoins Aand B. 777
Towards the Synthesis of Scyphostatin. 1885 Hano, Yoshio.
Guspanova, Janka. Mechanism on One-sided Wessely-Moser Rearrange-
A Novel Convenient Synthesis of 1,3,5,5-Tetrasubstituted ment Reaction. 877
Hexahydropyrimidine-4-thiones. 1171 Hao, Xiao-Jiang.
Three New Diterpene Alkaloids from Spiraea japonica.
1343
Hao, Xiao-Jiang.
H O-Terpenoidal Coumarins from Clausena excavata.
1807
Hachiken, Hiroko. Hao, Xiaojiang.
Reaction of 3-Ethoxycarbonylindolizine-1,2-dicarboxylic Six New O-Terpenoidal Coumarins, Excavacoumarins
Anhydride with (3-Bromo-4-pyridyl)triisopropoxytitanium: B-G from Clausena excavata. 2067
Synthesis of 5,12-Dimethylindolizino[2, 1-g]isoquinoline Hao, Xiaojiang.
(Ellipticine Analogue). 2123 Prieurianin-Type Tetranortriterpenoids from the Bark of
Hachiken, Hiroko. Dysoxylum hainanense. 2225
Reaction of 3-Ethoxycarbonylindolizine-1 ,2-dicarboxylic Harano, Kazunobu.
Anhydride: Synthesis of 2-Acylindolizines and Quinones. X-Ray Structures of a Pair of Atropisomers of 1-(3'-
2143 Substituted Benzoyl)-2-naphthylindolines and Some
Haddadin, Makhiuf J. Comments. 1
A Tetracycloundecane Derivative of Pyrrolidinobenz- Harano, Kazunobu.
oxazinone. 2221 A Diamine-Exchange Reaction of Dihydropyrazines.
Hagiwara, Hisahiro. 1677
Synthesis of Methylenebis(4-hydroxy-2-pyrone) or Harayama, Takashi.
Methylenebis(4-hydroxycoumarin) Derivatives by Reaction of N-Acylated Isofebrifugine with Acid. 2247
Organic Solid State Reaction. 549 Harigaya, Yoshihiro.
Hagiwara, Masanori. Total Syntheses of Kurasoins A and B, Novel Protein
Condensation Reactions of a Nitrodienamine with Organo- Farnesyltransferase Inhibitors, and Absolute Structures
copper and Alkyllithium Reagents Prepared from Pyrrole of Kurasoins A and B. 777
Derivatives. 1351 Harsanyi, Kalman.
Haider, Norbert. Synthesis of 5-Substituted Indole Derivatives, Part li.
Radicalic Ethoxycarbonylation of 3-lodopyridazines: An Synthesis of Sumatriptan through the Japp-Klingemann
Efficient Access to Tri- and Tetrasubstituted Pyridazines. Reaction. 665
2527 Harusawa, Shinya.
Haight, Anthony R. Synthesis of 4(5)-(5'-Amino-5'-deoxy-a-L-arabinofurano-
Synthesis of a 5-Substituted Benzo[b]thiophene. 1175
HETEROCYCLES, Voi. 53, No. 12, 2000
syl)imidazole and Its 5'-Derivatives Using Modified 447
Mitsunobu Cyclization: Synthetic Studies toward Novel Hayashi, Masumi.
Histamine H3-Ligands. 1957 Reactions of 1-Hydroxyindoles with p-Toluenesulfony!
Harusawa, Shinya. Chloride and p-Toluenesulfonic Acid. 2487
Stereoselective Synthesis of 4(5)-[(2S,3S)- and (2A,3A)- Hayashi, Toshikatsu.
3-Aminotetrahydrofuran-2-yl)imidazoles Using Modified Syntheses of Melatonin and Its Derivatives. 1725
and Standard Mitsunobu Cyclizations: Synthetic Studies Hayashi, Toshikatsu.
toward Novel Histamine H3-Ligands. 2739 Simple Syntheses of Indol-1-yl Glucosides. 1881
He, Hongping.
Hasegawa, Masakazu.
O-Terpenoidal Coumarins from Clausena excavata.
The First Total Synthesis of Bufobutanoic Acid by Two
1807
Routes Based on Nucleophilic Substitution Reaction
He, Hongping.
on Indole Nucleus. 1017
Six New O-Terpenoidal Coumarins, Excavacoumarins
Hasegawa, Masakazu.
B-G from Clausena excavata. 2067
Syntheses of Melatonin and Its Derivatives. 1725
He, Yineng.
Hasegawa, Masakazu.
O-Terpenoidal Coumarins from Clausena excavata.
Reactions of 1-Hydroxyindoles with p-Toluenesulfony!
1807
Chloride and p-Toluenesulfonic Acid. 2487
He, Yineng.
Hasegawa, Minoru.
Six New O-Terpenoidal Coumarins, Excavacoumarins
Synthesis of Phenazine 5,10-Dioxides from Benzo-
B-G from Clausena excavata. 2067
furoxan Catalyzed by Molecular Sieves. 2151
Heber, Dieter.
Hashimoto, Iwao.
3-(2-Benzoylally!)-4-hydroxy-6-methylpyran-2-ones:
Synthesis of New Dihydroxy-dioxygenated ortho-[2,x]-
Synthesis and Intra- and Intermolecular Nucieophilic
Cyclophanes. 2459
Additions. 2421
Hashimoto, Tomomi.
Hibino, Hajime.
Addition Reactin of Cyclic Ethers to 1,1-Ethylene-1H-
Reaction of 3-Ethoxycarbonylindolizine-1 ,2-dicarboxylic
azulenium lon. 2071
Anhydride with (3-Bromo-4-pyridy|)triisopropoxytitanium:
Hashimoto, Toshihiro.
Synthesis of 5,12-Dimethylindolizino[2, 1-g]isoquinoline
A Novel Dimeric Coumarin from Citrus lumia. 441
(Ellipticine Analogue). 2123
Hassan, Hammed H. A. M.
Hibino, Satoshi.
Synthesis of Bridged Head Methyl 3,4-O-(1',2'-Dimethyl-
The First Total Synthesis of (A)-(-)-Pyridindolol K2 and
cyclohexane-1',2'-diyl)-6,7-dideoxy-a-D-mannooct-6-
Its Enantiomer. 1877
enepyranose-8,2-lactone from D-Mannose. 397
Higashiyama, Kimio.
Hatano, Keiichiro.
Synthesis of (+)-Hupeol from (-)-Cytisine: Transform-
Stereochemical Aspects during Addition Reaction of
ation of a Cyclic Imine into a Cyclic Hemiacetal. 545
2-Cyano-1 ,2-dihydroisoquinolines with Bromine in
Higashiyama, Kimio.
Methanol with and without Pyridine. 821
Synthesis of Co-Symmetrical Chiral Aromatic Diamines
Hattori, Yuhji.
by Diastereoselective Additon to Bis(1,3-oxazolidinyl)-
Short Step Synthesis of (4A)-4-Hydroxymethyl-4-methyl-
aromatics with Grignard Reagents. 2499
2-hexene-1,5-diol: A Useful Chiral Synthon for Natural
Hino, Ayako.
Product Synthesis with Quaternary Carbon Center.
An Efficient Total Synthesis of Ellipticine. 11
733
Hino, Ayako.
Hayano, Kiyoharu.
A Concise Access to 6-Azabicyclo[3.1.0]hexanes via
Conformation and Configuration of Humulene Di- and Tri-
High-Pressure Promoted Cycloaddition Reaction of
epoxides Generated from Four Possible Conformations
Azides to ABH. 1499
of Humulene 9,10-Epoxide. 1269
Hirakura, Kazuhiro.
Hayashi, Hirokazu.
Three Diels-Alder Type Adducts, Ginsenoynes L, M, and
Synthesis of Novel Macrocyclic Compounds Utilizing
N, from the Roots of Panax ginseng. 2451
Characteristic Bonding Properties of Hypervalent Sulfur.
Hirose, Tetsushi.
1239
Violides N-P, New Briarane Diterpenes from a Gorgona-
Hayashi, Kazuhiko.
cean briareum Sp. 1789
Improved Synthesis of an Energetic Material, 1,3,3-
Hirose, Tomoyasu.
Trinitroazetidine Exploiting 1-Azabicyclo[1.1.0]butane.