Heterocycles an International Journal for Reviews and Communications in Heterocyclic Chemistry 1996: Vol 42 Index

23 Pages·1996·5 MB·English

HETEROCYCLES, Vol. 42, No. 2, 1996
Author Index Ando, Akira.
Volume 42, 1996 Synthesis of Fluorine Analogs of Natural Porphyrins
Potentially Useful for Diagnosis and Therapy of Cancer.
885
Aoyama, Toyohiko.
Reaction of Lithium Trimethylsilyldiazomethane with N,N-
Dialkylamides of a-Keto Acids and N,N-Disubstituted a-
Amino Ketones. 75
Arai, Toshie.
Biotransformation of Phenyl- and Pyridylalkane
Derivatives in Rat Liver 9,000xg Supernatant (S-9). 831
Atta-ur-Rahman.
Abbas, Samina. Withania somnifera - a Source of Exotic Withanolides.
Withania somnifera - a Source of Exotic Withanolides. 555
555 Azuma, Yutaka.
Abe, Takao. A Carbon-Carbon Bond Formation by the Reaction of 4-
A Facile Synthesis of B-Lactams by the Cyclization of B- Chloro-6-methy!-3-phenylethynyl-2H-pyran-2-one with
Amino Acids Exploiting 3,3'-(Phenylphosphory!)-bis(1,3- Active Methylene Derivatives. 789
thiazolidine-2-thione). 849
Achiwa, Kazuo.
Lipase AH-Catalyzed Asymmetric Synthesis of (S)-(-)-NB
818. 169
Aihara, Minako. B
Neighboring Assistance of a Hydroxyl Group on
Manganese Dioxide Oxidation of Benzyl Alcohols to Balzarini, Jan.
Lactones. 589 Synthesis, Conformation Analysis and Biological
Aikawa, Maki. Evaluation of 2-(5-Deoxy-f-D-ribofuranosyl)pyridine-4-
Diels-Alder Reaction of the Dihydropyridinones V : carboxamide. 173
Approach to the Ircinal B Core. 677 Bandoh, Hiroshi.
Aimi, Norio. An Asymmetric Synthesis of the Ant Venom Alkaloid
Stereochemical Assignment of Pseudoindoxy! Alkaloids. (3S,5S,8aR)-3-Butyl-5-(4-pentenyl)indolizidine via the
87 Sharpless Asymmetric Dihydroxylation. 39
Akai, Shuji. Bernath, Gabor.
Preparation of Novel Cyclic Hypervalent lodine(IIl) tert-Butylcyclopentane Derivatives. Part 8. Synthesis of
Compounds Having Azido, Cyano, and Nitrato Ligands. tert-Butylcyclopentane-fused Pyrimidin-4-ones. 625
47 Berova, Nina.
Akamatsu, Susumu. Synthesis of Philanthotoxin Analogs with Bulky Heads
Synthesis of Tricyclic Nitrogen-containing Heterocycles Including Porphyrins. Self-assembly Monitored by
by Palladium-catalyzed Cyclization of 2-Alkenyl-N-(o- Circular Dichroism. 723
iodobenzoyl)- and 2-Alkenyl-N-(o-iodophenylacetyl)- Billimoria, Adil D.
pyrrolidines. 155 Indoloquinazolines: A Century in Review. 453
Alderweireldt, Frank C. Bohsako, Akemi.
Synthesis, Conformation Analysis and Biological Importance of the Hydroxymethyl-quinuclidine Fragment
Evaluation of 2-(5-Deoxy-f-D-ribofuranosy|)pyridine-4- in the Catalytic Asymmetric Aldol Reactions Utilizing
carboxamide. 173 Quaternary Ammonium Fluorides Derived from Cinchona
Ali, Mohamed Ayman. Alkaloids. 93
Diels-Alder Reaction of the Dihydropyridinones V : Brossi, Arnold.
Approach to the Ircinal B Core. 677 Practical Total Syntheses of Physostigmines and of
Ando, Akira. Phenserines : A Synopsis. 229
Importance of the Hydroxymethyl-quinuclidine Fragment
in the Catalytic Asymmetric Aldo! Reactions Utilizing
Quaternary Ammonium Fluorides Derived from Cinchona
Alkaloids. 93
HETEROCYCLES, Vol. 42, No. 2, 1996
c Hydrolysis of Ilsomeric Tricyclic Orthoesters and AM1
Molecular Modelling of the Reaction Pathway. Further
Carroll, Anthony R. Evidence for Stereoelectronic Control. 617
Briarane Diterpenes from Micronesian Gorgonians. 325 Dockner, Michael.
Cava, Michael P. Versatile Synthesis of Enantiomerically Pure trans-2,5-
Indoloquinazolines: A Century in Review. 453 Disubstituted Pyrrolidines. 529
Cheng, Dai. Doi, Kazuyuki.
a-Amino Ketone Synthesis from Aldehydes and N-(a- Short Step Synthesis of 4-Substituted Indoles Using
Dialkylaminoalky!l)benzotriazoles. 273 Palladium-catalyzed C-C Bond Forming Reaction. 113
Chiaroni, Angéle. Doll, Martin K.-H.
Tandem Stereoselective Conjugate Additions to a,B- Tenuilobine - A New Polyamine Alkaloid from Oncinotis
Unsaturated Oxazolines. 635 tenuiloba. 319
Choshi, Tominari . Dory, Yves L.
A Convenient Route to the Imidazo[4,5-b]pyridines. 213 Hydrolysis of lsomeric Tricyclic Orthoesters and AM1
Choudhary, M. Iqbal Molecular Modelling of the Reaction Pathway. Further
Withania somnifera - a Source of Exotic Withanolides. Evidence for Stereoelectronic Control. 617
555 Du, Xinyao.
Cummings, Maxwell D. Biotransformation of Dibenzylbutanolides by Peroxidase
B-Lactamase Inhibitors: Synthesis and in vitro Evaluation Enzymes. Routes to the Podophyllotoxin Family. 479
of 6-[(1-Substituted 1,2,3-Triazol-4-yl)methylene]-
penicillanic Acid Sulfones. 653
Czajkowski, David P.
B-Lactamase Inhibitors: Synthesis and in vitro Evaluation
of 6-[(1-Substituted 1,2,3-Triazol-4-yl)methylene]-
penicillanic Acid Sulfones. 653 Eby, Paul.
B-Lactamase Inhibitors: Synthesis and in vitro Evaluation
of 6-[(1-Substituted 1,2,3-Triazol4-yl)methylene]-
penicillanic Acid Sulfones. 653
Egi, Masahiro.
D Preparation of Novel Cyclic Hypervalent lodine(III)
Compounds Having Azido, Cyano, and Nitrato Ligands.
Dahuron, Nathalie. 47
Tandem Stereoselective Conjugate Additions to «,- Eguchi, Shoji.
Unsaturated Oxazolines. 635 Heterocyclization of 5-Trifluoroacetyltricyclo[4.3.1 13,8).
Date, Tadamasa. undecan-4-one to Some 6- and 7-Membered Nitrogen
Synthesis of Aminobenzo[b]pyrrolizinone and Amino- Heterocycles. 333
benzo[b]indolizinone Derivatives. 251 Endo, Katsuya.
Dauben, William G. Neighboring Assistance of a Hydroxyl Group on
Yoshio Ban (1921-1994) Ambassador for Japanese Manganese Dioxide Oxidation of Benzy! Alcohols to
Chemistry. 21 Lactones. 589
De Bruyn, André. Endoh, Masaki.
Synthesis, Conformation Analysis and Biological Alkoxylation at Meta Position to Hydroxyl Group of L-
Evaluation of 2-(5-Deoxy-B-D-ribofuranosyl)pyridine-4- Tyrosine: Preparation of Alkyl (S)-2,4-Dialkoxyphenyl-
carboxamide. 173 alaninates. 445
De Clercaq, Erik. Esmans, Eddy L.
Synthesis, Conformation Analysis and Biological Synthesis, Conformation Analysis and Biological
Evaluation of 2-(5-Deoxy-B-D-ribofuranosy!)pyridine-4- Evaluation of 2-(5-Deoxy-f-D-ribofuranosyl)pyridine-4-
carboxamide. 173 carboxamide. 173
De Groot, Alex.
Synthesis, Conformation Analysis and Biological
Evaluation of 2-(5-Deoxy-B-D-ribofuranosyl)pyridine-4-
carboxamide. 173
Desiongchamps, Pierre.
HETEROCYCLES, Vol. 42, No. 2, 1996
tert-Butylcyclopentane-fused Pyrimidin-4-ones. 625
Fredenburgh, Laura E. Furukawa, Hiroshi.
New Approach to the Imidazolutidine Moiety of MK-996. Two New Bisacridone Alkaloids from Citrus Plants. 237
821 Furukawa, Naomichi.
Fuji, Kaoru. Highly Diastereoselective Oxidation of 1-Alkylsulfinyl-9-
Ring Opening of Optically Active cis-Disubstituted (alkylthio)dibenzothiophene with MCPBA in the Presence
Aziridino Alcohols: An Enantiodivergent Synthesis of of Trifluoroboran Etherate. 71
Functionalized Amino Alcohol Derivatives. 701
Fuji, Kaoru.
Asymmetric Syntheses of (-)-Aphanorphine and (-)-
Eptazocine. 811
Fujii, Tozo. G
Synthesis of L-Phenylalanine Derivatives Containing a
Sulfur Substituent at the 2-Position. 219 Gao, Lian-xun.
Fujimoto, Katsuhiko. Total Synthesis of (-)-Dactylynes. 745
Enantioselective [2,3]-Wittig Rearrangement via a Chiral Ge, Wei-Ying.
Boron Ester Enolate. 423 High Pressure Mediated Asymmetric Diels-Alder Reaction
Fujimoto, Katsuhiro. of Chiral Sulfinylacrylate Derivatives with Furan and 2-
Synthesis of Fused Pyrimidinones by Reaction of Amino- Methoxyfuran. 129
arenecarboxamide with Esters; Preparation of Pyrrolo- Greig, Nigel H.
[2,3-d]-, Thieno[2,3-d]-, lsoxazolo[5,4-d]-, and 1,2,3- Practical Total Syntheses of Physostigmines and of
Triazolo[4,5-d]pyrimidinones, and Quinazolones. 691 Phenserines A Synopsis. 229
Fujioka, Haruto.
A New Bis(zinc(Il)-cyclen) Complex as a Novel Chelator Guggisberg, Armin.
for Barbiturates and Phosphates. 775 Tenuilobine - A New Polyamine Alkaloid from Oncinotis
Fujita, Hirotake. tenuiloba. 319
New Anionic Cyclization of 4- and 5-Alkynylamines :
Synthesis of 2-Benzylidene Pyrrolidines and Piperidines.
385
Fukai, Toshio.
Variations in the Chemical Shift of Benzylic Methylene H
Carbon of Prenyl Group on Heterocyclic Prenylphenols.
911 Hachiya, Shun-ichiro.
Fukai, Yuki. Synthetic Studies of Halichondrin B, an Antitumor
Effect of Bromides on the Anomalous Photoarylation of Polyether Macrolide Isolated from a Marine Sponge 5.
5-Halo-1,3-dimethyluracils. 341 A Highly Concise and Efficient Synthesis of the Cq7~Cs54
Fukui, Hideto. Tricyclic JKL-Ring Part. 99
Total Synthesis of Mycalamide A. Further Synthetic Study Hamanaka, Nobuyuki.
of the Right Half. 159 Novel Nonprostanoid Prostacyclin (PGI) Mimetics with
Fukui, Naoko. Heterocyclic Moiety. 517
Asymmetric Pictet-Spengler Reaction Using «-Methy!- Hamann, Mark T.
benzylamine as a Chiral Auxiliary Group. 347 Briarane Diterpenes from Micronesian Gorgonians. 325
Fukui, Naoko. Hara, Hiroshi.
Diels-Alder Reaction of the Dihydropyridinones V : Alkoxylation at Meta Position to Hydroxyl Group of L-
Approach to the Ircinal B Core. 677 Tyrosine: Preparation of Alkyl! (S)-2,4-Dialkoxyphenyl-
Fukumoto, Keiichiro. alaninates. 445
Cyclobutane Strategy for the Synthesis of A-Ring Harada, Kazuho.
Aromatic Trichothecanes. 165 Synthesis of Novel Heterocycle-fused Furo[3,4-d]-
Fukumoto, Keiichiro. isoxazoles via Ring Transformation of 2-lsoxazoline-2-
The Synthesis of 1B-Fluorocarbapenem Derivative. oxides by Lewis Acid. 289
437 Harada, Kenichi.
Fulép, Ferenc. A Convenient Route to the Imidazo[4,5-b]pyridines. 213
tert-Butylcyclopentane Derivatives. Part 8. Synthesis of Harrison, Karl N.
HETEROCYCLES, Vol. 42, No. 2, 1996
Briarane Diterpenes from Micronesian Gorgonians. 325 An Enantioconvergent Construction of the Key
Hasegawa, Kazushi. Intermediate of (+)-Vincamine. 65
A Microwave-accelerated Intramolecular Diels-Alder Hiyama, Tamejiro.
Reaction. Approach to Compactin. 525 Synthesis of 5-Substituted Pyrimidine Nucleosides
Hashimoto, Kimiko. through a Palladium-catalyzed Cross-Coupling of
The Mechanism of Configuration Retention in the Alkenylhalosilanes. 375
Substitution Reaction of C4-Tosyloxyproline with Lithium Honda, Toshio.
Diarylcuprate. 489 Chiral Synthesis of Phosphodiesterase Inhibitor, (A)-(-)-
Hashimoto, Masaru. Rolipram, by Means of Enantioselective Deprotonation
One-Step Synthesis of (-)-5-epi-Hydantocidin. 503 Strategy. 109
Hashimoto, Shun-ichi. Hongo, Takahiko.
A Mild and Rapid Glycosylation Reaction between Biotransformation of Phenyl- and Pyridylalkane
Pyrimidine Bases and 2-Deoxyribofuranosy! N, N, N’, N’- Derivatives in Rat Liver 9,000xg Supernatant (S-9). 831
Tetramethylphosphoroamidates. 485 Horita, Kiyoshi.
Hashimoto, Shun-ichi. Synthetic Studies of Halichondrin B, an Antitumor
Dirhodium(Il) Tetrakis[3(S)-phthalimido-2-piperidinonate]: Polyether Macrolide Isolated from a Marine Sponge 5.
A Novel Dirhodium(Il) Carboxamidate Catalyst for A Highly Concise and Efficient Synthesis of the Cq7~Cs4
Asymmetric Cyclopropanation. 537 Tricyclic JKL-Ring Part. 99
Hatanaka, Yasuo. Hoshino, Osamu.
Synthesis of 5-Substituted Pyrimidine Nucleosides Alkoxylation at Meta Position to Hydroxy! Group of L-
through a Palladium-catalyzed Cross-Coupling of Tyrosine: Preparation of Alky! (S)-2,4Dialkoxyphenyl-
Alkenylhalosilanes. 375 alaninates. 445
Hatta, Taizo. Hosomi, Akira.
Cycloaddition Reactions of Methacryloy! lsocyanate with Diastereomeric Preparation of a- and B-Phenylthio
Arylideneamines. 533 Substituted N-Acylpyrazoles. 241
Hesse, Manfred. Hosono, Shigeru.
Tenuilobine - A New Polyamine Alkaloid from Oncinotis Rare Earth Salts Promoted Glycosidation of Glycosyl
tenuiloba. 319 Fluorides. 795
Hibino, Satoshi. Hosoya, Takamitsu.
A Convenient Route to the Imidazo[4,5-b]pyridines. 213 Total Syntheses of BE-12406 A and Its C(8)-Vinyl Analog.
Higashino, Takeo. 397
Synthesis of Fused Pyrimidinones by Reaction of Amino- Huang, Danwen.
arenecarboxamide with Esters; Preparation of Pyrrolo- Synthesis of Philanthotoxin Analogs with Bulky Heads
[2,3-d]-, Thieno[2,3-q]-, lsoxazolo[5,4-a]-, and 1,2,3- Including Porphyrins. Self-assembly Monitored by
Triazolo[4,5-d]pyrimidinones, and Quinazolones. 691 Circular Dichroism. 723
Hino, Tohru. Humphrey, Guy.
Professor Yoshio Ban (1921-1994). 23 New Approach to the Imidazolutidine Moiety of MK-996.
Hino, Tohru. 821
Asymmetric Pictet-Spengler Reaction Using a-Methy!- Hutchings, Richard.
benzylamine as a Chiral Auxiliary Group. 347 Asymmetric Dialkylation of Chiral 2-Benzazepine
Hino, Tohru. Formamidines. 475
Diels-Alder Reaction of the Dihydropyridinones V : Hyodo, Akio.
Approach to the Ircinal B Core. 677 Synthesis and Biological Evaluation of Sodium 28-[(2,5-
Hiramatsu, Hajime. Dihydro-6-hydroxy-2-methyl-5-oxo-1,2,4-triazin-3-yl)-
Synthesis of Aminobenzo[b]pyrrolizinone and Amino- sulfonylmethy|]-2a-methylpenam-3a-carboxylate 1,1-
benzo[b]indolizinone Derivatives. 251 Dioxide. 645
Hirao, Ken-ichi.
Preparation of Optically Active 8,8'-Disubstituted 1,1'-
Biisoquinoline. 415
Hirota, Kosaku.
Synthesis and DNA Photo-cleaving Activity of Novel
Heterocyclic N-Oxide - Acridine Hybrid Molecules. 31
Hiroya, Kou. Ihara, Masataka.
HETEROCYCLES, Vol. 42, No. 2, 1996
The Synthesis of 1B-Fluorocarbapenem Derivative. 437 Reaction of Vinylcyclopropanes. 565
limori, Takamasa. Ishibashi, Masami.
A Mild and Rapid Glycosylation Reaction between Sphingosine-related Marine Alkaloids: Cyclic Amino
Pyrimidine Bases and 2-Deoxyribofuranosyl N, N, N', N’- Alcohols. 943
Tetramethylphosphoroamidates. 485 Ishibuchi, Seigo.
Ikeda, Masazumi. Synthetic Application of Chiral 4-Methoxy-2-oxazolidinone
Synthesis of Tricyclic Nitrogen-containing Heterocycles Synthons to 2-Amino Alcohols of Biological Interest. 837
by Palladium-catalyzed Cyclization of 2-Alkenyl-N-(o- Ishida, Yohhei.
iodobenzoyl)- and 2-Alkenyl-N-(o-iodophenylacetyl)- The Synthesis of 1B-Fluorocarbapenem Derivative. 437
pyrrolidines. 155 Ishikawa, Fumihiro.
Ikegami, Shiro. Chiral Synthesis of Phosphodiesterase Inhibitor, (A)-(-)-
A Mild and Rapid Glycosylation Reaction between Rolipram, by Means of Enantioselective Deprotonation
Pyrimidine Bases and 2-Deoxyribofuranosy! N, N, N', N’- Strategy. 109
Tetramethylphosphoroamidates. 485 Ishizaki, Michiyo.
Ikota, Nobuo. An Enantioconvergent Construction of the Key
Theoretical Calculation-based Reproduction of Intermediate of (+)-Vincamine. 65
Thermodynamic, Kinetic Behaviors and Cytotoxicity of Ishizuka, Tadao.
Azasteganes. 43 Synthetic Application of Chiral 4-Methoxy-2-oxazolidinone
Imanishi, Takeshi. Synthons to 2-Amino Alcohols of Biological Interest. 837
Novel Indole-Ring Construction Method for the Synthesis Ito, Chihiro.
of 2-Trifluoromethylindoles. 513 Two New Bisacridone Alkaloids from Citrus Plants.
Imasho, Masaaki. 237
Synthesis of L-Phenylalanine Derivatives Containing a Ito, Katsuji.
Sulfur Substituent at the 2-Position. 219 Enantiospecific Ring Expansion of Oxetanes:
Imazato, Hitoshi. Stereoselective Synthesis of Tetrahydrofurans. 305
Asymmetric Syntheses of (-)-Aphanorphine and (-)- Ito, Yoshihiko.
Eptazocine. 811 New Synthesis of Quinoxaline Derivatives Based on
Inamoto, Masayuki. Palladium Catalyzed Oligomerization of 1,2-
Studies on Organometallic Compounds. IX. Synthesis of Diisocyanoarenes. 597
Bipyridine N-Oxides and Terpyridines by Palladium Iwai, Sakiko.
Catalyzed Cross-Coupling Reaction of Trimethylstanny|- Biotransformation of Phenyl- and Pyridylalkane
pyridines with Bromopyridines. 189 Derivatives in Rat Liver 9,000xg Supernatant (S-9). . 831
Inoue, Isao. Iwata, Chuzo.
Synthesis of Aminobenzo[b]pyrrolizinone and Amino- Reaction of 3-Aralkylsulfony!-2-(N-cyanoimino)-
benzo[b]indolizinone Derivatives. 251 thiazolidines with Oxygen Nucleophiles. 265
Inoue, Shoji.
(S)-2-Methyl-1 ,5-bis(1,3-dimethy|-6-lumazinyl)-1,5-
pentanedione from the Marine Polychaete, Odontosyllis
undecimdonta. 125
Inoue, Takehisa.
Asymmetric Syntheses of (-)-Aphanorphine and (-)-
Eptazocine. 811 Jamal, S. Arshad.
Inoue, Tsutomu. Withania somnifera - a Source of Exotic Withanolides.
Alkoxylation at Meta Position to Hydroxy! Group of L- 555
Tyrosine: Preparation of Alky! (S)-2,4-Dialkoxyphenyl- Joos, Pieter E.
alaninates. 445 Synthesis, Conformation Analysis and Biological
Inoue, Yoshinori. Evaluation of 2-(5-Deoxy-f-D-ribofuranosyl)pyridine-4-
A Facile Synthesis of B-Lactams by the Cyclization of B- carboxamide. 173
Amino Acids Exploiting 3,3'-(Phenylphosphoryl)-bis(1,3- Ju-ichi, Motoharu.
thiazolidine-2-thione). 849 Two New Bisacridone Alkaloids from Citrus Plants. 237
Isaka, Masahiko.
Carbometalation of Cyclopropenes. Stereoselective
Synthesis of Diviny! Ketones via 1,5-Hydrogen Migration
HETEROCYCLES, Vol. 42, No. 2, 1996
Ring Opening of Optically Active cis-Disubstituted
K Aziridino Alcohols: An Enantiodivergent Synthesis of
Functionalized Amino Alcohol Derivatives. 701
Kageyama, Akiko. Kawaguchi, Takayuki.
Diels-Alder Reaction of the Dihydropyridinones V: Synthesis of Aminobenzo[b]pyrrolizinone and Amino-
Approach to the Ircinal B Core. 677 benzo[b]indolizinone Derivatives. 251
Kaji, Eisuke. Kawano, Yoshikazu.
Synthesis of Novel Heterocycle-fused Furo[3,4-d]- Asymmetric Syntheses of (-)-Aphanorphine and (-)-
isoxazoles via Ring Transformation of 2-lsoxazoline-2- Eptazocine. 811
oxides by Lewis Acid. 289 Kawasaki, Toshiya.
Kajiwara, Masahiro. The First and Simple Synthesis of Indole Alkaloid,
A Microwave-accelerated Intramolecular Diels-Alder Bipolaramide. 281
Reaction. Approach to Compactin. 525 Kawate, Tomohiko.
Kakoi, Hisae. Asymmetric Pictet-Spengler Reaction Using a-Methyl-
(S)-2-Methyl-1,5-bis(1,3-dimethy!-6-lumaziny!)-1,5- benzylamine as a Chiral Auxiliary Group. 347
pentanedione from the Marine Polychaete, Odontosyllis Kiguchi, Toshiko.
undecimdonta. 125 Syntheses of Proposed Structure of Pseudodistomin A
Kanai, Kazuo. Triacetate and Its Regioisomers on Dieny! Side-Chain.
Chiral Synthesis of Phosphodiesterase Inhibitor, (A)-(-)- 509
Rolipram, by Means of Enantioselective Deprotonation Kim, Won-Sup.
Strategy. 109 Rare Earth Salts Promoted Glycosidation of Glycosyl
Kanai, Motomu. Fluorides. 795
Theoretical Calculation-based Reproduction of Kimura, Eiichi.
Thermodynamic, Kinetic Behaviors and Cytotoxicity of A New Bis(zinc(Il)-cyclen) Complex as a Novel Chelator
Azasteganes. 43 for Barbiturates and Phosphates. 775
Kanaoka, Yuichi. Kimura, Takeshi.
Professor Yoshio Ban (1921-1994). 23 Highly Diastereoselective Oxidation of 1-Alkylsulfinyl-9-
Kanaoka, Yuichi. (alkyithio)dibenzothiophene with MCPBA in the Presence
Chemical Identification of Binding Sites for Calcium of Trifluoroboran Etherate. 71
Channel Antagonists. 901 Kirihara, Masayuki.
Kaneko, Chikara. One-Step Synthesis of (-)-5-ep#Hydantocidin. 503
Conformation and Facial Selectivities of Chiral Six- Kiryu, Yoshimitsu.
membered 1,3-Diheterocycles Involving an Enone Ring Opening of Optically Active cis-Disubstituted
‘Function. 861 Aziridino Alcohols: an Enantiodivergent Synthesis of
Kanzaki, Ryouichi. Functionalized Amino Alcohol Derivatives. 701
Cycloaddition Reactions of Methacryloy! Isocyanate with Kita, Yasuyuki.
Arylideneamines. 533 Preparation of Novel Cyclic Hypervalent lodine(III)
Kashima, Choji. Compounds Having Azido, Cyano, and Nitrato Ligands.
Diastereomeric Preparation of «- and B-Phenylthio 47
Substituted N-Acylpyrazoles. 241 Kitahara, Yoshiyasu.
Kato, Daishiro. A Synthesis of the Derivatives of 1,2,3,5,10,10a-
Chiral Synthesis of Phosphodiesterase Inhibitor, (A)-(-)- Hexahydrobenz[flindolizine-6,9-dione Having Antifungal
Rolipram, by Means of Enantioselective Deprotonation Activity as a Simple Model of Saframycin A. 195
Strategy. 109 Kitajima, Mariko.
Katoh, Tadashi. Stereochemical Assignment of Pseudoindoxy! Alkaloids.
One-Step Synthesis of (-)-5-epi-Hydantocidin. 503 87
Katritzky, Alan R. Kobayashi, Hiroshi.
a-Amino Ketone Synthesis from Aldehydes and N-(c- A Mild and Rapid Glycosylation Reaction between
Dialkylaminoalky!)benzotriazoles. 273 Pyrimidine Bases and 2-Deoxyribofuranosyl N, N, N', N-
Katsuki, Tsutomu. Tetramethylphosphoroamidates. 485
Enantiospecific Ring Expansion of Oxetanes: Kobayashi, Junichi.
Stereoselective Synthesis of Tetrahydrofurans. 305 Sphingosine-related Marine Alkaloids: Cyclic Amino
Kawabata, Takeo. Alcohols. 943
HETEROCYCLES, Vol. 42, No. 2, 1996
Kobayashi, Toshiyuki. A Synthesis of the Derivatives of 1,2,3,5,10,10a-
Cycloaddition Reactions of Methacryloyl Ilsocyanate with Hexahydrobenz[flindolizine-6,9-dione Having Antifungal
Arylideneamines. 533 Activity as a Simple Model of Saframycin A. 195
Koga, Hiroshi. Kubota, Hideki.
Practical Radical Deoxygenation of Erythromycins by Enantioselective Allylic Alkylation and Amination
Barton Reaction. 499 Catalyzed by a Chiral P/N Ligand-Palladium Complex.
Koga, Kenji. 543
Enantioselective Allylic Alkylation and Amination Kubota, Katsumi.
Catalyzed by a Chiral P/N Ligand-Palladium Complex. Carbometalation of Cyclopropenes. Stereoselective
543 Synthesis of Divinyl Ketones via 1,5-Hydrogen Migration
Kohno, Harumichi. Reaction of Vinylcyclopropanes. 565
A Novel Cyclization of Electron Deficient N-Benzene- Kugo, Yasuhiro.
sulfonyl-B-phenethylamines Using Ethy! Chloro- Synthesis of Tricyclic Nitrogen-containing Heterocycles
(methylthio)acetate. Synthesis of Ethyl 1,2,3,4- by Palladium-catalyzed Cyclization of 2-Alkenyl-N-(o-
Tetrahydroisoquinoline-1-carboxylates. 141 iodobenzoyl)- and 2-Alkeny|-N-(o-iodophenylacetyl)-
Koike, Tohru. pyrrolidines. 155
A New Bis(zinc(Il)-cyclen) Complex as a Novel Chelator Kumadaki, Itsumaro.
for Barbiturates and Phosphates. 775 Synthesis of Fluorine Analogs of Natural Porphyrins
Koizumi, Toru. Potentially Useful for Diagnosis and Therapy of Cancer.
High Pressure Mediated Asymmetric Diels-Alder Reaction 885
of Chiral Sulfinylacrylate Derivatives with Furan and 2- Kumagai, Toshio.
Methoxyfuran. 129 A Facile Synthesis of B-Lactams by the Cyclization of B-
Koizumi, Yuichi. Amino Acids Exploiting 3,3'-(Phenylphosphoryl)-bis(1,3-
A Synthesis of the Derivatives of 1,2,3,5,10,10a- thiazolidine-2-thione). 849
Hexahydrobenz[flindolizine-6,9-dione Having Antifungal Kunieda, Takehisa.
Activity as a Simple Mode! of Saframycin A. 195 Synthetic Application of Chiral 4-Methoxy-2-oxazolidinone
Kojima, Naoshi. Synthons to 2-Amino Alcohols of Biological Interest. 837
Nucleosides and Nucleotides. 138. Synthesis of 3-Halo-3- Kunugita, Chieko.
deazainosines: Conformational Lock with the Halogen at Synthesis and Biological Evaluation of Sodium 2-{(2,5-
the 3-Position of the 3-Deazainosine in anti- Dihydro-6-hydroxy-2-methyl-5-oxo-1 ,2,4-triazin-3-yl)-
Conformation. 149 sulfonylmethy!]-2a-methylpenam-3a-carboxylate 1,1-
Kojima, Yutaka. Dioxide. 645
New Synthesis of Quinoxaline Derivatives Based on Kuribayashi, Harumi.
Palladium Catalyzed Oligomerization of 1,2- Dirhodium(I!) Tetrakis[3(S)-phthalimido-2-piperidinonate]:
Diisocyanoarenes. 597 A Novel Dirhodium(Il) Carboxamidate Catalyst for
Kondo, Kigen. Asymmetric Cyclopropanation. 537
Novel Nonprostanoid Prostacyclin (PGlp) Mimetics with Kurihara, Mika.
Heterocyclic Moiety. 517 Stereochemical Assignment of Pseudoindoxy! Alkaloids.
Kondo, Yoshinori. 87
Halogen-Magnesium Exchange Reaction of lodoindole Kuroboshi, Manabu.
Derivatives. 105 Synthesis of 5-Substituted Pyrimidine Nucleosides
Kondoh, Katsunori. through a Palladium-catalyzed Cross-Coupling of
Novel Indole-Ring Construction Method for the Synthesis Alkenylhalosilanes. 375
of 2-Trifluoromethylindoles. 513 Kurosaki, Ryuichi.
Konopski, Leszek. Asymmetric Syntheses of (-)-Aphanorphine and (-)-
Synthesis and Stereochemistry of 2-Methyl-4H-912,- Eptazocine. 811
dioxa-1 ,4-diazadispiro[5.2.5.2]tetradec-1-en-3-one and Kutney, James P.
Its 2H-Imidazolo-2-spirocyclohexane Analogue. Biotransformation of Dibenzylbutanolides by Peroxidase
An Anomalous Michael Type Cyclocondensation. 737 Enzymes. Routes to the Podophyllotoxin Family. 479
Kosaka, Kazuhiro.
Biotransformation of Phenyl- and Pyridylalkane
Derivatives in Rat Liver 9,000xg Supernatant (S-9). 831
Kubo, Akinori.
HETEROCYCLES, Vol. 42, No. 2, 1996
L penicillanic Acid Sulfones. 653
Maki, Yoshifumi.
Langlois, Nicole. Synthesis and DNA Photo-cleaving Activity of Novel
Tandem Stereoselective Conjugate Additions to a,B- Heterocyclic N-Oxide - Acridine Hybrid Molecules. 31
Unsaturated Oxazolines. 635 Maruno, Masao.
Langlois, Yves. Total Synthesis of the Major Metabolites of Gomisin A.
Synthesis and Stereochemistry of 2-Methyl-4H-192,- Synthesis of Homochiral Met A-ll, Met A-lll, Met D, and
dioxa-1 ,4-diazadispiro[5.2.5.2]tetradec-1-en-3-one and Met F. 359
Its 2H-Imidazolo-2-spirocyclohexane Analogue. Matile, Stefan.
An Anomalous Michael Type Cyclocondensation. 737 Synthesis of Philanthotoxin Analogs with Bulky Heads
Larsen, Robert D. Including Porphyrins. Self-assembly Monitored by
New Approach to the Imidazolutidine Moiety of MK-996. Circular Dichroism. 723
821 Matsuda, Akira.
Li, Shigui. Nucleosides and Nucleotides. 138. Synthesis of 3-Halo-3-
Hydrolysis of lsomeric Tricyclic Orthoesters and AM1 deazainosines: Conformational Lock with the Halogen at
Molecular Modelling of the Reaction Pathway. Further the 3-Position of the 3-Deazainosine in anti
Evidence for Stereoelectronic Control. 617 Conformation. 149
Liu, Hsing-Jang. Matsuda, Hideo.
Total Synthesis of (-)-Qinghaosu IV (Artemisinin D, Dirhodium(Il) Tetrakis[3(S)-phthalimido-2-piperidinonate]:
Arteannuin D). 493 A Novel Dirhodium(II) Carboxamidate Catalyst for
Liu, Ji. Asymmetric Cyclopropanation. 537
New Approach to the Imidazolutidine Moiety of MK-996. Matsuhashi, Chiho.
821 Enantioselective [2,3]-Wittig Rearrangement via a Chiral
Lu, Bao-yuan. Boron Ester Enolate. 423
Practical Total Syntheses of Physostigmines and of Matsuhashi, Hayao.
Phenserines : A Synopsis. 229 Synthesis of 5-Substituted Pyrimidine Nucleosides
through a Palladium-catalyzed Cross-Coupling of
Alkenylhalosilanes. 375
Matsukura, Hiroko.
Total Synthesis of Mycalamide A. Further Synthetic Study
of the Right Half. 159
Matsumoto, Miyoko.
Machida, Minoru. One-Step Synthesis of (-)-5-ep+#Hydantocidin. 503
Intramolecular Photoreaction of Thiobarbiturates with an Matsumoto, Takashi.
Alkeny! Group in Their N-Side Chain. Regioselective Total Syntheses of BE-12406 A and Its C(8)-Vinyl Analog.
Synthesis of Fused Pyrimidine Derivatives through 397
Photocycloaddition of Mono- and Dithiobarbiturates. Matsunaga, Hiroshi.
117 A Facile Synthesis of B-Lactams by the Cyclization of B-
Machida, Minoru. Amino Acids Exploiting 3,3'-(Phenylphosphoryl)-bis(1,3-
Photoreaction of Thiobenzamide with 2-Vinylfuran thiazolidine-2-thione). 849
Analogues. Facile Synthesis of Tetracyclic Indole System Matsutani, Takafumi.
121 Synthesis of N.2',3',5'-Tetrabenzoyl-f-D-adenosine
Maekawa, Kaori. Catalyzed by Metal lodides. 57
Reaction of 3-Aralkylsulfony|-2-(N-cyanoimino)- Meyers, A. I.
thiazolidines with Oxygen Nucleophiles. 265 Asymmetric Dialkylation of Chiral 2-Benzazepine
Maiti, Samarendra N. Formamidines. 475
Synthesis and Biological Evaluation of Sodium 2B-{(2,5- Micetich, Ronald G.
Dihydro-6-hydroxy-2-methy|-5-oxo-1 ,2,4-triazin-3-yl)- Synthesis and Biological Evaluation of Sodium 28-[(2,5-
sulfonylmethy!]-2a-methylpenam-3a-carboxylate 1,1- Dihydro-6-hydroxy-2-methy|-5-oxo-1 ,2,4-triazin-3-yl)-
Dioxide. 645 sulfonylmethyl]-2a-methylpenam-3a-carboxylate 1,1-
Maiti, Samarendra N. Dioxide. 645
B-Lactamase Inhibitors: Synthesis and in vitro Evaluation Micetich, Ronald G.
of 6-[(1-Substituted 1,2,3-Triazol-4-yl)methylene]- $-Lactamase Inhibitors: Synthesis and in vitro Evaluation
HETEROCYCLES, Vol. 42, No. 2, 1996
of 6-[(1-Substituted 1,2,3-Triazol-4-yl)methylene]- Catalyzed by Metal lodides. 57
penicillanic Acid Sulfones. 653 Murai, Akio.
Mikami, Yuzuru. Total Synthesis of (-)-Dactylynes. 745
A Synthesis of the Derivatives of 1,2,3,5,10,10a- Murakami, Masahiro.
Hexahydrobenz[flindolizine-6,9-dione Having Antifungal New Synthesis of Quinoxaline Derivatives Based on
Activity as a Simple Model of Saframycin A. 195 Palladium Catalyzed Oligomerization of 1,2-
Minakawa, Noriaki. Diisocyanoarenes. 597
Nucleosides and Nucleotides. 138. Synthesis of 3-Halo-3- Murakami, Yasuoki.
deazainosines: Conformational Lock with the Halogen at Synthetic Studies of 1,2,3,4-Tetrahydro-1,3,4-trioxo-B-
the 3-Position of the 3-Deazainosine in anti- carboline Alkaloids |. 83
Conformation. 149 Murata, Yoshinori.
Mitsuhashi, Hiroshi. Aprotic Chloride and Bromide-promoted Alkyne-Iminium
Total Synthesis of the Major Metabolites of Gomisin A. lon Cyclizations. 549
Synthesis of Homochiral Met A-Il, Met A-Ill, Met D, and Musgrave, Richard P.
Met F. 359 a-Amino Ketone Synthesis from Aldehydes and N-(a-
Miura, Masatomo. Dialkylaminoalkyl)benzotriazoles. 273
Biotransformation of Phenyl- and Pyridylalkane
Derivatives in Rat Liver 9,000xg Supernatant (S-9). 831
Miyabe, Hideto.
Novel Indole-Ring Construction Method for the Synthesis
of 2-Trifluoromethylindoles. 513 N
Miyashita, Akira.
Synthesis of Fused Pyrimidinones by Reaction of Amino- Nagai, Masashi.
arenecarboxamide with Esters; Preparation of Pyrrolo- Synthesis of N._2',3',5'-Tetrabenzoyl-f-D-adenosine
[2,3-d]-, Thieno[2,3-d]-, lsoxazolo[5,4-d]-, and 1,2,3- Catalyzed by Metal lodides. 57
Triazolo[4,5-d]pyrimidinones, and Quinazolones. 691 Nagao, Yoshimitsu.
Miyashita, Kazuyuki. A Facile Synthesis of S-Lactams by the Cyclization of B-
Novel Indole-Ring Construction Method for the Synthesis Amino Acids Exploiting 3,3'-(Phenylphosphoryl)-bis(1 ,3-
of 2-Trifluoromethylindoles. 513 thiazolidine-2-thione). 849
Miyata, Junji. Nagao, Yuuki.
Cyclobutane Strategy for the Synthesis of A-Ring Novel Nonprostanoid Prostacyclin (PGI) Mimetics with
Aromatic Trichothecanes. 165 Heterocyclic Moiety. 517
Mizuguchi, Ryuzo. Nagareya, Noriko.
Cycloaddition Reactions of Methacryloy! lsocyanate with Two New Bisacridone Alkaloids from Citrus Plants. 237
Arylideneamines. 533 Nagasawa, Masaaki.
Momose, Takefumi. Synthetic Studies of Halichondrin B, an Antitumor
An Asymmetric Synthesis of the Ant Venom Alkaloid Polyether Macrolide Isolated from a Marine Sponge 5.
(3S,5S,8aR)-3-Butyl-5-(4-pentenyl)indolizidine via the A Highly Concise and Efficient Synthesis of the Cq7~C54
Sharpless Asymmetric Dihydroxyiation. 39 Tricyclic JKL-Ring Part. 99
Mori, Miwako. Naidu, Rajina.
Short Step Synthesis of 4-Substituted Indoles Using Biotransformation of Dibenzylbutanolides by Peroxidase
Palladium-catalyzed C-C Bond Forming Reaction. 113 Enzymes. Routes to the Podophyllotoxin Family. 479
Morimoto, Hiroshi. Naito, Takeaki.
Synthetic Studies of Novel 5-Azacarbapenems. 577 Syntheses of Proposed Structure of Pseudodistomin A
Morone, Mieko. Triacetate and Its Regioisomers on Dieny! Side-Chain.
A Carbon-Carbon Bond Formation by the Reaction of 4- 509
Chloro-6-methyl-3-phenylethynyl-2H-pyran-2-one with Nakagawa, Masako.
Active Methylene Derivatives. 789 Asymmetric Pictet-Spengler Reaction Using a-Methyl-
Morooka, Kohei. benzylamine as a Chiral Auxiliary Group. 347
Synthetic Application of Chiral 4-Methoxy-2-oxazolidinone Nakagawa, Masako.
Synthons to 2-Amino Alcohols of Biological Interest. 837 Diels-Alder Reaction of the Dihydropyridinones V :
Mukaiyama, Teruaki. Approach to the Ircinal B Core. 677
Synthesis of N.,2',3',5'-Tetrabenzoy|-B-0-adenosine Nakagawa, Tadakiyo.
HETEROCYCLES, Vol. 42, No. 2, 1996
Total Synthesis of Mycalamide A. Further Synthetic Study Asymmetric Syntheses of (-)-Aphanorphine and (-)-
of the Right Half. 159 Eptazocine. 811
Nakai, Takeshi. Nishihara, Chihiro.
Enantioselective [2,3]-Wittig Rearrangement via a Chiral Reaction of 3-Aralkylsulfony!-2-(N-cyanoimino)-
Boron Ester Enolate. 423 thiazolidines with Oxygen Nucleophiles. 265
Nakai, Tatsuya. Nitta, Makoto.
A Synthesis of the Derivatives of 1,2,3,5,10,10a- New Anionic Cyclization of 4- and 5-Alkynylamines :
Hexahydrobenz[flindolizine-6,9-dione Having Antifungal Synthesis of 2-Benzylidene Pyrrolidines and Piperidines.
Activity as a Simple Model of Saframycin A. 195 385
Nakajima, Noriyuki. Niwa, Sachiko.
One-Step Synthesis of (-)-5-epi-Hydantocidin. 503 Synthetic Studies of 1,2,3,4-Tetrahydro-1 ,3,4-trioxo-B-
Nakajima, Yamakoshi Yoko. carboline Alkaloids |. 83
High Pressure Mediated Asymmetric Diels-Alder Reaction Node, Manabu.
of Chiral Sulfinylacrylate Derivatives with Furan and 2- Asymmetric Syntheses of (-)-Aphanorphine and (-)-
Methoxyfuran. 129 Eptazocine. 811
Nakamoto, Yumi. Nomura, Sumihiro.
Reaction of 3-Aralkylsulfony|-2-(N-cyanoimino)- Synthesis of Aminobenzo[b]pyrrolizinone and Amino-
thiazolidines with Oxygen Nucleophiles. 265 benzo[bjindolizinone Derivatives. 251
Nakamura, Eiichi. Nomura, Taro.
Carbometalation of Cyclopropenes. Stereoselective Variations in the Chemical Shift of Benzylic Methylene
Synthesis of Divinyl Ketones via 1,5-Hydrogen Migration Carbon of Prenyl Group on Heterocyclic Prenylphenols.
Reaction of Vinylcyclopropanes. 565 911
Nakamura, Hiroshi.
Alkoxylation at Meta Position to Hydroxy! Group of L-
Tyrosine: Preparation of Alky! (S)-2,4-Dialkoxypheny!-
alaninates. 445
Nakanishi, Koji. Oo
Synthesis of Philanthotoxin Analogs with Bulky Heads
Including Porphyrins. Self-assembly Monitored by Oda, Kazuaki.
Circular Dichroism. 723 Photoreaction of Thiobenzamide with 2-Vinylfuran
Nakano, Takao. Analogues. Facile Synthesis of Tetracyclic Indole System.
Synthetic Studies of Novel 5-Azacarbapenems. 577 121
Nakata, Tadashi. Oda, Kuniyuki.
Total Synthesis of Mycalamide A. Further Synthetic Study Synthetic Studies of Novel 5-Azacarbapenems. 577
of the Right Half. 159 Ogasawara, Kunio.
Nakayama, Hidetaka. An Enantioconvergent Construction of the Key
Highly Diastereoselective Oxidation of 1-Alkylsulfinyl-9- Intermediate of (+)-Vincamine. 65
(alkylthio)dibenzothiophene with MCPBA in the Presence Ogasawara, Kunio.
of Trifluoroboran Etherate. 71 A New Synthesis of (-)-Mesembrine Employing Sharpless
Nakayama, Hitoshi. AD Reaction and New Radical-initiated Reaction. 135
Chemical Identification of Binding Sites for Calcium Ogawa, Hideki.
Channel Antagonists. 901 Reaction of Lithium Trimethylsilyldiazomethane with N,N-
Narai, Satoshi. Dialkylamides of a-Keto Acids and N,N-Disubstituted o-
A Microwave-accelerated Intramolecular Diels-Alder Amino Ketones. 75
Reaction. Approach to Compactin. 525 Ogawa, Yoshitaka.
Nemoto, Hideo. Beckmann Rearrangement of 4,5,6-Trisubstituted 3-
Cyclobutane Strategy for the Synthesis of A-Ring Acetylpyridin-2-one Oximes. 35
Aromatic Trichothecanes. 165 Ogihara, Kazuhito.
Ninomiya, Ichiya. Synthetic Studies of Halichondrin B, an Antitumor
Syntheses of Proposed Structure of Pseudodistomin A Polyether Macrolide Isolated from a Marine Sponge 5.
Triacetate and Its Regioisomers on Dieny! Side-Chain A Highly Concise and Efficient Synthesis of the C37~C54
509 Tricyclic JKL-Ring Part. 99
Nishide, Kiyoharu. Ohba, Masashi.