Biopharmaceutics and Drug Disposition 1992: Vol 13 Table of Contents

9 Pages·1992·1.8 MB·English

BIOPHARMACEUTICS & DRUG DISPOSITION
(Biopharm. drug dispos.)
CONTENTS
VOLUME 13, ISSUE NOS. 1-9 (1992)
Issue No. 1, January
Use of a Microbial Model for the Determination of Drug Effects on Cell
Metabolism and Energetics: Study of Citrulline-Malate: J. Briand,
H. Blehaut, R. Calvayrac and D. Laval-Martin .
Nonlinearities in Amoxycillin Pharmacokinetics I. Disposition Studies in
the Rat: F. Torres-Molina, J. £. Peris-Ribera, M. C. Garcia-Carbonell,
J.C. Aristorena, L. Granero and J. M. Pla-Delfina
Nonlinearities in Amoxycillin Pharmacokinetics II. Absorption Studies
in the Rat: F. Torres-Molina, J. E. Peris-Ribera, M. C. Garcia-
Carbonell, J. C. Aristorena and J. M. Pla-Delfina
Pharmacokinetics and Acetylation of Sulfa-2-Monomethoxine in
Humans: T. B. Vree, E. W. J. Beneken Kolmer, Y. A. Hekster, M.
Shimoda, M. Ono and T. Miura
Linear Pharmacokinetics of Haloperidol in the Rat: Y. F. Cheng and
L. K. Paalzow .
Issue No. 2, March
Effect of Dehydration on the Disposition Kinetics of Erythromycin in
Rabbits: M. Ahmad, S. K. Niazi, T. Ahmad, N. A. Muzaffar and
M. Nawaz
Pharmacokinetics of the Antidepressant Levoprotiline after Intravenous
and Peroral Administration in Healthy Volunteers: G. Kaiser,
R. Ackermann, W. Dieterle, 1. W. Reimann and P. R. Bieck
Methimazole Increases the Plasma Concentrations of the Albendazole
Metabolites of Netobimin in Sheep: C. E. Lanusse and R. K. Prichard
Prediction of Netilmicin Disposition in Neonates: M. Darwish,
M. Batayneh, J. Jenkins, M. Scott, P. S. Collier and J.C. McEInay
A Pharmacokinetic and Tolerance Study of Romazarit in Patients with
Rheumatoid Arthritis: P. E. O. Williams, H. A. Bird, S. Minty, P. S.
Helliwell, G. J. Muirhead, J. Bentley and A. York
Brain Regional Pharmacokinetics of Biperiden in Rats: K. Yokogawa,
E. Nakashima, J. Ishizaki, M. Hasegawa, H. Kido and F. Ichimura
BIOPHARMACEUTICS & DRUG DISPOSITION
(Biopharm. drug dispos.)
CONTENTS
VOLUME 13, ISSUE NOS. 1-9 (1992)
Issue No. 1, January
Use of a Microbial Model for the Determination of Drug Effects on Cell
Metabolism and Energetics: Study of Citrulline-Malate: J. Briand,
H. Blehaut, R. Calvayrac and D. Laval-Martin .
Nonlinearities in Amoxycillin Pharmacokinetics I. Disposition Studies in
the Rat: F. Torres-Molina, J. £. Peris-Ribera, M. C. Garcia-Carbonell,
J.C. Aristorena, L. Granero and J. M. Pla-Delfina
Nonlinearities in Amoxycillin Pharmacokinetics II. Absorption Studies
in the Rat: F. Torres-Molina, J. E. Peris-Ribera, M. C. Garcia-
Carbonell, J. C. Aristorena and J. M. Pla-Delfina
Pharmacokinetics and Acetylation of Sulfa-2-Monomethoxine in
Humans: T. B. Vree, E. W. J. Beneken Kolmer, Y. A. Hekster, M.
Shimoda, M. Ono and T. Miura
Linear Pharmacokinetics of Haloperidol in the Rat: Y. F. Cheng and
L. K. Paalzow .
Issue No. 2, March
Effect of Dehydration on the Disposition Kinetics of Erythromycin in
Rabbits: M. Ahmad, S. K. Niazi, T. Ahmad, N. A. Muzaffar and
M. Nawaz
Pharmacokinetics of the Antidepressant Levoprotiline after Intravenous
and Peroral Administration in Healthy Volunteers: G. Kaiser,
R. Ackermann, W. Dieterle, 1. W. Reimann and P. R. Bieck
Methimazole Increases the Plasma Concentrations of the Albendazole
Metabolites of Netobimin in Sheep: C. E. Lanusse and R. K. Prichard
Prediction of Netilmicin Disposition in Neonates: M. Darwish,
M. Batayneh, J. Jenkins, M. Scott, P. S. Collier and J.C. McEInay
A Pharmacokinetic and Tolerance Study of Romazarit in Patients with
Rheumatoid Arthritis: P. E. O. Williams, H. A. Bird, S. Minty, P. S.
Helliwell, G. J. Muirhead, J. Bentley and A. York
Brain Regional Pharmacokinetics of Biperiden in Rats: K. Yokogawa,
E. Nakashima, J. Ishizaki, M. Hasegawa, H. Kido and F. Ichimura
VOLUME CONTENTS
Pharmacokinetics of Nitroglycerin and its Metabolites After Adminis-
tration of Sustained-Release Tablets: H.-R. Kwon, P. Green and S. H.
Curry 5 ;
ANNOUNCEMENT .
Issue No. 3, April
Kinetic Analysis of Tissue Distribution of Doxorubicin Incorporated in
Liposomes in Rats: Part I: H. Harashima, S. Ohshima, Y. Midori, K.
Yachi, H. Kikuchi and H. Kiwada
Absence of Food Effects on the Pharmacokinetics of Terfenadine: M. G.
Eller, B. J. Walker, L. Yuh, K. K. Antony, B. E. McNutt and R. A.
Okerholm.
A General Method for Calculating the Mean Transit Times and Distri-
bution Rate Parameters of Catenary Metabolites: H. Cheng
Methylxanthine Levels in Breast Milk of Lactating Women of Different
Ethnic and Socioeconomic Classes: J. Blanchard, C. W. Weber and
L.-E. Shearer ; ; ; . ; : ; ‘ .
Pharmacokinetics of Ketoprofen in Rats: Effect of Age and Dose: J. H.
Satterwhite and F. D. Boudinot.
Pharmacokinetics of Teicoplanin Upon Multiple Dose Intravenous
Administration to Normal Healthy Male Volunteers: G. A. Thompson,
J. A. Smithers, M. T. Kenny, J. K. Dulworth, H. K. Kulmala, L. Yuh,
E. W. Lewis and K. K. Antony .
SHORT COMMUNICATIONS
Organ Distribution and Stability of Phosphorothioated Oligodeoxyribo-
nucleotides in Mice: G. Goodarzi, M. Watabe and K. Watabe
Equations for the Fraction of Bioavailable Dose Remaining in the Body
in the One-Compartment Model: P. Macheras, M. Symillides and
C. Reppas
Issue No. 4, May
Pharmacodynamics as a Tool to Assess the Bioequivalence of Non-
Systemically Available Drugs: Size of the Sample Required: P. Du
Souich, J.-G. Besner and G. Caillé
In Vitro Reduction of Rhein Anthraquinone to Rhein Anthrone by Rat
Cecal Microflora and Some Intestinal Bacterial Strains: P. De Witte,
A. Van Hoestenberghe and H. Eyssen
IV VOLUME CONTENTS
Pharmacokinetics of Ketotifen After Oral Administration to Healthy
Male Subjects: A. Grahnén, A. Loénnebo, O. Beck, S.-A. Eckernas,
B. Dahlstrom and B. Lindstr6m
A Simplified Approach for Evaluation of Hepatic Drug-Oxidizing
Activity with a Simultaneous Determination of Caffeine and Tri-
methadione and Their Demethylated Metabolites in Rats with a
Selective Cytochrome P-450 Inducer: E. Tanaka, A. Ishikawa,
Y. Yamamoto, E. Uchida, S. Kobayashi, H. Yasuhara and S. Misawa
Comparison of Disposition Behavior and De-Coppering Effect of Tri-
ethylenetetramine in Animal Model for Wilson’s Disease (Long-Evans
Cinnamon Rat) with Normal Wistar Rat: K. Iseki, M. Kobayashi,
A. Ohba, K. Miyazaki, Y. Li, Y. Togashi and N. Takeichi .
Absorption and Disposition of Fluvastatin, an Inhibitor of HMG-CoA
Reductase, in the Rabbit: F. L. S. Tse and D. Labbadia
Effect of Basic Drugs on the Hepatic Uptake of Ouabain by Sinusoidal
Plasma Membrane Vesicles Isolated from Rat Liver: K. Okudaira,
K. Yachi, Y. Sawada, Y. Sugiyama, T. Iga and M. Hanano
SHORT COMMUNICATION
Pharmacokinetics of Drugs in Blood: VII: Unusual Distribution and
Blood Storage Effect of Vancomycin: W. G. Shin, M. G. Lee, M. H. Lee
and N. D. Kim.
Issue No. 5, July
REVIEW ARTICLE
Drugs and the Liver. Part III: Ageing of the Liver and the Metabolism of
Drugs: K. Woodhouse
RESEARCH PAPERS
Effect of Indomethacin on the Pharmacokinetics of Methotrexate in
Rabbits: T. A. O. Najjar, A. R. M. Morad and R. M. A. Khan
Effect of Food and Relative Bioavailability Following Single Doses of
Diclofenac 150 mg Hydrogel Bead (HGB) Capsules in Healthy Humans:
K. M. Thakker, S. Mangat, W. Wagner,J . Castellana and G. M. Kochak
Pharmacokinetics of Ibuprofen Enantiomers After Single and Repeated
Doses in Man: J. Oliary, M. Tod, P. Nicolas, O. Petitjean and G. Caillé
Distribution Kinetics of FK-506, a Novel Immunosuppressant, After
Intravenous Administration to Rats in Comparison with Cyclosporin
A: K. Takada, H. Usuda and M. Oh-Hashi
VOLUME CONTENTS
Plasma Disposition and Hemodynamic Effects ofa Single Oral Dose of
Isosorbide Dinitrate in Human Males and Females: K. Nakatsu, J. F.
Brien, G. Savard, E. B. Toffelmire, H. Abdollah, B. M. Bennett and
G. S. Marks
‘In Vitro’ Action of Histamine and Cimetidine on Amylase Secretion in
the Rat Pancreas: L. J. Murillo, J. Torre-Cisneros, A. Blanco-Molina,
J. Lopez-Miranda, R. A. F. de la Puebla and F. Pérez-Jiménez
SHORT COMMUNICATION
Pharmacokinetics/Pharmacodynamics of Labetalol in Three Pregnant
Ewes Using High-performance Liquid ee M.S. Leloux
and H. W. Jongsma . : ; : ; ‘
LETTERS TO THE EDITOR
Enantioselective versus Non-Enantioselective Assays in Comparative
Bioavailability Studies with Racemic are W. D. ie tae:x . <3,
Dickinson and J. Gal : :
Enantioselective versus Non-Enantioselective Assays in Comparative
Bioavailability Studies with Racemic Drugs: F. Jamali
ANNOUNCEMENT .
Issue No. 6, August
Prediction of the Volume of Distribution of 7-Hydroxycoumarin in Man
from in vitro and ex vivo Data Obtained in Rat: W. A. Ritschel, R. D.
Johnson, N. N. Vachharajani and A. S. Hussain
Influence of Probenecid and Paracetamol (Acetaminophen) on
Zidovudine Glucuronidation in Human Liver in vitro: F. Kamali and
M.D. Rawlins .
Distribution of Carbamazepine and its Epoxide in Blood Compartments
in Adolescent and Adult Epileptic Patients: J. Bonneton, P. Genton and
E. Mesdjian
Rapid Toxicological Model for Use in Assessing Ocular Drugs: C. M.
Ellingson, R. D. Schoenwald, C. F. Barfknecht, C. S. Rao and S. L.
Laban
Studies on the Intravenous Pharmacokinetics in Rabbit and in vitro
Protein Binding of Two New Salts of Erythromycin: Erythromycin
Maltobionate and Erythromycin Fumarate: S. K. Basu, P. K. Manna
and B. B. Goswami .
Pharmacokinetics and Metabolism of Codeine in Humans: T. B. Vree,
C. P. W. G. M. Verwey-van Wissen
vi VOLUME CONTENTS
Extended Least Squares Curve Fitting: A Comparison of SIPHAR and
MK MODEL: I. D. Cockshott and J. Haywood .
Issue No. 7, October
RESEARCH PAPERS
Simultaneous Modelling of Mexiletine and Hydroxy-methyl-mexiletine
Data After Single- and Multiple-dose Administration of a Sustained-
release Mexiletine Formulation: R. Bruno, Y. Santoni, A. Iliadis, P.
Djiane, A. Serradimigni and J. P. Cano
Pharmacokinetics of Oxatomide Given Percutaneously to Healthy
Volunteers: C. Benvenuti, M. Broggini, V. Bott, M. Valenti, G.
Broccali and L. Dal Bo
Bioavailability of Lithium from Lithium citrate Syrup Versus Conven-
tional Lithium Carbonate Tablets: P. J. M. Guelen, T. J. Janssen,
T.C. M. De Witte, T. B. Vree and K. Benson
Effect of Congestive Heart Failure on Clentiazem Pharmacokinetics in
a Dog Model: A. K.-Laflamme, G. Caille, R. Cardinal, D. Croteau,
C. Lamoureux and C. Lambert .
The Effects of Chronic Oral Diltiazem and Cimetidine Dosing on the
Pharmacokinetics and Negative Dromotropic Action of Intravenous
and Oral Diltiazem in the Dog: C. Maskasame, S. Lankford and
S.A. Bai .
Simultaneous Monitoring of Bemoradan Pharmacokinetics and Hemo-
dynamics in Mongrel Dogs: S.-M. Huang, R. Falotico, B. Haertlein
and I. L. Smith.
SHORT COMMUNICATIONS
In vivo Evaluation of the Effect of the Size and Opsonization on the
Hepatic Extraction of Liposomes in Rats: an Application of Oldendorf
Method: H. Harashima, Y. Ohnishi and H. Kiwada
Extrahepatic Production of the Lignocaine Metabolite Monoethyl-
glycinexylidide (MEGX): R. W. Sallie, J. M. Tredger and R. Williams
Issue No. 8, November
Comparative Bioavailability and Steady State Fluctuations of Tegretol
Commercial and Carbamazepine Oros Tablets in Adult and Pediatric
Epileptic Patients: K. M. Thakker, S. Mangat, W. R. Garnett, R. H.
Levy and G. M. Kochak
VOLUME CONTENTS
Applicability of Teicoplanin Dosage Adjustment Guidelines for Renally
Impaired Patients over the Range of3 to 30 MG KG“ ': J. A. Smithers,
G. A. Thompson, M. T. Kenny, J. K. Dulworth, H. K. Kulmala, E. W.
Lewis, S. J. Ruberg, B. E. Shapiro, W. F. Keane and C. E. Halstenson
Pharmacokinetics of Alfuzosin After Single Oral Administration to
Healthy Volunteers, of Three Different Doses: P. Salva, G. Bianchetti,
P. Morselli, G. Garcia-Teresa and J. Costa
Disposition Kinetics of 7,12-Dimethylbenz(A) Anthracene in Rats: S. K.
Niazi and M. Hussain : ’ ; :
Input Rate-Dependent Stereoselective Pharmacokinetics: Enantiomeric
Oral Bioavailability and Blood Concentration Ratios after Constant
Orai Input: R. Mehvar ;
The Metabolism of CGS 15873 in Man Using StS able ‘oe Pattern
Recognition Techniques: M. Leal, M. J. Hayes and M. L. Powell
SHORT COMMUNICATION
Inappropriate Inclusion of Non-Quantifiable Plasma Concentrations in
the Estimation of Extent of Absorption: A. J. Jackson
Issue No. 9, December
Immunosuppressive Effect of Cyclosporine in the Hyperlipidemic Rat
Model: D. R. Luke
Nonlinear Pharmacokinetics of Hepatobiliary Transport of Rose Bengal
in Rats After IV Bolus Administration with Varying Doses: H. K.
Wang, S. Miyachi, M. Yamazaki, Y. Sawada, Y. B. Chung, T. Iga,
M. Hanano and Y. Sugiyama
Clinical Pharmacokinetics of Procaterol: Dose Proportionality After
Administration of Single Oral Doses: M. A. Eldon, D. S. Blake, M. J.
Coon, G. D. Nordblom, A. J. Sedman and W. A. Colburn .
Moxisylyte Plasma Kinetics in Humans After Intracavernous Adminis-
tration: P. Costa, F. Bressolle, B. Sarrazin, J. Mosser, H. Navratil and
M. Galtier
Sex-Differences in the Disposition of Substituted Benzamides: Pharma-
cokinetics of a Gastroprokinetic Agent (4-Amino-5-Chloro-2-
[2-(Methylsulfinyl) Ethoxy]-N-[2-(Diethylamino)Ethyl] Benzamide
Hydrochloride) (ML-1035) in Male and Female New Zealand White
Rabbits: N. Rao, K. W. Otis and K.-K. Hwang . ; i
Human Dolasetron Pharmacokinetics: I. Disposition Following
Single-Dose Intravenous Administration to Normal Male Subjects:
H. Boxenbaum, T. Gillespie, K. Heck and W. Hahne .
Viil VOLUME CONTENTS
Pharmacokinetics of progesterone in Ovariectomized Rats After Single
Dose Intravenous Administration: N. K. Gangrade, F. D. Boudinot
and J.C. Price . : ‘ : : ‘ : d ; .
Author Index ; : : . ; y ; : : ; . ae
Keyword Index . : ; ; ‘ : 5 ‘ ‘ ; : oto
Volume Contents . : ; : 3 ‘ : . ; ; ; ii
Indexed or abstracted by Analytical Abstracts, BIOMED Database (Institute for Scientific
Information—ISI), BIOSIS, Cambridge Scientific Abstracts, Chemical Abstracts Service, CIS
Abstracts, Current Awareness in Bio. Sciences, Excerpta Medica, Index Medicus, Int. Pharmaceutical
Abstracts, Reference Update, Research Alert (ISI), Science Citation Index (ISI), SCISEARCH
Database (ISI), VINITI-USSR Academy of Sciences
Copyright © 1992 by John Wiley & Sons Ltd.
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