Biochemical Pharmacology 2002: Vol 64 Table of Contents

13 Pages·2002·3.9 MB·English

Biochemical Pharmacology 64 (2002) 1795-1806
Contents of Volume 64
1 July 2002 67 NMR and pattern recognition studies on liver
extracts and intact livers from rats treated with a-
naphthylisothiocyanate
Commenta
; Vv / Nigel J. Waters, Elaine Holmes, Catherine J. Waterfield,
1 Interleukin-1B converting enzyme (caspase-1) in
Ce | R. Duncan Farrant and Jeremy K. Nicholson
intestinal inflammation
Britta Siegmund 79 = DNA structural alterations induced by bis-netropsins
modulate human DNA topoisomerase I cleavage
activity and poisoning by camptothecin
MOLECULAR AND CELLULAR PHARMACOLOGY Alyona Sukhanova, Sergei Grokhousky,
») y +) SO 5 .
9 Similarities and differences in the coupling of human Michael Ermishov, Konstantin Mochalov,
B,- and B,-adrenoceptors to Gsa splice variants Alexei Zhuze, Vladimir Oleinikov and Igor Nabiev
Katharina Wenzel-Seifert, Hui-Yu Liu and Roland Seifert 91 Membrane heme as a host factor in reducing effec-
21 = Identification of a signaling cascade for interleukin-8 tiveness of dihydroartemisinin
production by Helicobacter pylori in human gastric Phantip Vattanaviboon, Noppadol Siritanaratkul,
epithelial cells Jidapa Ketpirune, Prapon Wilairat and
Yoshihisa Nozawa, Katsushi Nishihara, Yongyuth Yuthavong
Richard M. Peek Jr., Motoko Nakano, 99. Modulati ve rears eee ie :
Tatsuya Uji, Hirofusa Ajioka, Naosuke Matsuura ee ee ee ee
ipheral benzodiazepine receptor ligands in breast can-
and Hidekazu Miyake ll
cer cells
31. =C haracterization of glomerular cell phenotypes fol- Renate Strohmeier, Marc Roller, Nicole Sanger,
lowing repeated cycles of benzola]pyrene injury in Rainald Knecht and Herbert Kuhl
vitro
AbD Gui. Nawolons © Aisiatieo. 109 eee . is an endogenous inhibitor of soluble
Christopher M. Bral, J. Kevin Kerzee, sc i oe :
Russell C. Bowes III and Kenneth S. Ramos Markus Koglin and Sénke Behrends
41. = Alterations in membrane-bound and cytoplasmic K-
ras protein levels in mouse lung induced by treatment NEUROSCIENCE
with lovastatin, cholestyramine, or niacin: effects are
117 Arachidonic acid release and prostaglandin F,, for-
highly mouse strain dependent
mation induced by phenylarsine oxide in PC12 cells:
Richard J. Calvert, Gayatri Ramakrishna, possible involvement of secretory phospholipase Az
Shirley Tepper, Bhalchandra A. Diwan,
activity
| Lucy M. Anderson and David Kritchevsk
| of . Keiko Ohsawa, Asako Mori, Syunji Horie,
nl 49 Analysis of rainbow trout Ah receptor protein iso- Takeshi Saito, Yasunobu Okuma,
forms in cell culture reveals conservation of function Yasuyuki Nomura and Toshihiko Murayama
in Ah receptor-mediated signal transduction a
| 125 Effects of (—)-nicotine and (—)-cotinine on 6-hydro-
Richard S. Pollenz, Brian Necela and Sorat se ae
xydopamine-induced oxidative stress and neurotoxi-
Katherine Marks-Sojka Cee
city: relevance for Parkinson’s disease
61 = Effector coupling of stably transfected human A; ade- Ramon Soto-Otero, Estefania Méndez-Alvarez,
nosine receptors in CHO cells Alvaro Hermida-Ameijeiras, Ana Maria Lopez-Real
Martin Englert, Ursula Quitterer and Karl-Norbert Klotz and José Luis Labandeira-Garcia
PII: SO0006-2952(02)01531-9
Contents of Volume 64
191 Mechanism of action of non-cisplatin type DNA-tar-
GENE EXPRESSION AND DEVELOPMENT
geted platinum anticancer agents: DNA interactions
Gene expression profiling of drug metabolism and
of novel acridinylthioureas and their platinum con-
toxicology markers using a low-density DNA micro-
jugates
array
Hemanta Baruah, Christopher L. Rector,
Francoise de Longueville, Dominic Surry,
Susanne M. Monnier and Ulrich Bierbach
Georgina Meneses-Lorente, Vincent Bertholet,
Inhibition of phosphate transport in rat heart mito-
Valérie Talbot, Stephanie Evrard, Nathalie Chandelier,
Andrew Pike, Phil Worboys, Jean-Paul Rasson, chondria by 3’-azido-3’-deoxythymidine due to stimu-
lation of superoxide anion mitochondrial production
Béatrice Le Bourdellés and José Remacle
Daniela Valenti, Anna Atlante, Maria Barile and
Salvatore Passarella
GASTROINTESTINAL AND RENAL PHARMACOLOGY
Enhanced resistance of HeLa cells to cisplatin by
Inhibition of transport across the hepatocyte canali-
overexpression of y-glutamyltransferase
cular membrane by the antibiotic fusidate
Sandrine Daubeuf, Pierre Leroy, Aldo Paolicchi,
Konrad A. Bode, Markus G. Donner,
Alfonso Pompella, Maria Wellman,
Inka Leier and Dietrich Keppler
Marie Madeleine Galteau and Athanase Visvikis
Effects of polysulfated glycosaminoglycan and triam-
ERRATUM cinolone acetonid on the production of proteinases
and their inhibitors by IL-1o treated articular chon-
Erratum to “Drug-resistant human lung cancer cells
drocytes
are more sensitive to selenium cytotoxicity: effects on
thioredoxin reductase and glutathione reductase”. Thorsten Sadowski and Jiirgen Steinmeyer
[Biochem. Pharmacol. 63 (2002) 1875-1884]
Inhibition of matrix-proteases by polyphenols: che-
Linda Bjérkhem-Bergman, Kerstin Jonsson, mical insights for anti-inflammatory and anti-inva-
Lennart C. Eriksson, Jerker M. Olsson, sion drug design
Soren Lehmann, Christer Paul and Mikael Bjornstedt
Luigi Sartor, Elga Pezzato, Isabella Dell’ Aica,
Rosamaria Caniato, Susan Biggin and Spiridione Garbisa
15 July 2002 3'-Azido-2’,3'-dideoxythymidine induced deficiency
of thymidine kinases 1, 2 and deoxycytidine kinase
in H9 T-lymphoid cells
Bettina Groschel, Andreas Kaufmann, Gerold Hover,
Commentary
Jaroslav Cinatl, Hans Wilhelm Doerr, Paul Noordhuis,
Lysophosphatidylcholine as a ligand for immunoregu-
Willem J.P. Loves, Godefridus J. Peters and
lation
Jindrich Cinatl Jr.
Janusz H.S. Kabarowski, Yan Xu and Owen N. Witte
Relationship between the activation of heat shock fac-
tor and the suppression of nuclear factor-«B activity in
rat hepatocyte cultures treated with cyclosporine A
MOLECULAR AND CELLULAR PHARMACOLOGY
David Andrés, Carmen Diez-Ferndndez,
Inhibition of heparin synthesis by methotrexate in
Antonio Castrillo and Maria Cascales
rats in vivo
See : 355
Identification of two C-terminal amino acids, Ser
Sisi Marcondes, Elaine C. Bau, Edson Antunes,
and Thr’?’, required for short-term homologous
Carl P. Dietrich, Helena B. Nader and
desensitization of t-opioid receptors
Gilberto De Nucci
Hung-Li Wang, Wen-Teng Chang, Chia-Yu Hsu,
Induction of cyclooxygenase-2 by staurosporine
Pei-Chen Huang, Yu-Wen Chow and Allen H. Li
through the activation of nuclear factor for IL-6
(NF-IL6) and activator protein 2 (AP2) in an osteo- Novel mechanism of Vitamin E protection against
blast-like cell line cyclosporine A cytotoxicity in cultured rat hepatocytes
Chiu-Ya Wang, Huey-Jing Lei, Chi-Ying Fred Huang, David Andrés and Maria Cascales
Zhongjian Zhang, Anil B. Mukherjee and
Modulation of L-arginine transport and nitric oxide
Chiun-Jye Yuan
production by gabexate mesylate
Renal organic cation and nucleoside transport
Giuliana Leoncini, Raffaele Pascale and
Rong Chen, Johan W. Jonker and J. Arly Nelson Maria Grazia Signorello
Contents of Volume 64 1797
285 Hyperekplexia mutation of glycine receptors: Matthew Z. Dieter, Sarah L. Freshwater,
decreased gating efficacy with altered binding ther- Willy A. Solis, Daniel W. Nebert and
modynamics Timothy P. Dalton
Gabor Maksay, Timea Biro and Bodo Laube
353 Erratum to “Expression of rat aldehyde reductase
AKR7AI1: influence of age sex and tissue-specific
(CHEMOANDT MHETAEBOLRIC AINPHIBYITO RS inducibility”. [Biochem. Pharmacol. 62 (2001)
1511-1519]
289 Covalent binding of the anticancer drug ellipticine to
Anne Grant, Louise Staffas, Louise Mankowitz,
DNA in V79 cells transfected with human cyto-
Vincent P. Kelly, Margaret M. Manson,
chrome P450 enzymes
Joseph W. DePierre, John D. Hayes and
Eva Frei, Christian A. Bieler, Volker M. Arlt,
Elizabeth M. Ellis
Manfred Wiessler and Marie Stiborova
297 Carbonyl reduction of the potential cytostatic drugs
benfluron and 3,9-dimethoxybenfluron in human in 1 August 2002
vitro
Lenka Skdlova, Milan Nobilis, Barbora Szotakova,
Eliska Kondrovd, Michal Savlik, Vladimir Wsol, Commentary
Lydiane Pichard-Garcia and Edmund Maser 359 Designer glucocorticoids
Jeffrey N. Miner
GENE ExPREANSD SDEIVELOOPNMEN T
307 Activation of the y-glutamyltransferase promoter 2 in Rapid Communication
the rat colon carcinoma cell line CC531 by histone 363 Brain mitochondrial uncoupling protein 2 (UCP2): a
deacetylase inhibitors is mediated through the Spl protective stress signal in neuronal injury
binding motif
Ingo Bechmann, Sabrina Diano, Craig H. Warden,
Idun Merete Mikkelsen, Nils-Erik Huseby, Tamas Bartfai, Robert Nitsch and Tamas L. Horvath
Athanase Visvikis and Ugo Moens
369 Uncoupling protein 2 (UCP2) lowers alcohol sensi-
tivity and pain threshold
INFLAMMATION AND IMMUNOPHARMACOLOGY
Balazs Horvath, Claudia Spies, Gyongyi Horvath,
317 Induction of interleukin 8 release from the HMC-1 Wolfgang J.K ox, Suzanne Miyamoto, Sean Barry,
mast cell line: Synergy between stem cell factor and Craig H. Warden, Ingo Bechmann, Sabrina Diano,
activators of the adenosine A>}, receptor Jill Heemskerk and Tamas L. Horvath
Christopher J. Meade, Liam Worrall,
Dawn Hayes and Ursula Protin
MOLECULAR AND CELLULAR PHARMACOLOGY
327 GPI 6150, a PARP inhibitor, reduces the colon injury
375 Agents that elevate cyclic AMP induce receptor
caused by dinitrobenzene sulfonic acid in the rat
phosphorylation primarily at serine 331 in HEK 293
Emanuela Mazzon, Laura Dugo, Jia-He Li,
cells overexpressing human thromboxane receptor &
Rosanna Di Paola, Tiziana Genovese,
Shuichi Yamamoto, Fengxiang Yan,
Achille P. Caputi, Jie Zhang and Salvatore Cuzzocrea
Huiping Zhou and Hsin-Hsiung Tai
it ae
GASTROINTESTINAL AND RENAL PHARMACOLOGY 385 Phorbol ester-induced contractility and Ca“" influx
in human cultured prostatic stromal cells
339 Indomethacin-induced mitochondrial dysfunction
John M. Haynes, Lydia Iannazzo and Henryk Majewski
and oxidative stress in villus enterocytes
Jayasree Basivireddy, Anju Vasudevan, 393 Modulations of P450 mRNA in liver and mammary
Molly Jacob and Kunissery A. Balasubramanian gland and P450 activities and metabolism of estrogen
in liver by treatment of rats with indole-3-carbinol
Thomas L. Horn, Mark A. Reichert, Robin L. Bliss and
ERRATA
Danuta Malejka-Giganti
351 Erratum to “Tyrphostin AG879, a tyrosine kinase
405 Inhibition by adenine dinucleotides of ATP-induced
inhibitor: prevention of transcriptional activation of
prostacyclin release by bovine aortic endothelial cells
the electrophile and the aromatic hydrocarbon
response elements”. [Biochem. Pharmacol. 61 Luminita H. Pojoga, Maricela Haghiac and
(2001) 215-225] Richard H. Hilderman
Contents of Volume 64
Cell culture model for acetaminophen-induced hepa- Richard Steinbrugger, Walter Jager, Georg Krupitza,
tocyte death in vivo Howard L. Elford and Thomas Szekeres
Robert H. Pierce, Christopher C. Franklin,
Jean S. Campbell, Robert P. Tonge, Weichao Chen,
NEUROSCIENCE
Nelson Fausto, Sidney D. Nelson and Sam A. Bruschi
Lack of correlation between NF-«B activation and
Endothelin-l-induced arachidonic acid release by induction of programmed cell death in PC12 pheo-
cytosolic phospholipase A> activation in rat vascular chromocytoma cells treated with 6-hydroxydopamine
smooth muscle via extracellular signal-regulated or the cannabinoid receptor 1-agonist CP55,940
kinases pathway
Nina Erlandsson, Bernd Baumann, Oliver G. Rossler,
Lucia Trevisi, Sergio Bova, Gabriella Cargnelli, Katrin Kaufmann, Klaus M. Giehl, Thomas Wirth and
Giulio Ceolotto and Sisto Luciani Gerald Thiel
Inhibition of platelet P2Y12 and «2A receptor signal-
ing by cGMP-dependent protein kinase HORMONES AND GROWTH FACTORS
Barsom Aktas, Petra Honig-Liedl, Ulrich Walter and
Reduction of bFGF-induced smooth muscle cell pro-
Jorg Geiger
liferation and endothelin receptor mRNA expression
Inhibition of mitochondrial permeability transition by mevastatin and atorvastatin
and release of cytochrome c by anti-apoptotic nucleo- Cang-Bao Xu, Emelie Stenman and Lars Edvinsson
side analogues
Quantitation of estradiol receptors alpha and beta
Luzheng Xue, Vilma Borutaite and Aviva M. Tolkovusky
and progesterone receptors in human breast tumors
Ribonucleotide reductase and thymidine phosphory- by real-time reverse transcription-polymerase chain
lation: two potential targets of azodicarbonamide reaction. Correlation with protein assays
Christine Fagny, Michel Vandevelde, Michal Svoboda Patricia de Cremoux, Carine Tran-Perennou,
and Patrick Robberecht Caroline Elie, Evelyne Boudou, Catherine Barbaroux,
Marie France Poupon, Yann De Rycke, Bernard Asselain
Anti-inflammatory drugs modulate Clq secretion in
and Henri Magdelénat
human peritoneal macrophages in vitro
Dominik Faust, Bora Akoglu, Dimitrios Zgouras,
Ernst-Heinrich Scheuermann, Vladan Milovic INFLAMMATION AND IMMUNOPHARMACOLOGY
and Jtirgen Stein
Effect of pirfenidone against vanadate-induced kid-
Substrate-dependent, non-hyperbolic kinetics of pig ney fibrosis in rats
brain prolyl oligopeptidase and its tight binding inhi-
Mohammed Ali Al-Bayati, Yan Xie, F. Charles Mohr,
bition by JTP-4819 Solomon B. Margolin and Shri N. Giri
Jarkko I. Venadldinen, Risto O. Juvonen,
Markus M. Forsberg, Arturo Garcia-Horsman,
CARDIOVASCULAR AND PULMONARY PHARMACOLOGY
Antti Poso, Erik A.A. Wallen, Jukka Gynther and
Pekka T. Madnnisto Analysis of oxidative processes and of myelin figures
formation before and after the loss of mitochondrial
transmembrane potential during 7B-hydroxycholes-
(CHEMOTHERAPY AND METABOLIC INHIBITORS
terol and 7-ketocholesterol-induced apoptosis: com-
A novel stereo-selective sulfonylurea, 1-[1-(4-amino- parison with various pro-apoptotic chemicals
benzoyl)-2,3-dihydro-1H-indol-6-sulfonyl]-4-phenyl-
Carole Miguet-Alfonsi, Céline Prunet, Serge Monier,
imidazolidin-2-one, has antitumor efficacy in in vitro
Ginette Besséde, Stéphanie Lemaire-Ewing,
and in vivo tumor models
Arnaud Berthier, Franck Ménétrier, Dominique Neel,
Chang Woo Lee, Dong Ho Hong, Sang Bae Han, Philippe Gambert and Gérard Lizard
Sang-Hun Jung, Hyung Chin Kim, Robert L. Fine,
Sang-Han Lee and Hwan Mook Kim
GASTROINTESTINAL AND RENAL PHARMACOLOGY
Trimidox, an inhibitor of ribonucleotide reductase,
synergistically enhances the inhibition of colony for- Enhancement of protein kinase C activity and che-
mation by Ara-C in HL-60 human promyelocytic miluminescence intensity in mitochondria isolated
leukemia cells from the kidney cortex of rats treated with cephalor-
idine
Monika Fritzer-Szekeres, Alexandra Salamon,
Michael Grusch, Zsuzsanna Horvath, Thomas Héchtl, Yuka Kohda and Munekazu Gemba
Contents of Volume 64 1799
ERRATUM 633 Role of temperature on protein and mRNA cyto-
chrome P450 3A (CYP3A) isozymes expression and
J01 Erratum to “Chronic ethanol administration
midazolam oxidation by cultured rat precision-cut
decreases the ligand binding properties and the cel-
liver slices
lular content of the mannose 6-phosphate/insulin-
Eleni Rekka, Ekaterina Evdokimova,
like growth factor II receptor in rat hepatocytes”.
Stéphane Eeckhoudt, Geoffray Labar and
[Biochem. Pharmacol. 63 (2002) 1229-1239]
Pedro Buc Calderon
James Haorah, Daniel L. McVicker, James C. Byrd,
Richard G. MacDonald and Terrence M. Donohue Jr. 645 G protein-coupled receptor for nicotinic acid in
mouse macrophages
Anna Lorenzen, Christina Stannek, Anja Burmeister,
15 August 2002 Ivars Kalvinsh and Ulrich Schwabe
(CHEMOTHERAPY AND METABOLIC INHIBITORS
Commentary
649 Insufficiently charged isosteric analogue of spermine:
903 Toxic, halogenated cysteine S-conjugates and target-
interaction with polyamine uptake, and effect on
ing of mitochondrial enzymes of energy metabolism
Caco-2 cell growth
Arthur J.L. Cooper, Sam A. Bruschi and M.W. Anders
Lyudmila Turchanowa, Alexander S. Shvetsov,
Alexander V. Demin, Alex R. Khomutov,
Heather M. Wallace, Jvirgen Stein and Vladan Milovic
MOLECULAR AND CELLULAR PHARMACOLOGY
965 Enhancement of glutathione-dependent haemin 657 Effects of in vivo treatment of rats with trimethyltin
degradation by ascorbic acid chloride on respiratory properties of rat liver mito-
chondria
Cheng-Gang Zou, Nihal S. Agar and
Graham Lloyd Jones Cecilie Resen-Fellie Skarning, Ludvig Nord Varhaug,
Frode Fonnum and Harald Osmundsen
973 Modulation of P-glycoprotein expression and function
by curcumin in multidrug-resistant human KB cells 669 Effects of antifolates on the binding of 5-fluoro-2’-
deoxyuridine monophosphate to thymidylate
Songyot Anuchapreeda, Pranee Leechanachai,
synthase
Melissa M. Smith, Suresh V. Ambudkar and
Porn-ngarm Limtrakul Clasina L. van der Wilt, Kees Smid and
Godefridus J. Peters
983 Distinct interactions of Gyy-jongs Gsx-shorty aNd Gyoir
with GTP, ITP, and XTP
NEUROSCIENCE
Hui-Yu Liu and Roland Seifert
677 Biphasic effects of oxethazaine, a topical anesthetic,
995 Inhibition of the activity of T lymphocyte Kv1.3
on the intracellular Ca“ concentration of PC12 cells
channels by extracellular zinc ? .
Yasusuke Masuda, Tamami Oguma and Akira Kimura
Andrzej Teisseyre and Jerzy W. Mozrzymas
Cationic liposomes as delivery systems for double-
HORMONES AND GROWTH FACTORS
stranded PNA-DNA chimeras exhibiting decoy
activity against NF-«B transcription factors 689 Synergistic effect of dimethyl sulfoxide on glucagon-
like peptide 1 (GLP-1)-stimulated insulin secretion
Monica Borgatti, Laura Breda, Rita Cortesi,
Claudio Nastruzzi, Alessandra Romanelli, and gene transcription in INS-1 cells: characteriza-
Michele Saviano, Nicoletta Bianchi, Carlo Mischiati, tion and implications
Carlo Pedone and Roberto Gambari Daniel M. Kemp and Joel F. Habener
|
|
617 mRNA expression profiles for the response of human
{
tumor cell lines to the antimalarial drugs artesunate,
\ GENE EXPRESSION AND DEVELOPMENT
arteether, and artemether
699 Human histamine N-methyltransferase pharmacoge-
Thomas Efferth, Armin Olbrich and Rudolf Bauer
netics: gene resequencing, promoter characterization,
625 Up-regulation of Aya adenosine receptors by proin- and functional studies of a common 5’-flanking
flammatory cytokines in rat PC12 cells region single nucleotide polymorphism (SNP)
Maria L. Trincavelli, Barbara Costa, Daniela Tuscano, Liewei Wang, Bianca Thomae, Bruce Eckloff,
Antonio Lucacchini and Claudia Martini Eric Wieben and Richard Weinshilboum
1800 Contents of Volume 64
711 Expression and activity of the DNA repair enzyme ura- Jacques Pouysségur, Véronique Volmat and
cil DNA glycosylase during organogenesis in the rat Philippe Lenormand
conceptus and following methotrexate exposure in vitro
Antioxidants and oxidants regulated signal transduc-
Robert K. Vinson and Barbara F. Hales tion pathways
Edward D. Owuor and Ah-Ng Tony Kong
STRUCTURAL BIOLOGY
Activation of mitogen-activated protein kinases
Structural and functional characterization of an acidic (MAPKs) by aromatic hydrocarbons: role in the reg-
platelet aggregation inhibitor and hypotensive phos- ulation of aryl hydrocarbon receptor (AHR) function
pholipase A> from Bothrops jararacussu snake venom
Zongqing Tan, Xiaoging Chang, Alvaro Puga and
Silvia H. Andrido-Escarso, Andreimar M. Soares, Ying Xia
Marcos R.M. Fontes, André L. Fuly,
The c-Jun N-terminal kinases in cerebral microglia:
Fernando M.A. Corréa, José C. Rosa,
immunological functions in the brain
Lewis J. Greene and José R. Giglio
Ute Hidding, Kirsten Mielke, Vicki Waetzig,
Differential binding to the o/B-tubulin dimer of
Stephan Brecht, Uwe Hanisch, Alexander Behrens,
vinorelbine and vinflunine revealed by nuclear mag-
Erwin Wagner and Thomas Herdegen
netic resonance analyses
Inflammatory signal transduction in Crohn’s disease
Christine Fabre, Jerzy Czaplicki, Michel Wright,
and novel therapeutic approaches
Bridget Hill, Jean Marc Barret, Jacques Fahy
and Alain Milon Catherine van Montfrans, Maikel Peppelenbosch,
Anje A. te Velde and Sander van Deventer
INFLAMMATION AND IMMUNOPHARMACOLOGY Growth signaling in breast cancer cells: outcomes and
promises of proteomics
In vivo anti-complement effect of bilirubin-I[Xa
Eric Adriaenssens, Jéréme Lemoine,
Sandra M. Arriaga, Adriana M. Almard and
Ikram El Yazidi-Belkoura and Hubert Hondermarck
Aldo D. Mottino
Sodium tanshinone IIA sulfonate derived from Dan-
RECEPTOR SIGNALING
shen (Salvia miltiorrhiza) attenuates hypertrophy
induced by angiotensin II in cultured neonatal rat Divalent cations and the relationship between aA
cardiac cells and BA domains in integrins
Kyoko Takahashi, Xinshou Ouyang, Katsuko Komatsu, Kah-Tong Seow, Jian-Ping Xiong, M. Amin Arnaout,
Norio Nakamura, Masao Hattori, Akemichi Baba and Jutta Welge, Friedrich Rippmann and
Junichi Azuma Simon L. Goodman
A homogenous assay to monitor the activity of the
Erratum
insulin receptor using Bioluminescence Resonance
Erratum to “Mechanism of action of non-cisplatin
Energy Transfer
type DNA-targeted platinum anticancer agents:
Tarik Issad, Nicolas Boute and Karine Pernet
DNA interactions of novel acridinylthioureas and
their platinum conjugates”. [Biochem. Pharmacol.
64 (2002) 191-200]
CELL CYCLE CONTROL
Hemanta Baruah, Christopher L. Rector,
Identifying in vivo targets of cyclin-dependent kinase
Susanne M. Monnier and Ulrich Bierbach
inhibitors by affinity chromatography
Marie Knockaert and Laurent Meijer
September 2002 ErbB-2-induced mammary tumor growth: the role of
cyclin D1 and p27Kip1
Cell signaling, transcription and translation as ther- James Hulit, Richard. J. Lee, Robert G. Russell and
Richard G. Pestell
apeutic targets
Marc Diederich Independent contribution of three different pathways
to ultraviolet-B-induced apoptosis
SIGNALING PATHWAYS Dagmar Kulms and Thomas Schwarz
Fidelity and spatio-temporal control in MAP kinase Cell-specific regulation of apoptosis by glucocorti-
(ERKs) signalling coids: implication to their anti-inflammatory action
Contents of Volume 64 1801
Abraham Amsterdam, Kimihisa Tajima and 943 Transcriptional regulators of the human multidrug
Ravid Sasson resistance | gene: recent views
Stéphane Labialle, Landry Gayet, Eric Marthinet,
851 Prospects for targeting the Bcl-2 family of proteins to
Dominique Rigal and Loris G. Baggetto
develop novel cytotoxic drugs
Jonathan B. Baell and David C.S. Huang 949 Function of AP-1 target genes in mesenchymal—
epithelial cross-talk in skin
865 Regulation of p53: intricate loops and delicate bal-
Peter Angel and Axel Szabowski
ances
957 Evasion from proteasomal degradation by mutated
Moshe Oren, Alexander Damalas, Tanya Gottlieb,
Fos proteins expressed from FBJ-MSV and FBR-
Dan Michael, Jan Taplick, Juan Fernando Martinez
Leal, Ruth Maya, Miri Moas, Rony Seger, Yoichi Taya MSV osteosarcomatogenic retroviruses
and Avri Ben-Ze’ev Claire Acquaviva, Guillaume Bossis, Patrizia Ferrara,
Frédérique Brockly, Isabelle Jariel-Encontre and
873 Identification of cytokine-induced nuclear factor-
Marc Piechaczyk
kappaB target genes in ovarian and breast cancer cells
963 Regulation of the transcriptional activity of the
Valérie Deregowski, Sylvie Delhalle, Valérie Benoit,
nuclear factor-KB p65 subunit
Vincent Bours and Marie-Paule Merville
Linda Vermeulen, Gert De Wilde, Sofie Notebaert,
883 Nuclear factor-kappa B and cancer: its role in preven-
Wim Vanden Berghe and Guy Haegeman
tion and therapy
971 Reduction of tumor necrosis factor-alpha (TNF-a)
Alok C. Bharti and Bharat B. Aggarwal
related nuclear factor-kappaB (NF-«B) translocation
Is HIF-1a a pro- or an anti-apoptotic protein? but not inhibitor kappa-B (Ix-B)-degradation by Rho
Jean-Pascal Piret, Denis Mottet, Martine Raes and protein inhibition in human endothelial cells
Carine Michiels Stefan Hippenstiel, Bernd Schmeck, Joachim Seybold,
Matthias Kriill, Christoph v. Eichel-Streiber and
Norbert Suttorp
NUTRIENTS REGULATED GENE EXPRESSION
979 Differential activity by DNA-induced quarternary
893 Is there a single mechanism for fatty acid regulation
structures of POU transcription factors
of gene transcription?
Attila Reményi, Alexey Tomilin, Hans R. Scholer and
Eric Duplus and Claude Forest
Matthias Wilmanns
903 Signaling cross-talk between hypoxia and glucose via
985 Multiple signaling pathways leading to the activation
hypoxia-inducible factor 1 and glucose response ele-
of interferon regulatory factor 3
ments
Marc J. Servant, Nathalie Grandvaux and John Hiscott
Thomas Kietymann, Anja Krones-Herzig and
Kurt Jungermann 993 Signal transduction to hypoxia-inducible factor 1
Gregg L. Semenza
913 Genomic responses to herbal extracts: lessons from in
vitro and in vivo studies with an extract of Ginkgo
biloba SIGNAL TRANSDUCTION, STRESS RESPONSE AND AGING
Kishorchandra Gohil
999 Age-related decline in cellular response to oxidative
stress: links to growth factor signaling pathways with
common defects
TRANSCRIPTIONAL REGULATION
Nikki J. Holbrook and Shizuo Ikeyama
919 Designed transcription factors as tools for therapeu-
| tics and functional genomics 1007 Stress-induced premature senescence and tissue age-
ing
Fyodor D. Urnov and Edward J. Rebar
} |
| | Olivier Toussaint, Véronique Royer, Michel Salmon and
925 Diversity of acetylation targets and roles in transcrip-
\ José Remacle
tional regulation: the human immunodeficiency virus
type 1 promoter as a model system 1011 Stress-induced premature senescence and replicative
senescence are different phenotypes, proteomic evi-
Vincent Quivy and Carine Van Lint
dence
S|
935 Oxidative stress, transcription factors and chromatin
Jean-Francois Dierick, Francois Eliaers, José Remacle,
remodelling in lung inflammation
Martine Raes, Stephen J. Fey, Peter Mose Larsen and
Irfan Rahman Olivier Toussaint
Contents of Volume 64
THIOLS, PROTEIN THIOLATION AND CELL SIGNALING 1111 Chemosensitization by fibroblast growth factor-2 is
not dependent upon proliferation, S-phase accumula-
1019 Cellular glutathione and thiols metabolism
tion, or p53 status
Dale A. Dickinson and Henry Jay Forman
Aaron B. Coleman, Marianne Z. Metz,
1027 Glutathione catabolism as a signaling mechanism Cécile A. Donohue, Roderich E. Schwarz and
Susan E. Kane
Aldo Paolicchi, Silvia Dominici, Lisa Pieri,
Emilia Maellaro and Alfonso Pompella 1125 Use of Chlamydomonas reinhardtii mutants for antic-
ancer drug screening
1037 Glutathione, iron and Parkinson’s disease
Karine Maucourt, Manjul Agarwal, Brigitte René and
Srinivas Bharath, Michael Hsu, Deepinder Kaur,
Serge Fermandjian
Subramanian Rajagopalan and Julie K. Andersen
1133 Effects of nitrosopropofol on mitochondrial energy-
1049 Glutathionylation of proteins by glutathione disulfide
converting system
S-oxide
Roberto Stevanato, Federico Momo, Michela Marian,
Kuo-Ping Huang and Freesia L. Huang
Maria Pia Rigobello, Alberto Bindoli,
1057 Cell signalling and the glutathione redox system Marcantonio Bragadin, Ezio Vincenti and Guido Scutari
Giuseppe Filomeni, Giuseppe Rotilio and 1139 Effect of free iron on collagen synthesis, cell prolif-
Maria Rosa Ciriolo eration and MMP-2 expression in rat hepatic stellate
cells
1065 Thioredoxins and related proteins in photosynthetic
organisms: molecular basis for thiol dependent regu- Concetta Gardi, Beatrice Arezzini, Vittoria Fortino and
lation Mario Comporti
Jean-Pierre Jacquot, Eric Gelhaye, Nicolas Rouhier,
Catherine Corbier, Claude Didierjean and André Aubry
(CHEMOTHERAPY AND METABOLIC INHIBITORS
1147 Regulation of anandamide tissue levels by N-arachi-
donylglycine
1 October 2002
Sumner H. Burstein, Susan M. Huang,
Timothy J. Petros, Ronald G. Rossetti,
J Michael Walker and Robert B. Zurier
Commentary
1071 A novel pathway regulating the mammalian target of 1151 Inhibition of cytochrome P450 2E1 by propofol in
rapamycin (mTOR) signaling human and porcine liver microsomes
Jie Chen and Yimin Fang Corinne Lejus, Alain Fautrel, Yannick Mallédant and
André Guillouzo
MOLECULAR AND CELLULAR PHARMACOLOGY
HORMONES AND GROWTH FACTORS
1079 Effects of FK228, a novel histone deacetylase inhibi-
1157 Contribution of different phospholipases and arachi-
tor, on human lymphoma U-937 cells in vitro and in
donic acid metabolites in the response of gallbladder
vivo
smooth muscle to cholecystokinin
Yuka Sasakawa, Yoshinori Naoe, Takeshi Inoue,
Soledad Alcon, Sara Morales, Pedro J. Camello and
Tatsuya Sasakawa, Masahiko Matsuo,
Maria J. Pozo
Toshitaka Manda and Seitaro Mutoh
SU9516, a cyclin-dependent kinase 2 inhibitor, pro-
INFLAMMATION AND IMMUNOPHARMACOLOGY
motes accumulation of high molecular weight E2F
complexes in human colon carcinoma cells 1169 Cyclic AMP differentially modulates CD40L expres-
sion on human naive and memory CD4" T cells
Bo Yu, Maureen E. Lane and Scott Wadler
Denise Wingett and Christopher P. Nielson
Complementary DNA cloning and characterization
of cytochrome P450 2D29 from Japanese monkey 1179 Biochemical and biological properties of phospholi-
liver pases A> from Bothrops atrox snake venom
Hiroyuki Hichiya, Chie Takemi, Daisuke Tsuzuki, Milton M. Kanashiro, Rita de Cdssia M. Escocard,
Shigeo Yamamoto, Kazuo Asaoka, Satoshi Suzuki, Jorge H. Petretski, Maura V. Prates, Elias W. Alves,
Tetsuo Satoh, Sumio Shinoda, Hiroyuki Kataoka Olga L.T. Machado, Wilmar Dias da Silva and
and Shizuo Narimatsu Thereza L. Kipnis
Contents of Volume 64 1803
1187 Role of mast cell chymase in allergen-induced bipha- 1251 Modulation of agonist responses at the A; adenosine
sic skin reaction receptor by an irreversible antagonist, receptor—G
protein uncoupling and by the G protein activation
Yoshiaki Tomimori, Nobuo Tsuruoka,
state
Harukazu Fukami, Kayo Saito, Chika Horikawa,
Masayuki Saito, Tsuyoshi Muto, Namino Sugiura, Anna Lorenzen, Margot W. Beukers,
Kyoko Yamashiro, Motoo Sumida, Saki Kakutani and Piet Hein van der Graaf, Heidrun Lang,
Yoshiaki Fukuda Jacqueline van Muijlwijk-Koezen, Miriam de Groote,
Wiro Menge, Ulrich Schwabe and Adriaan P. IJzerman
15 October 2002
CHEMOTHERAPY AND METABOLIC INHIBITORS
1267 The activity profile of the hexacyclic camptothecin
derivative DX-8951f in experimental human colon
Commentary
cancer and ovarian cancer
1195 Glutamate antagonists limit tumor growth
Annemarie H. van Hattum, Herbert M. Pinedo,
Wojciech Rzeski, Chrysanthy Ikonomidou and
Hennie M.M. Schliiper, Caroline A.M. Erkelens,
Lechoslaw Turski
Akiko Tohgo and Epie Boven
1279 Novel competitive irreversible inhibitors of aldehyde
MOLECULAR AND CELLULAR PHARMACOLOGY dehydrogenase (ALDH1): restoration of chemosensi-
tivity of L1210 cells overexpressing ALDH 1 and induc-
1201 Characterization of the cAMP binding site of purified
tion of apoptosis in BAF; cells overexpressing bel
S-adenosyl-homocysteine hydrolase from bovine kid-
Gerard Quash, Guy Fournet, Jacqueline Chantepie,
ney
Jacques Gore, Claude Ardiet, Dominique Ardail,
Doris Kloor, Lusine Danielyan and
Yvonne Michal and Uwe Reichert
Hartmut Osswald
1207 Antagonist interaction with endogenous AT, recep-
NEUROSCIENCE
tors in human cell lines
1293 Degradation of nociceptin (orphanin FQ) by mouse
Ilse Verheijen, Patrick M.L. Vanderheyden,
spinal cord synaptic membranes is triggered by endo-
Jean-Paul De Backer, Serge Bottari and
peptidase-24.11: an in vitro and in vivo study
Georges Vauquelin
Chikai Sakurada, Shinobu Sakurada, Tohru Orito,
1215 Contribution of apoptosis in the cytotoxicity of the
Koichi Tan-No and Tsukasa Sakurada
oxaliplatin—irinotecan combination in the HT29
human colon adenocarcinoma cell line
Stéphanie Arnould, Sylvie Guichard,
1 November 2002
Isabelle Hennebelle, Georges Cassar,
Roland Bugat and Pierre Canal
1227 Diverse functional coupling of cyclooxygenase 1 and Commentary
2 with final prostanoid synthases in liver macro- 1305 Role of the Fas/Fas ligand system in female reproduc-
phages tive organs: survival and apoptosis
Sabine Schade, Yevgeniya Bezugla, Angelika Kolada, Gil Mor, Shawn Straszewski and Marijke Kamsteeg
Sabine Kamionka, Roland Scheibe and Peter Dieter
1233 Potentiation of 1,25-dihydroxyvitamin D3-induced RAPID COMMUNICATION
differentiation of human promyelocytic leukemia
1317 Expression and purification of a recombinant form of
cells into monocytes by costunolide, a germacrano-
human aromatase from Escherichia coli
lide sesquiterpene lactone
Fangming Zhang, Dujin Zhou, Yeh-Chih Kao,
Seung H. Kim, So N. Kang, HyeoungJ . Kim and
Jinging Ye and Shiuan Chen
Tae S. Kim
1243 Comparative analysis of human and rat S1P5 (edg8):
differential expression profiles and sensitivities to MOLECULAR AND CELLULAR PHARMACOLOGY
antagonists 1325 Pro-apoptotic actions of exisulind and CP461 in
Anke Niedernberg, Constanze R. Scherer, SW480 colon tumor cells involve B-catenin and
Andreas E. Busch and Evi Kostenis cyclin D1 down-regulation
Contents of Volume 64
Han Li, Li Liu, Mary L. David, Clark M. Whitehead,
15 November 2002
Ming Chen, John R. Fetter, GerhardJ . Sperl,
Rifat Pamukcu and W. Joseph Thompson
1337 Evidence for the presence of glutamatergic receptors Commentary
in adult Schistosoma mansoni 1425 Endoplasmic reticulum (ER) stress: hepatitis C virus
Dayde Lane Mendonga-Silva, Renata Fittipaldi Pesséa induces an ER-nucleus signal transduction pathway
and Francois Noél and activates NF-KB and STAT-3
Gulam Waris, Keith D. Tardif and Aleem Siddiqui
1345 Inhibition of prostaglandin E) production by taiwa-
nin C isolated from the root of Acanthopanax chiisa-
nensis and the mechanism of action
MOLECULAR AND CELLULAR PHARMACOLOGY
Hyun Seung Ban, Sanghyun Lee, Yong Pil Kim,
Role of noradrenaline on the expression of the Na‘/
Kouya Yamaki, Kuk Hyun Shin and Kazuo Ohuchi
K*-ATPase 2 isoform and the contractility of cul-
1355 Predicting plasma protein binding of drugs: a new tured rat vas deferens
approach
Luis Eduardo M. Quintas, Simone S.L. Lafayette,
Nicole A. Kratochwil, Walter Huber, Francis Miiller, Afonso Caricati-Neto, Aron Jurkiewicz and
Manfred Kansy and Paul R. Gerber Francois Noel
1375 The antiproliferative activity of resveratrol results in 1439 5-Fluorouracil inhibits nitric oxide production
apoptosis in MCF-7 but not in MDA-MB-231 human through the inactivation of IkB kinase in stomach
breast cancer cells: cell-specific alteration of the cell cancer cells
cycle In Duk Jung, So Young Yang, Chang Gyo Park,
Kyung Bok Lee, Jong Seung Kim, Seok Yong Lee,
Eulalia Pozo-Guisado, Alberto Alvarez-Barrientos,
Sonia Mulero-Navarro, Belen Santiago-Josefat and Jeung Whan Han, Hyang Woo Lee and Hoi Young Lee
Pedro M. Fernandez-Salguero
1447 Molecular cloning and characterization of mouse
CYP2J6, an unstable cytochrome P450 isoform
1387 The molecular and enzyme kinetic basis for the
diminished activity of the cytochrome P450 2D6.17 Jixiang Ma, J. Alyce Bradbury, Lorraine King,
(CYP2D6.17) variant. Potential implications for Robert Maronpot, Linda S. Davis, Matthew D. Breyer
CYP2D6 phenotyping studies and the clinical use of and Darryl C. Zeldin
CYP2D6 substrate drugs in some African populations
Enhanced activity of human N-myristoyltransferase
Tashinga E. Bapiro, Julia A. Hasler,
by dimethyl sulfoxide and related solvents in the pre-
Marianne Ridderstrom and Collen M. Masimirembwa
sence of serine/threonine-containing peptide sub-
strates
(CHEMOTHERAPY AND METABOLIC INHIBITORS Mohammed Khysar Pasha, Jonathan R. Dimmock,
Morley D. Hollenberg and Rajendra K. Sharma
1399 Haem polymerase as a novel target of antimalarial
1469 UVB light suppresses nitric oxide production by mur-
action of cyproheptadine
ine keratinocytes and macrophages
Rashmi Agrawal, Renu Tripathi, Babu L. Tekwani,
S.K. Jain, Guru P. Dutta and Onkar P. Shukla Runa Sur, Diane E. Heck, Thomas M. Mariano,
Yang Jin, William J. Murphy and Jeffrey D. Laskin
1407 Enhanced activity of liposomal polymyxin B against
1483 Differential effect of simvastatin on activation of
Pseudomonas aeruginosa in a rat model of lung infec-
Rac; vs. activation of the heat shock protein 27-
tion
mediated pathway upon oxidative stress, in human
Abdelwahab Omvi, Zacharias E. Suntres and
smooth muscle cells
Pang N. Shek
Pascale Négre-Aminou, Rick E.W. van Leeuwen,
G. Christa F. van Thiel, Paul van den IJssel,
NEUROSCIENCE Wilfried W. de Jong, Roy A. Quinlan and
Louis H. Cohen
1415 Anxiolytic effect of wogonin, a benzodiazepine recep-
tor ligand isolated from Scutellaria baicalensis Georgi
(CHEMOTHERAPY AND METABOLIC INHIBITORS
Kwok Min Hui, Michael S.Y. Huen, Hong Yan Wang,
Hui Zheng, Erwin Sigel, Roland Baur, Hong Ren,
1493 Analytical and pharmacokinetic studies with 5-
Zhi Wang Li, J. Tze-Fei Wong and Hong Xue chloro-2'-deoxycytidine